Search in:

Journal of Enzyme Inhibition and Medicinal Chemistry Volume 28, 2013 - Issue 5

Submit an article Journal homepage

Free access

675

Views

CrossRef citations to date

Altmetric

Research Article

Regioselective acylation of congeners of 3-amino-1H-pyrazolo[3,4-b]quinolines, their activity on bacterial serine/threonine protein kinases and in vitro antibacterial (including antimycobacterial) activity

Gennady B. LapaGause Institute of New Antibiotics, B. Pirogovskaya 11, Moscow, 119313, RussiaCorrespondence[email protected]

O. B. BekkerVavilov Institute of General Genetics, Gubkin St. 3, Moscow, 119991, Russia

E. P. MirchinkGause Institute of New Antibiotics, B. Pirogovskaya 11, Moscow, 119313, Russia

V. N. DanilenkoVavilov Institute of General Genetics, Gubkin St. 3, Moscow, 119991, Russia

M. N. PreobrazhenskayaGause Institute of New Antibiotics, B. Pirogovskaya 11, Moscow, 119313, Russia

Pages 1088-1093 | Received 02 Apr 2012, Accepted 24 Jul 2012, Published online: 07 Sep 2012

Cite this article
https://doi.org/10.3109/14756366.2012.716056

Full Article
Figures & data
References
Citations
Metrics
Reprints & Permissions
View PDF PDF

Citations (13)

Keep up to date with the latest research on this topic with citation updates for this article.

Subscribe to citation updates

Articles from other publishers (13)

G. B. Lapa, P. Gruber, G. Untergasser, N. I. Moiseeva & J. Hofmann. (2023) New Biological Evaluation of Thienoquinolines as Disruptors of the PKCε/RACK2 Protein–Protein Interaction. Moscow University Chemistry Bulletin 77:S1, pages S46-S54.
Crossref

Pethaperumal Iniyavan, Anusha Avadhani, Yogendra Kumar, Arkalagud Satyanarayana Jeevan Chakravarthy, Mary Antony Palluruthiyil & Hiriyakkanavar Ila. (2022) Synthesis of novel 9‐amino /aryl/oxo‐2‐(het)arylthiazolo[4,5‐ b ]quinolines via palladium catalyzed N ‐arylation ‐cyclization protocol . Journal of Heterocyclic Chemistry.
Crossref

Andrzej Danel, Ewa Gondek, Mateusz Kucharek, Paweł Szlachcic & Arkadiusz Gut. (2022) 1H-Pyrazolo[3,4-b]quinolines: Synthesis and Properties over 100 Years of Research. Molecules 27:9, pages 2775.
Crossref

Ana Donaire-Arias, Ana Maria Montagut, Raimon Puig de la Bellacasa, Roger Estrada-Tejedor, Jordi Teixidó & José I. Borrell. (2022) 1H-Pyrazolo[3,4-b]pyridines: Synthesis and Biomedical Applications. Molecules 27:7, pages 2237.
Crossref

Ashley King & Meghan S. Blackledge. (2021) Evaluation of small molecule kinase inhibitors as novel antimicrobial and antibiofilm agents. Chemical Biology & Drug Design 98:6, pages 1038-1064.
Crossref

Vrushabendra Basavanna, Srikantamurthy Ningaiah, Manasa Chandramouli, Anjali Sobha & Shridevi Doddamani. (2021) Quinolinyl-pyrazoles: synthesis and pharmacological evolution in the recent decennial. Journal of the Iranian Chemical Society 18:7, pages 1479-1522.
Crossref

Fátima C. Teixeira, Carla Lucas, M. João M. Curto, Vânia André, M. Teresa Duarte & António P. S. Teixeira. (2021) Synthesis of novel pyrazolo[3,4- b ]quinolinebisphosphonic acids and an unexpected intramolecular cyclization and phosphonylation reaction . Organic & Biomolecular Chemistry 19:11, pages 2533-2545.
Crossref

