Mechanism of In Vitro Percutaneous Absorption Enhancement of Carvedilol by Penetration Enhancers

REFERENCES

• R Langer. (2004). Transdermal drug discovery: past progress, current status, and future prospects. Adv. Drug Deliver. Rev. 56 (5):556–557.
   Web of Science ®Google Scholar
• IH Blank. (1964). Penetration of low molecular weight alcohols into skin – the effect of concentration of alcohol and type of vehicle. J. Invest. Dermatol. 43:415–420.
   PubMedGoogle Scholar
• J Hadgraft. (1996). Recent developments in topical and transdermal delivery. Eur. J . Drug Metab. Pharmacokinet. 21:165–173.
   PubMed Web of Science ®Google Scholar
• J Hadgraft. (1999). Passive enhancement strategies in topical and transdermal drug delivery. Int. J. Pharm. 184:1–6.
   PubMed Web of Science ®Google Scholar
• RH Guy. (1998). Iontophoresis: Recent developments. J. Pharm. Pharmcol. 50 (4):371–374.
   PubMed Web of Science ®Google Scholar
• S Mitragotri, D Blankschtein, and R Langer. (1996). Transdermal drug delivery using low frequency sonophoresis. Pharm. Res. 13 (3):411–420.
   PubMed Web of Science ®Google Scholar
• M Mollgard. Synergistic effects in percutaneous enhancementPharmaceutical Skin Penetration EnhancementKA Walters, and J Hadgraft. Marcel Dekker, New York, (1993) 229–242.
   Google Scholar
• K Sugibayashi, S Nakayama, T Seki, K Hosoyak, and Y Morimoto. (1992). Mechanism of skin permeation enhancing effect by laurocapram. J. Pharm. Sci. 81:58–64.
   PubMed Web of Science ®Google Scholar
• K Zhao, and J Singh. (2000). Mechanism(s) of in-vitro percutaneous absorption enhancement of tamoxifen by enhancers. J. Pharm. Sci. 89 (6):771–780.
   PubMed Web of Science ®Google Scholar
• BJ Aungst, JA Blake, NJ Rogers, and MA Husain. (1990). Transdermal oxymorphone formulation development and methods for evaluating flux, lag times for two skin permeation enhancing vehicles. J. Pharm. Sci. 79:1072–1076.
   PubMed Web of Science ®Google Scholar
• GA Burdock. Encyclopedia of Food and Color Additives. CRC Press, Baco RatonFL, (1997) 230–231461–462. 1051–1054..
   Google Scholar
• CY Goates, and K Knutson. Enhanced permeation of polar compounds through human epidermis. I. Permeability and membrane structural change in the presence of short chain alcoholsBiochim. Biophys. Acta. , , (1994) 1195169–179.
   Google Scholar
• H Tanojo, JA Bouwstra, HE Junginger, and HE Bodd. Subzero thermal analysis of human stratum corneumPharm. Res. , , (1994) 111610–1616.
   Google Scholar
• F Dreher, P Walde, P Walther, and E Wehrli. (1997). Interaction of a lecithin microemulsion gel with human stratum corneum and its effect on transdermal port. J. Control. Rel. 45:131–140.
   Web of Science ®Google Scholar
• M Goodman, and BW Barry. Action of penetration enhancer on human stratum corneum as assessed by differential scanning calorimetryPercutaneous AbsorptionRL Bronaugh, and HL Maibach. Marcel Dekker, New York and Basel, (1989) 567–593.
   Google Scholar
• SC Shin, EY Shin, and CW Cho. (2000). Enhancing effects of fatty acids on piroxicam permeation through rat skins. Drug. Dev. Ind. Pharm. 26 (5):563–566.
   PubMed Web of Science ®Google Scholar
• C Dollery. Therapeutic drugs. Vol. 1. Churchill Livingstone, Edinburg, (1999) 76–81.
   Google Scholar
• MNA Chisty, RA Bellantone, DR Taft, and FM Plakogiannis. In-vitro evaluation of the release of albuterol sulfate from polymer gels: effect of fatty acids on drug transport across biological membranesDrug Dev. Ind. Pharm. , , (2002) 281221–1229.
   Google Scholar
• G Chaurasia, D Bhadra, S Bhadra, and NK Jain. (2005). UV spectrophotometric determination of carvedilol. Indian J. Pharm. Sci. 67 (5):606–608.
   Google Scholar
• HK Vaddi, PC Ho, and SY Chan. (2002). Terpenes in propylene glycol as skin extraction enhancers: permeation and partition of haloperidol, fourier transform infrared spectroscopy and differential scanning calorimetry. J. Pharm. Sci. 91 (7):1639–1651.
   PubMed Web of Science ®Google Scholar
• B Bergh, JA Bouwstra, HE Junginger, and PW Wertz. (1999). Elasticity of vesicles affect hairless mouse skin structure and permeability. J. Control. Rel. 62 (3):367–379.
   PubMed Web of Science ®Google Scholar
• G Kantarc, I Ozguney, HY Karasulu, T Guneri, and G Basdemir. (2005). In-vitro permeation of diclofenac sodium from novel microemulsion formulations through rabbit skin. Drug Dev. Res. 65 (1):17–25.
   Web of Science ®Google Scholar
• GM Golden, DB Guzek, RR Harris, JE McKie, and RO Potts. (1986). Lipid thermotropic transition in human stratum corneum. J. Invest. Dermatol. 86:255–269.
   PubMed Web of Science ®Google Scholar
• GM Golden, JE McKie, and RO Potts. (1987). Role of stratum corneum lipid fluidity in transdermal drug flux. J. Pharm. Sci. 76:25–28.
   PubMed Web of Science ®Google Scholar
• AM Knutson, RO Potts, DB Guzek, GM Golden, JE McKie, WJ Lambert, and WI Higuchi. (1985). Macromolecular physical-chemical considerations in understanding the stratum corneum. J. Control. Rel. 2:67–87.
   Google Scholar
• CS Leopold, and BC Lippold. (1995). An attempt to clarify the mechanism of the penetration enhancing effects of lipophilic vehicles with differential scanning calorimetry (DSC). J. Pharm. Pharmacol. 47:276–281.
   PubMed Web of Science ®Google Scholar
• DB Bommannan, RO Potts, and RH Guy. (1991). Examination of the effect of ethanol on human stratum corneum in vivo using infrared spectroscopy. J. Control. Rel. 16:299–304.
   Web of Science ®Google Scholar
• K Bhatia, and J Singh. Mechanism of transport enhancement of LHRH through porcine epidermis by terpenes and iontophoresis: permeability and lipid extraction studiesPharm. Res. , , (1998) 151857–1862.
   Google Scholar
• DJ Moore, and ME Rerek. Insight into the molecular organization of lipids in the skin barrier from infrared spectroscopy studies of SC lipids modelsActa Dermatol. , , (2000) 20816–22.
   Google Scholar
• K Moser, K Kriwet, A Naik, YN Kalia, and RH Guy. Passive skin penetration enhancement and its quantification in vitroEur. J. Pharm. Biopharm. , , (2001) 52103–112.
   Google Scholar
• S Yum, E Lee, L Taskovic, and F Theeuwes. Permeation enhancement with ethanol: mechanism of action through skinDrug Permeation EnhancementDS Hsich. Marcel Dekker, New York, (1994) 143–170.
   Google Scholar
• A Sintov, A Zeevi, R Uzan, and A Nyska. Influence of pharmaceutical gel vehicles containing oleic acid/ sodium oleate combinations on hairless mouse skin, a histological evaluationEur. J. Pharm. Biopharm. , , (1999) 47299–303.
   Google Scholar