257
Views
9
CrossRef citations to date
0
Altmetric
Research Articles

Development of galangal essential oil-based microemulsion gel for transdermal delivery of flurbiprofen: simultaneous permeability evaluation of flurbiprofen and 1,8-cineole

, , , , , , & show all
Pages 91-100 | Received 19 Sep 2019, Accepted 14 Dec 2019, Published online: 08 Jan 2020

References

  • Richy F, Rabenda V, Mawet A, et al. Flurbiprofen in the symptomatic management of rheumatoid arthritis: a valuable alternative. Int J Clin Pract. 2007;61(8):1396–1406.
  • Jamali Dr F, Collins DS, Berry BW, et al. Comparative bioavailability of two flurbiprofen products: stereospecific versus conventional approach. Biopharm Drug Dispos. 1991;12(6):435–445.
  • Han F, Yin R, Shi XL, et al. Cloud point extraction-HPLC method for determination and pharmacokinetics study of flurbiprofen in rat plasma after oral and transdermal administration. J. Chromatogr. B. 2008;868(1-2):64–69.
  • Trommer HH, Neuber R. Overcoming the stratum corneum: the modulation of skin penetration. Skin Pharmacol Physiol. 2006;19(2):106–121.
  • Parhi R, Suresh P, Mondal S, et al. Novel penetration enhancers for skin applications: a review. CDD. 2012;9(2):219–230.
  • Herman A, Herman AP. Essential oils and their constituents as skin penetration enhancer for transdermal drug delivery: a review. J Pharm Pharmacol. 2015;67(4):473–485.
  • Zhang LC, Hu JH, Li L, et al. In vivo and in vitro evaluation of essential oils from Ligusticum chuanxiong HORT on the transdermal delivery of flurbiprofen in rabbits. Biol Pharm Bull. 2006;29(6):1217–1222.
  • Charoo NA, Shamsher AA, Kohli K, et al. Improvement in bioavailability of transdermally applied flurbiprofen using tulsi (Ocimum sanctum) and turpentine oil. Colloid Surfaces B. 2008;65(2):300–307.
  • Van Zyl L, Du Preez J, Gerber M, et al. Essential fatty acids as transdermal penetration enhancers. J. Pharm. Sci. 2016;105(1):188–193.
  • Abubakar IB, Malami I, Yahaya Y, et al. A review on the ethnomedicinal uses, phytochemistry and pharmacology of Alpinia officinarum Hance. J. Ethnopharmacol. 2018;224:45–62.
  • Podshivalov AV, Bronnikov S, Zuev VV, et al. Synthesis and characterization of polyurethane-urea microcapsules containing galangal essential oil: statistical analysis of encapsulation. J. Microencapsul. 2013;30(2):198–203.
  • Yao JH, Jiang QD, Cai H, et al. Cytotoxicity and penetration enhancement activity of essential oils from warming the interior medicinals with hot or warm property in terms of Traditional Chinese Medicine. J Tradit Chin Med. 2018;38(2):257–265.
  • Chen J, Jiang QD, Chai YP, et al. Natural terpenes as penetration enhancers for transdermal drug delivery. Molecules. 2016;21(12):1709.
  • Shukla T, Upmanyu N, Agrawal M, et al. Biomedical applications of microemulsion through dermal and transdermal route. Biomed Pharmacother. 2018;108:1477–1494.
  • Mishra R, Prabhavalkar KS, Bhatt LK. Preparation, optimization, and evaluation of Zaltoprofen-loaded microemulsion and microemulsion-based gel for transdermal delivery. J. Liposome Res. 2016;26(4):297–306.
  • Said M, Elsayed I, Aboelwafa AA, et al. Transdermal agomelatine microemulsion gel: pyramidal screening, statistical optimization and in vivo bioavaiablity. Drug Deliv. 2017;24(1):1159–1169.
  • Catanzano O, Straccia MC, Miro A, et al. Spray-by-spray in situ cross-linking alginate hydrogels delivering a tea tree oil microemulsion. Eur J Pharm. 2015;66:20–28.
  • Liu C-H, Chang F-Y, Hung D-K. Terpene microemulsions for transdermal curcumin delivery: Effects of terpenes and cosurfactants. Colloids Surf B Biointerfaces. 2011;82(1):63–70.
