Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 25, Issue 3 (2010)

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Journal of Enzyme Inhibition and Medicinal Chemistry, Volume 25, Issue 3 (2010)

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Research Article

Article
New insights into homopiperazine-based 5-HT1A/5-HT7R ligands: synthesis and biological evaluation
Eduard Badarau, Aurélien Putey, Franck Suzenet, Benoit Joseph, Andrzej Bojarski, Adriana Finaru & Gérald Guillaumet
Pages: 301-305
Published online: 29 Oct 2009
AbstractforNew insights into homopiperazine-based 5-HT1A/5-HT7R ligands: synthesis and biological evaluation | Full Text | References | PDF (913.5 KB)
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Article
Synthesis and biological activity of progesterone derivatives as 5α-reductase inhibitors, and their effect on hamster prostate weight
Eugene Bratoeff, Armando Zambrano, Ivonne Heuze, Anay Palacios, Daniela Ramírez & Marisa Cabeza
Pages: 306-311
Published online: 29 Oct 2009
AbstractforSynthesis and biological activity of progesterone derivatives as 5α-reductase inhibitors, and their effect on hamster prostate weight | Full Text | References | PDF (964 KB)
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Article
Evaluation of the antifungal and plasma membrane H+-ATPase inhibitory action of ebselen and two ebselen analogs in S. cerevisiae cultures
Blase Billack, Magdalena Piętka-Ottlik, Michelle Santoro, Stacia Nicholson, Jacek Młochowski & Cesar Lau-Cam
Pages: 312-317
Published online: 09 Mar 2010
AbstractforEvaluation of the antifungal and plasma membrane H+-ATPase inhibitory action of ebselen and two ebselen analogs in S. cerevisiae cultures | Full Text | References | PDF (794.4 KB)
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Article
Why acetylcholinesterase reactivators do not work in butyrylcholinesterase
Jiří Wiesner, Zdeněk Kříž, Kamil Kuča, Daniel Jun & Jaroslav Koča
Pages: 318-322
Published online: 29 Oct 2009
AbstractforWhy acetylcholinesterase reactivators do not work in butyrylcholinesterase | Full Text | References | PDF (1 MB)
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Article
3-Arylidene-5-(4-isobutylphenyl)-2(3H)-furanones: a new series of anti-inflammatory and analgesic compounds having antimicrobial activity
Mumtaz Mohammad Alam, Asif Husain, Syed M. Hasan, Suruchi Khanna & Mohammad Shaquiquzzaman
Pages: 323-330
Published online: 02 Nov 2009
Abstractfor3-Arylidene-5-(4-isobutylphenyl)-2(3H)-furanones: a new series of anti-inflammatory and analgesic compounds having antimicrobial activity | Full Text | References | PDF (695.6 KB)
  • 518 Views
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Article
Synthesis and biological evaluation of biguanide and dihydrotriazine derivatives as potential inhibitors of dihydrofolate reductase of opportunistic microorganisms
Seema Bag, Nilesh R. Tawari, Sherry F. Queener & Mariam S. Degani
Pages: 331-339
Published online: 29 Oct 2009
AbstractforSynthesis and biological evaluation of biguanide and dihydrotriazine derivatives as potential inhibitors of dihydrofolate reductase of opportunistic microorganisms | Full Text | References | PDF (755.9 KB)
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Article
Pharmacokinetic parameters and a theoretical study about metabolism of BR-AEA (a salbutamol derivative) in rabbit
Marvin Antonio Soriano-Ursúa, Jose Correa-Basurto, Juan Romero-Huerta, Octavio Elizalde-Solis, Luis Alejandro Galicia-Luna & Jose Guadalupe Trujillo-Ferrara
Pages: 340-346
Published online: 29 Oct 2009
AbstractforPharmacokinetic parameters and a theoretical study about metabolism of BR-AEA (a salbutamol derivative) in rabbit | Full Text | References | PDF (1 MB)
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Article
4-(4-Morpholinophenyl)-6-arylpyrimidin-2-amines: synthesis, spectral analysis, and in vitro microbiological evaluation
J. Thanusu, V. Kanagarajan & M. Gopalakrishnan
Pages: 347-353
Published online: 29 Oct 2009
Abstractfor4-(4-Morpholinophenyl)-6-arylpyrimidin-2-amines: synthesis, spectral analysis, and in vitro microbiological evaluation | Full Text | References | PDF (718.5 KB)
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Article
Exploring QSAR for CYP11B2 binding affinity and CYP11B2/CYP11B1 selectivity of diverse functional compounds using GFA and G/PLS techniques
Partha P. Roy & Kunal Roy
Pages: 354-369
Published online: 24 Dec 2009
AbstractforExploring QSAR for CYP11B2 binding affinity and CYP11B2/CYP11B1 selectivity of diverse functional compounds using GFA and G/PLS techniques | Full Text | References | PDF (879.1 KB)
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Article
Mechanistic studies on human N-acetylgalactosamine kinase
Andrew Agnew & David Timson
Pages: 370-376
