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Original Research

Promising Swellable Floating Bupropion Tablets: Formulation, in vitro/in vivo Evaluation and Comparative Pharmacokinetic Study in Human Volunteers

ORCID Icon, ORCID Icon, , &
Pages 2741-2757 | Published online: 14 Jul 2020

References

  • PlodkowskiRA, NguyenQ, SundaramU, NguyenL, ChauDL, St JeorS. Bupropion and naltrexone: a review of their use individually and in combination for the treatment of obesity. Exp Opinion Pharmacother. 2009;10(6):1069–1081.
  • LayekB, MandalS. Natural polysaccharides for controlled delivery of oral therapeutics: a recent update. Carbohydr Polym. 2020;230:115617. doi:10.1016/j.carbpol.2019.11561731887888
  • Abd El-AzizMF, IsmailS, TadrosMI, ElnabarawiMA. Alfuzosin hydrochloride-loaded low-density gastroretentive sponges: development, in vitro characterization and gastroretentive monitoring in healthy volunteers via MRI. Pharm Dev Technol. 2020;1–13.
  • LinH-L, ChenL-C, ChengW-T, ChengW-J, HoH-O, SheuM-T. Preparation and characterization of a novel swellable and floating gastroretentive drug delivery system (sfGRDDS) for enhanced oral bioavailability of nilotinib. Pharmaceutics. 2020;12(2):137. doi:10.3390/pharmaceutics12020137
  • ChoiriS, SulaimanTS, RohmanA. Assessment of the effect of polymers combination and effervescent component on the drug release of swellable gastro-floating tablet formulation through compartmental modeling-based approach. 2020 Drug Dev Ind Pharm. 1–30. just-accepted.
  • RossiA, ContiC, ColomboG, et al. Floating modular drug delivery systems with buoyancy independent of release mechanisms to sustain amoxicillin and clarithromycin intra-gastric concentrations. Drug Dev Ind Pharm. 2016;42(2):332–339. doi:10.3109/03639045.2015.105439726065531
  • JayasreeJ, SivaneswariS, HemalathaG, PreethiN, MounikaB, MurthySV. Role of various natural, synthetic and semi-synthetic polymers on drug release kinetics of losartan potassium oral controlled release tablets. Int J Pharm Investig. 2014;4(4):183. doi:10.4103/2230-973X.143118
  • LewisGA, MathieuD, Phan-Tan-LuuR. Pharmaceutical Experimental Design. New York, USA: CRC press; 1998.
  • NjorogeGG, SimbauniJA, KoskeJA. An optimal split plot design for performing a mixture process experiment. Sci J Appl Mathematics Stat. 2017;5:15–23. doi:10.11648/j.sjams.20170501.13
  • JonesB, GoosP. I-optimal versus D-optimal split-plot response surface designs. J Qual Technol. 2012;44(2):85–101. doi:10.1080/00224065.2012.11917886
  • ChappidiSR, BhargavE, MarikunteV, et al. A cost effective (QbD) approach in the development and optimization of rosiglitazone maleate mucoadhesive extended release tablets in vitro and ex vivo. Adv Pharm Bulletin. 2019;9(2):281. doi:10.15171/apb.2019.032
  • USP.35. Convention USP. United States Pharmacopeia;2011:35
  • JiJ, HeX, YangX-L, et al. The in vitro/vivo evaluation of prepared gastric floating tablets of berberine hydrochloride. AAPS Pharm Sci Tech. 2017;18(6):2149–2156. doi:10.1208/s12249-016-0696-7
  • El NabarawiMA, TeaimaMH, RaaE-M, El NabarawyNA, GaberDA. Formulation, release characteristics, and bioavailability study of gastroretentive floating matrix tablet and floating raft system of mebeverine HCl. Drug Des Devel Ther. 2017;11:1081. doi:10.2147/DDDT.S131936
  • YeomDW, SongYS, KimSR, et al. Development and optimization of a self-microemulsifying drug delivery system for ator vastatin calcium by using D-optimal mixture design. Int J Nanomedicine. 2015;10:3865.26089663
  • DashS, MurthyPN, NathL, ChowdhuryP. Kinetic modeling on drug release from controlled drug delivery systems. Acta Pol Pharm. 2010;67(3):217–223.20524422
  • ZhangY, HuoM, ZhouJ, et al. DDSolver: an add-in program for modeling and comparison of drug dissolution profiles. AAPS J. 2010;12(3):263–271. doi:10.1208/s12248-010-9185-120373062
  • RazaA, ShenN, LiJ, ChenY, WangJ-Y. Formulation of zein based compression coated floating tablets for enhanced gastric retention and tunable drug release. Eur J Pharm Sci. 2019;132:163–173. doi:10.1016/j.ejps.2019.01.02530695689
  • ZhangY, HuoM, ZhouJ, XieS. PKSolver: an add-in program for pharmacokinetic and pharmacodynamic data analysis in microsoft excel. Computer Methods Programs Biomed. 2010;99(3):306–314.