  • Ahad A, Aqil M, Ali A. Investigation of antihypertensive activity of carbopol valsartan transdermal gel containing 1,8-cinecole. Int J Biol Macromol. 2014;64:144–149.
  • Jiang Q, Wu Y, Zhang H, et al. Development of essential oils as skin permeation enhancers: penetration enhancement effect and mechanism of action. Pharm Biol. 2017;55(1):1592–1600.
  • Zhu XM, Li Y, Xu F, et al. Skin electrical resistance measurement of oxygen-containing terpenes as penetration enhancers: role of stratum corneum lipids. Molecules. 2019;24(3):523.
  • Zhang J, Michniak-Kohn BB. Investigation of microemulsion and microemulsion gel formulations for dermal delivery of clotrimazole. Int J Pharm. 2018;536(1):345–352.
  • Ch.Liu X, Quan P, Li SS, et al. Time dependence of the enhancement effect of chemical enhancers:Molecular mechanisms of enhancing kinetics. J Control Release. 2017;248:33–44.
  • Amin S, Kohli K, Khar RK, et al. Mechanism of in vitro percutaneous absorption enhancement of carvedilol by penetration enhancers. Pharm Dev Technol. 2008;13(6):533–539.
  • Shen Q, Li WJ, Li WY. The effect of clove oil on the transdermal delivery of ibuprofen in the rabbit by in vitro and in vivo methods. Drug Dev Ind Pharm. 2007;33(12):1369–1374.
  • Shen T, Xu H, Weng W, et al. Development of a reservoir-type transdermal delivery system containing eucalyptus oil for tetramethylpyrazine. Drug Deliv. 2013;20(1):19–24.
  • Das MK, Bhattacharya A, Ghosal SK. Effect of different terpene-containing essential oils on percutaneous absorption of trazodone hydrochloride through mouse epidermis. Drug Deliv. 2006;13(6):425–431.
  • Valgimigli L, Gabbanini S, Berlini E, et al. Lemon (Citrus limon, Burm.f.) essential oil enhances the trans-epidermal release of lipid- (A,E) and water- (B6, C) soluble vitamins from topical emulsions in reconstructed human epidermis. Int J Cosmet Sci. 2012;34(4):347–356.
  • Akbari J, Saeedi M, Farzin D, et al. Transdermal absorption enhancing effect of the essential oil of Rosmarinus officinalis on percutaneous absorption of Na diclofenac from topical gel. Pharm Biol. 2015;53(10):1442–1447.
  • Lan Y, Chen Y, Zhang Y, et al. Essential oil from Zanthoxylum bungeanum Maxim. and its main components used as transdermal penetration enhancers: a comparative study. J Zhejiang Univ Sci B. 2014;15(11):940–952.
  • Monti D, Chetoni P, Burgalassi S, et al. Effect of different terpene-containing essential oils on permeation of estradiol through hairless mouse skin. Int J Pharm. 2002;237(1-2):209–214.
  • Danielsson I, Lindman B. The definition of microemulsion. Colloids Surf. 1981;3(4):391–392.
  • Linghu KG, Wu GP, Fu LY, et al. 1,8-Cineole ameliorates LPS-induced vascular endothelium dysfunction in mice via PPAR-γ dependent regulation of NF-ĸB. Front Pharmacol. 2019;10:178.
  • Santos FA, Silva RM, Campos AR, et al. 1,8-Cineole (eucalyptol), a monoterpene oxide attenuates the colonic damage in rats on actue TNBS-colitis. Food Chem Toxicol. 2004;42(4):579–584.
  • Liapi C, Anifantis G, Chinou I, et al. Antinociceptive properties of 1,8-cineole and beta-pinene, from the essential oil of Eucalyptus camaldulensis leaves, in rodents. Planta Med. 2007;73(12):1247–1254.
  • Jiang F, Wu G, Li W, et al. Preparation and protective effects of 1,8-cineole-loaded self-microemulsifying drug delivery system on lipopolysaccharide-induced endothelial injury in mice. Eur J Pharm Sci. 2019;127:14–23.
  • Alam P, Alqasoumi SI, Abdel-Kader MS. Simultaneous determination of menthol and eucalyptol by the densitometric HPTCL method in some external analgesic formulations. J Chromatogr Sci. 2016;54(1):58–63.

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.