Development of Controlled-Release Buccoadhesive Hydrophilic Matrices of Diltiazem Hydrochloride: Optimization of Bioadhesion, Dissolution, and Diffusion Parameters

REFERENCES

• McElnay J.C. Buccal Absorption of Drugs. Encyclopedia of Pharmaceutical Technology, J. Swarbrick, J.C. Boylan. Marcel Dekker, New York 1990; Vol. 2: 189–211
   Google Scholar
• Rathbone M.J., Drummond B.K., Tucker I.G. The Oral Cavity as a Site for Systemic Drug Delivery. Adv. Drug Del. Rev. 1994; 13: 1–22
   Web of Science ®Google Scholar
• Chidambaram N., Srivatsava A.K. Buccal Drug Delivery Systems. Drug Dev. Ind. Pharm. 1995; 21(9)1009–1036
   Web of Science ®Google Scholar
• Khanna R., Agarwal S.P., Ahuja A. Mucoadhesive Buccal Drug Delivery: A Potential Alternative to Conventional Therapy. Indian J. Pharm. Sci. 1998; 60(1)1–11
   Google Scholar
• Mazzo D.J., Obetz C.L., Shuster J. Diltiazem Hydrochloride. Analytical Profiles of Drug Substances and Excipients, H.G. Brittain. Academic Press, San Diego, CA 1994; Vol. 23: 53–98
   Google Scholar
• Buckley M.M.-T., Grant S.M., Goa K.L., McTavish D., Sorkin E.M. Diltiazem: A Reappraisal of Its Pharmacological Properties and Therapeutic Use. Drugs 1990; 39(5)757–806
   PubMed Web of Science ®Google Scholar
• Vatsraj N.B., Zia H., Needham T. (2000) Formulation and Optimization of a Sustained Release Tablet of Ketorolac Tromethamine. Proceedings of International Symposium on Controlled Release of Bioactive Materials, Paris, July, 7–132000. Controlled Release Society, Paris, 8444
   Google Scholar
• Gohel M.C., Amin A.F. Formulation Design and Optimization of Modified-Release Microsphere of Diclofenac Sodium. Drug Dev. Ind. Pharm. 1999; 25(2)247–251
   PubMed Web of Science ®Google Scholar
• Doornbos D.A., Haan P. Optimization Techniques in Formulation and Processing. Encyclopedia of Pharmaceutical Technology, J. Swarbrick, J.C. Boylan. Marcel Dekker, New York 1995; Vol. 11: 77–160
   Google Scholar
• Lewis G.A., Mathieu D., Phan-Tan-Luu R. Pharmaceutical Experimental Design. Drugs and Pharmaceutical Sciences. Marcel Dekker, New York 1999; Vol. 92, (Singh,B. Ahuja,N. Book Review on Pharmaceutical Experimental Design, Int. J. Pharm. 2000, 195, 247–248)
   Google Scholar
• Bolton S. Optimization Techniques. Pharmaceutical Statistics: Practical and Clinical Applications, 2nd Ed. Marcel Dekker, New York 1990; 532–570
   Google Scholar
• Kettaneh-Wold N. Use of Experimental Design in the Pharmaceutical Industry. J. Pharm. Biomed. Anal. 1991; 9(8)605–610
   PubMed Web of Science ®Google Scholar
• Gupta A., Garg S., Khar R.K. Measurement of Bioadhesive Strength of Mucoadhesive Buccal Tablets: Design of an In Vitro Assembly. Indian Drugs 1993; 30(4)152–155
   Google Scholar
• Singh B., Singh S.A. Comprehensive Computer Program for the Study of Drug Release Kinetics from Compressed Matrices. Indian J. Pharm. Sci. 1998; 60(6)358–362
   Google Scholar
• Singh B., Kaur T., Singh S. Correction of Raw Dissolution Data for Loss of Drug and Volume During Sampling. Indian J. Pharm. Sci. 1997; 59: 196–199
   Google Scholar
• Korsmeyer R.W., Gurny R., Doelker E., Buri P., Peppas N.A. Mechanisms of Solute Release from Porous Hydrophilic Polymers. Int. J. Pharm. 1983; 15: 25–35
   Web of Science ®Google Scholar
• Zhang H., Robinson J.R. In Vitro Methods for Measuring Permeability of the Oral Mucosa. Oral Mucosal Drug Delivery, M.J. Rathbone. Drugs and The Pharmaceutical Sciences; Marcel Dekker, New York 1996; Vol. 74: 85–100
   Google Scholar
• Singh B., Gupta R.K. (1996) FACTOP: A Software Aid to Optimize Pharmaceutical Dosage Forms Through Factorial Design. 48th Indian Pharmaceutical Congress, ChennaiIndia, Dec, 26–291996. Indian Pharmaceutical Congress Association, MumbaiIndia, 42, AP 63
   Google Scholar
• Box G.E.P., Connor L.R., Cousins W.R., Davies O.L., Himsworth F.R., Sillitto G.P. The Design and Analysis of Industrial Experiments, 2nd Ed., O.L. Davies. Oliver and Boyd, London 1960
   Google Scholar
• Bolton S. Factorial Designs. Pharmaceutical Statistics: Practical and Clinical Applications, 2nd Ed. Marcel Dekker, New York 1990; 308–337
   Google Scholar
• Ahuja A., Dogra M., Agarwal S.P. Development of Buccal Tablets of Diltiazem Hydrochloride. Indian J. Pharm. Sci. 1995; 57(1)26–30
   Google Scholar
• Saisivam S., Muhammed Ashereff M.H., Maria Gerald N.S., Rajan, Jayaprakash S., Nagarajan M. Design and Evaluation of Diltiazem Hydrochloride Buccal Patches. Indian J. Pharm. Sci. 2000; 62(3)236–238
   Google Scholar
• Han R.-Y., Fang J.-Y., Sung K.C., Hu O.Y.P. Mucoadhesive Buccal Disks for Novel Nalbuphine Prodrug Controlled Delivery: Effect of Formulation Variables on Drug Release and Mucoadhesive Performance. Int. J. Pharm. 1999; 177: 201–209
   PubMed Web of Science ®Google Scholar
• Guo J.-H. Bioadhesive Polymer Buccal Patches for Buprenorphine Controlled Delivery: Formulation, In Vitro Adhesion and Release Properties. Drug Dev. Ind. Pharm. 1994; 20(18)2809–2821
   Web of Science ®Google Scholar
• Peppas N.A., Sahlin J.J. A Simple Equation for the Description of Solute Release. III. Coupling of Diffusion and Relaxation. Int. J. Pharm. 1989; 57: 169–172
   Web of Science ®Google Scholar