  • RazaviM, KarimianH, YeongCH, et al. Gastroretentive behavior of orally administered radiolabeled tamarind seed formulations in rabbits validated by gamma scintigraphy. Drug Des Devel Ther. 2017;11:1. doi:10.2147/DDDT.S115466
  • AllenL, AnselHC. Ansel’s Pharmaceutical Dosage Forms and Drug Delivery Systems. Lippincott Williams & Wilkins; 2013.
  • ChenY-C, HoH-O, LeeT-Y, SheuM-T. Physical characterizations and sustained release profiling of gastroretentive drug delivery systems with improved floating and swelling capabilities. Int J Pharm. 2013;441(12):162–169. doi:10.1016/j.ijpharm.2012.12.00223237874
  • MostafaviA, EmamiJ, VarshosazJ, DaviesNM, RezazadehM. Development of a prolonged-release gastroretentive tablet formulation of ciprofloxacin hydrochloride: pharmacokinetic characterization in healthy human volunteers. Int J Pharm. 2011;409(12):128–136. doi:10.1016/j.ijpharm.2011.02.03521371548
  • SahuA, VermaA, SinghS. Preparation of hydrophilic swelling controlled-release floating matrix tablets containing HPMC and chitosan. Int J Pharm Pharm Sci. 2012;4(1):406–411.
  • ViridénA, WittgrenB, LarssonA. Investigation of critical polymer properties for polymer release and swelling of HPMC matrix tablets. Eur j Pharm Sci. 2009;36(23):297–309. doi:10.1016/j.ejps.2008.10.02119038336
  • AiT, ShangL, HeC, et al. Development of multi-layered gastric floating tablets based on konjac glucomannan: a modified calcium supplement with enhanced bioavailability. Food Funct. 2019;10(10):6429–6437. doi:10.1039/C9FO01107B31517352
  • QiX, ChenH, RuiY, YangF, MaN, WuZ. Floating tablets for controlled release of ofloxacin via compression coating of hydroxypropyl cellulose combined with effervescent agent. Int J Pharm. 2015;489(12):210–217. doi:10.1016/j.ijpharm.2015.05.00725956047
  • RazaviM, NyamathullaS, KarimianH, NoordinMI. Novel swellable polymer of orchidaceae family for gastroretentive drug delivery of famotidine. Drug Des Devel Ther. 2014;8:1315. doi:10.2147/DDDT.S68517
  • RathiM, MedhekarR, PawarA, YewaleC, GudsoorkarV. Floating and bioadhesive delivery system of metoprolol succinate: formulation, development and in vitro evaluation. Asian J Pharm. 2014;6:3.