Published online: 29 Oct 2009
AbstractforMechanistic studies on human N-acetylgalactosamine kinase | Full Text | References | PDF (871.2 KB)
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Article
Isolation and partial sequence of a Kunitz-type elastase specific inhibitor from marama bean (Tylosema esculentum)
Deepa Nadaraja, Susan T. Weintraub, Kevin W. Hakala, Nicholas E. Sherman & Barry Starcher
Pages: 377-382
Published online: 02 Nov 2009
AbstractforIsolation and partial sequence of a Kunitz-type elastase specific inhibitor from marama bean (Tylosema esculentum) | Full Text | References | PDF (877.7 KB)
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Article
Mechanochemical synthesis and in vitro anti-Helicobacter pylori and uresase inhibitory activities of novel zinc(II)–famotidine complex
Muhammad Amin, Mohammad S. Iqbal, Roy W. Hughes, Safyan A. Khan, Paul A. Reynolds, Virve I. Enne, Sajjad-ur-Rahman & Akmal S. Mirza
Pages: 383-390
Published online: 26 Oct 2009
AbstractforMechanochemical synthesis and in vitro anti-Helicobacter pylori and uresase inhibitory activities of novel zinc(II)–famotidine complex | Full Text | References | PDF (777.8 KB)
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Article
RETRACTED: Larvicidal effects of the major essential oil of Pittosporum tobira against Aedes aegypti (L.)
Ill-Min Chung, Su-Hyun Seo, Eun-Young Kang, Won-Hwan Park & Hyung-In Moon
Pages: 391-393
Published online: 29 Oct 2009
AbstractforRETRACTED: Larvicidal effects of the major essential oil of Pittosporum tobira against Aedes aegypti (L.) | Full Text | References | PDF (1.5 MB)
  • 1128 Views
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Article
Design, synthesis, cytotoxic evaluation, and QSAR study of some 6H-indolo[2,3-b]quinoxaline derivatives
N. S. Hari Narayana Moorthy, C. Karthikeyan & Piyush Trivedi
Pages: 394-405
Published online: 16 Mar 2010
AbstractforDesign, synthesis, cytotoxic evaluation, and QSAR study of some 6H-indolo[2,3-b]quinoxaline derivatives | Full Text | References | PDF (821.8 KB)
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Article
Isolation and identification of antioxidant and hyaluronidase inhibitory compounds from Ficus microcarpa L. fil. bark
Changwei Ao, Tatsunori Higa, Hui Ming, Yu-ting Ding & Shinkichi Tawata
Pages: 406-413
Published online: 16 Mar 2010
AbstractforIsolation and identification of antioxidant and hyaluronidase inhibitory compounds from Ficus microcarpa L. fil. bark | Full Text | References | PDF (949.1 KB)
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Article
Nostotrebin 6, a bis(cyclopentenedione) with cholinesterase inhibitory activity isolated from Nostoc sp. str. Lukešová 27/97
Petr Zelík, Alena Lukešová, Jan Čejka, Miloš Buděšínský, Vladimír Havlíček, Alexander Čegan & Jiří Kopecký
Pages: 414-420
Published online: 16 Mar 2010
AbstractforNostotrebin 6, a bis(cyclopentenedione) with cholinesterase inhibitory activity isolated from Nostoc sp. str. Lukešová 27/97 | Full Text | References | PDF (971.4 KB)
  • 842 Views
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Article
Binding conformations and QSAR of CA-4 analogs as tubulin inhibitors
Si Yan Liao, Jin Can Chen, Ti Fang Miao, Yong Shen & Kang Cheng Zheng
Pages: 421-429
Published online: 29 Oct 2009
AbstractforBinding conformations and QSAR of CA-4 analogs as tubulin inhibitors | Full Text | References | PDF (1.4 MB)
  • 557 Views
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Article
Synthesis, Physico-Chemical investigations of Co(II), Ni(II) and Cu(II) complexes and their in vitro microbial, cytotoxic, DNA cleavage studies
Gangadhar B. Bagihalli & Sangamesh A. Patil
Pages: 430-439
Published online: 07 Apr 2010
AbstractforSynthesis, Physico-Chemical investigations of Co(II), Ni(II) and Cu(II) complexes and their in vitro microbial, cytotoxic, DNA cleavage studies | Full Text | References | PDF (1 MB)
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Short Communications

Article
Conferin, potent antioxidant and anti-inflammatory isoflavone from Caragana conferta Benth
Amna Nisar Khan, Shagufta Perveen, Abdul Malik, Nighat Afza, Lubna Iqbal, Mehreen Latif & Muhammad Saleem
Pages: 440-444
Published online: 20 Apr 2010
AbstractforConferin, potent antioxidant and anti-inflammatory isoflavone from Caragana conferta Benth | Full Text | References | PDF (725 KB)
  • 514 Views
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Article
Template synthesis of macrocyclic complexes and their spectroscopic and antibacterial studies
D. P. Singh, Vidhi Grover, Ramesh Kumar & Kiran Jain
Pages: 445-449
Published online: 16 Nov 2009
AbstractforTemplate synthesis of macrocyclic complexes and their spectroscopic and antibacterial studies | Full Text | References | PDF (624 KB)
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