153
Views
22
CrossRef citations to date
0
Altmetric
Research Article

Development and in-vitro evaluation of modified release tablets including ethylcellulose microspheres loaded with diltiazem hydrochloride

, &
Pages 135-152 | Received 28 Apr 2005, Accepted 20 Jun 2005, Published online: 08 Oct 2008

References

  • Amperiadou A, Georgarakis M. Controlled release salbutamol sulphate microcapsules prepared by emulsion solvent-evaporation technique and study on the release affected parameters. International Journal of Pharmaceutics 1995; 115: 1–8
  • Bayomi MA, Al-Suwayeh SA, El-heiw AM, Mesnad AF. Preparation of casein-chitosan microspheres containing diltiazem hydrochloride by an aqueous coacervation technique. Pharmaceutica Acta Helvetiae 1998; 73: 187–192
  • Bhalerao SS, Lalla JK, Rane MS. Study of processing parameters influencing the properties of diltiazem hydrochloride microspheres. Journal of Microencapsulation 2001; 18: 299–307
  • BP. Appendix XII G. Uniformity of weight (mass). Pharmacopoeia Commision, LondonBritish 2000; 1
  • Çelik M. Compaction of multiparticulate oral dosage forms. Multiparticulate oral drug delivery, I Ghebre-Sellassie. Marcel Dekker Inc, New York 1994; 181–215
  • Chiao CSL, Price JC. Formulation, preparation and dissolution characteristics of propranolol hydrochloride microspheres. Journal of Microencapsulation 1994; 11: 153–159
  • Çomoğlu T, Gönül N, Baykara T. The effects of pressure and direct compression on tabletting of microsponges. International Journal of Pharmaceutics 2002; 242: 191–195
  • Das SK, Das NG. Preparation and in vitro dissolution profile of dual polymer (Eudragit®RS100 and RL100) microparticles of diltiazem hydrochloride. Journal of Microencapsulation 1998; 15: 445–452
  • Hasçiçek C, Gönül N, Erk N. Mucoadhesive microspheres containing gentamicin sulfate for nasal administration: Preparation and in vitro characterization. Il Farmaco 2003; 58: 11–16
  • Horoz BB, Kılıçarslan M, Yüksel N, Baykara T. Effect of different dispersing agents on the characteristics of Eudragit microspheres prepared by a solvent evaporation method. Journal of Microencapsulation 2004; 21: 191–202
  • Huang H, Ghebre-Sellassie I. Preparation of microspheres of water-soluble pharmaceuticals. Journal of Microencapsulation 1989; 6: 219–225
  • Kakish HF, Tashtoush B, Ibrahim HG, Najib NM. A novel approach for the preparation of highly loaded polymeric controlled release dosage forms of diltiazem HCl and diclofenac sodium. European Journal of Pharmaceutics and Biopharmaceutics 2002; 54: 75–81
  • Kawata M, Nakamura M, Goto S, Aoyama T. Preparation and dissolution pattern of Eudragit RS microcapsules containing ketoprofen. Chemical & Pharmaceutical Bulletin 1986; 34: 2618–2623
  • Kelly JG, O’Malley K. Clinical pharmacokinetics of calcium antagonists: An update. Clinical Pharmacokinetics 1992; 22: 416–433
  • Kim CK, Kim MJ, Oh KH. Preparation and evaluation of sustained release microspheres of terbutaline sulfate. International Journal of Pharmaceutics 1994; 106: 213–219
  • Kollidon®SR Technical Information [Internet]. Basf Ag: Fine Chemicals: Pharma Solutions: Excipients, 2001 July [cited 2004 July 20]; Available online at: http://www.pharma-solutions.basf.com (20 July 2004)
  • Kristmundsdóttir T, Gudmundsson Ó S, Ingvarsdóttir K. Release of diltiazem from Eudragit microparticles prepared by spray-drying. International Journal of Pharmaceutics 1996; 137: 159–165
  • Kristmundsdóttir T, Ingvarsdóttir K. Influence of emulsifying agents on the properties of cellulose acetate butyrate and ethylcellulose microcapsules. Journal of Microencapsulation 1994; 11: 633–639
  • Mateovic T, Kriznar B, Bogataj M, Mrhar A. The influence of stirring rate on biopharmaceutical properties of Eudragit RS microspheres. Journal of Microencapsulation 2002; 19: 29–36
  • Oates JA, Brown NJ. Antihypertensive agents and the drug therapy of hypertension. Goodman & Gilman's the pharmacological basis of therapeutics.10th, AG Gilman. Pergamon, New York 2001; 871–893
  • Obaidat AA, Obaidat RM. Controlled release of tramadol hydrochloride from matrices prepared using glyceryl behenate. European Journal of Pharmaceutics and Biopharmaceutics 2001; 52: 231–235
  • Pather SI, Russell I, Syce JA, Neau SH. Sustained release theophylline tablets by direct compression part 1: Formulation and in vitro testing. International Journal of Pharmaceutics 1998; 164: 1–10
  • Robinson JR, Li VHK, Lee VHL. Influence of drug properties and routes of drug administration on the design of sustained and controlled release systems. Controlled drug delivery fundamentals and applications.2nd, JR Robinson, VHL Lee. Marcel Dekker Inc., New York 1987; 4–94
  • Sood A, Pachagnula R. Drug release evaluation of diltiazem CR preparations. International Journal of Pharmaceutics 1998; 175: 95–107
  • Soppimath KS, Kulkarni AR, Aminabhavi TM. Encapsulation of antihypertensive drugs in cellulose-based matrix microspheres: Characterization and release kinetics of microspheres and tableted microspheres. Journal of Microencapsulation 2001; 18: 397–409
  • Sreenivasa Rao B, Ramana Murthy KV. Studies on rifampicin release from ethylcellulose coated nonpareil beads. International Journal of Pharmaceutics 2002; 231: 97–106
  • Sveinsson SJ, Kristmundsdóttir T, Ingvarsdóttir K. The effect of tableting on the release characteristics of naproxen and ibuprofen microcapsules. International Journal of Pharmaceutics 1993; 92: 29–34
  • Tirkkonen S, Paronen P. Release of indomethacin from tabletted ethylcellulose microcapsules. International Journal of Pharmaceutics 1993; 92: 55–62
  • USP XXIV/NF XIX. United States of Pharmacopoeia Convention Inc., RockvilleUSA 2000; 2149–2152
  • Vilivalam VD, Adeyeye CM. Development and evaluation of controlled-release diclofenac microspheres and tabletted microspheres. Journal of Microencapsulation 1994; 11: 455–470

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.