  • AburahmaMH, MahmoudAA. Biodegradable ocular inserts for sustained delivery of brimonidine tartrate: preparation and in vitro/in vivo evaluation. Aaps Pharmscitech. 2011;12(4):1335–1347. doi:10.1208/s12249-011-9701-321979886
  • EspositoE, MenegattiE, CortesiR. Hyaluronan-based microspheres as tools for drug delivery: a comparative study. Int J Pharm. 2005;288(1):35–49. doi:10.1016/j.ijpharm.2004.09.00115607256
  • KerdsakundeeN, MahattanadulS, WiwattanapatapeeR. Development and evaluation of gastroretentive raft forming systems incorporating curcumin-Eudragit® EPO solid dispersions for gastric ulcer treatment. Eur J Pharm Biopharm. 2015;94:513–520. doi:10.1016/j.ejpb.2015.06.02426143367
  • RazaviM, KarimianH, YeongCH, et al. Gamma scintigraphic study of the hydrodynamically balanced matrix tablets of metformin HCl in rabbits. Drug Des Devel Ther. 2015;9:3125. doi:10.2147/DDDT.S82935
  • AliA, IqbalM, AkhtarN, et al. Assessment of xanthan gum based sustained release matrix tablets containing highly water-soluble propranolol HCl. Acta Pol Pharm. 2013;70(2):283–289.23614284
  • RazaviM, KarimianH, YeongCH, ChungLY, NyamathullaS, NoordinMI. Gamma scintigraphic evaluation of floating gastroretentive tablets of metformin HCl using a combination of three natural polymers in rabbits. Drug Des Devel Ther. 2015;9:4373. doi:10.2147/DDDT.S86263
  • JainAK, SöderlindE, ViridénA, et al. The influence of hydroxypropyl methylcellulose (HPMC) molecular weight, concentration and effect of food on in vivo erosion behavior of HPMC matrix tablets. J Controlled Release. 2014;187:50–58. doi:10.1016/j.jconrel.2014.04.058
  • AlsarraIA, El-BagoryI, BayomiMA. Chitosan and sodium sulfate as excipients in the preparation of prolonged release theophylline tablets. Drug Dev Ind Pharm. 2005;31(45):385–395. doi:10.1080/0363904050021456316093204
  • LopesCM, BettencourtC, RossiA, ButtiniF, BarataP. Overview on gastroretentive drug delivery systems for improving drug bioavailability. Int J Pharm. 2016;510(1):144–158. doi:10.1016/j.ijpharm.2016.05.01627173823
  • ZhangC, YangF-Q. Konjac glucomannan, a promising polysaccharide for OCDDS. Carbohydr Polym. 2014;104:175–181. doi:10.1016/j.carbpol.2013.12.08124607175
  • YusifRM, HashimIIA, MohamedEA, BadriaFA-E. Gastrftableoretentive matrix tablets of boswellia oleogum resin: preparation, optimization, in vitro evaluation, and cytoprotective effect on indomethacin-induced gastric ulcer in rabbits. Aaps Pharmscitech. 2016;17(2):328–338. doi:10.1208/s12249-015-0351-826092303
  • MissaghiS, FegelyKA, Rajabi-SiahboomiAR. Investigation of the effects of hydroalcoholic solutions on textural and rheological properties of various controlled release grades of hypromellose. AAPS PharmSciTech. 2009;10(1):77–80. doi:10.1208/s12249-008-9181-219148758
  • PhaechamudT, DarunkaisornW. Drug release behavior of polymeric matrix filled in capsule. Saudi Pharm J. 2016;24(6):627–634. doi:10.1016/j.jsps.2015.04.00327829804
  • McPhillipsH, CraigD, RoyallP, HillV. Characterisation of the glass transition of HPMC using modulated temperature differential scanning calorimetry. Int J Pharm. 1999;180(1):83–90. doi:10.1016/S0378-5173(98)00407-410089295
  • KimJS, ChaKH, KangSY, et al. In vivo gastric residence and gastroprotective effect of floating gastroretentive tablet of DA-9601, an extract of Artemisia asiatica, in beagle dogs. Drug Des Devel Ther. 2016;10:1917.