Niccolò Cantini, Andrei I. Khlebnikov, Letizia Crocetti, Igor A. Schepetkin, Giuseppe Floresta, Gabriella Guerrini, Claudia Vergelli, Gianluca Bartolucci, Mark T. Quinn & Maria Paola Giovannoni. (2021) Exploration of nitrogen heterocycle scaffolds for the development of potent human neutrophil elastase inhibitors. Bioorganic & Medicinal Chemistry 29, pages 115836.
Crossref

Elisabeth Bou-Petit, Arnau Plans, Nieves Rodríguez-Picazo, Antoni Torres-Coll, Cristina Puigjaner, Mercè Font-Bardia, Jordi Teixidó, Santiago Ramon y Cajal, Roger Estrada-Tejedor & José I. Borrell. (2020) C4–C5 fused pyrazol-3-amines: when the degree of unsaturation and electronic characteristics of the fused ring controls regioselectivity in Ullmann and acylation reactions. Organic & Biomolecular Chemistry 18:27, pages 5145-5156.
Crossref

Puay-Wah Phuan, Joseph-Anthony Tan, Amber A. Rivera, Lorna Zlock, Dennis W. Nielson, Walter E. Finkbeiner, Peter M. Haggie & Alan S. Verkman. (2019) Nanomolar-potency ‘co-potentiator’ therapy for cystic fibrosis caused by a defined subset of minimal function CFTR mutants. Scientific Reports 9:1.
Crossref

Chandrabose Karthikeyan, Haneen Amawi, Arabela Guedes Viana, Leticia Sanglard, Noor Hussein, Maria Saddler, Charles R. AshbyJr.Jr., N.S. Hari Narayana Moorthy, Piyush Trivedi & Amit K. Tiwari. (2018) lH-Pyrazolo[3,4-b]quinolin-3-amine derivatives inhibit growth of colon cancer cells via apoptosis and sub G1 cell cycle arrest. Bioorganic & Medicinal Chemistry Letters 28:13, pages 2244-2249.
Crossref

Zhi Xu, Chuan Gao, Qing-Cheng Ren, Xu-Feng Song, Lian-Shun Feng & Zao-Sheng Lv. (2017) Recent advances of pyrazole-containing derivatives as anti-tubercular agents. European Journal of Medicinal Chemistry 139, pages 429-440.
Crossref

V. N. Maksimova, A. I. Naidenova, O. V. Ershov, O. E. Nasakin & V. A. Tafeenko. (2017) Synthesis of 3-aminopyrazolo[3,4-b]pyridine-4-carbonitriles. Russian Journal of Organic Chemistry 52:12, pages 1830-1834.
Crossref

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Order Reprints Request Corporate Permissions

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

Request Academic Permissions

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.

Share icon
Back to Top

Related research

People also read lists articles that other readers of this article have read.

Recommended articles lists articles that we recommend and is powered by our AI driven recommendation engine.

Cited by lists all citing articles based on Crossref citations.
Articles with the Crossref icon will open in a new tab.

People also read
Recommended articles
Cited by

To cite this article:

Reference style: APA Chicago Harvard

Citation copied to clipboard

Reference styles above use APA (6th edition), Chicago (16th edition) & Harvard (10th edition)

Download citation

Download a citation file in RIS format that can be imported by citation management software including EndNote, ProCite, RefWorks and Reference Manager.

Choose format: RIS BibTex RefWorks Direct Export

Choose options: Citation Citation & abstract Citation & references

Regioselective acylation of congeners of 3-amino-1H-pyrazolo[3,4-b]quinolines, their activity on bacterial serine/threonine protein kinases and in vitro antibacterial (including antimycobacterial) activity

Articles from other publishers (13)

Information for

Open access

Opportunities

Help and information

Your download is now in progress and you may close this window

Login or register to access this feature

Regioselective acylation of congeners of 3-amino-1H-pyrazolo[3,4-b]quinolines, their activity on bacterial serine/threonine protein kinases and in vitro antibacterial (including antimycobacterial) activity

Citations (13)

Articles from other publishers (13)

Reprints and Corporate Permissions

Academic Permissions

Related research

To cite this article:

Download citation

Information for

Open access

Opportunities

Help and information

Keep up to date