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Review

Update on the clinical utility and practical use of ropivacaine in Chinese patients

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Pages 1269-1276 | Published online: 09 Sep 2014

References

  • McClellan KJ Faulds D Ropivacaine: an update of its use in regional anaesthesia Drugs 2000 60 1065 1093 11129123
  • Wong JO Tan TD Leung PO Tseng KF Cheu NW Spinal anesthesia with two different dosages of 0.75% glucose-free ropivacaine: a comparison of efficacy and safety in Chinese parturients undergoing cesarean section Acta Anaesthesiol Sin 2003 41 131 138 14601199
  • imshealth.com [homepage on the internet] China Hospital Pharmaceutical Audit (IMSHealth) Available from: http://www.imshealth.com/portal/site/imshealth Accessed August 13, 2014
  • Buckenmaier CC3rd Bleckner LL Anaesthetic agents for advanced regional anaesthesia: a North American perspective Drugs 2005 65 745 759 15819588
  • Schug SA Saunders D Kurowski I Paech MJ Neuraxial drug administration: a review of treatment options for anaesthesia and analgesia CNS Drugs 2006 20 917 933 17044729
  • Kindler CH Paul M Zou H Amide local anesthetics potently inhibit the human tandem pore domain background K+ channel TASK-2 (KCNK5) J Pharmacol Exp Ther 2003 306 84 92 12660311
  • Hansen TG Ropivacaine: a pharmacological review Expert Rev Neurother 2004 4 781 791 15853505
  • Rosenberg PH Heinonen E Differential sensitivity of A and C nerve fibres to long-acting amide local anaesthetics Br J Anaesth 1983 55 163 167 6830678
  • Benhamou D Ghosh C Mercier FJ A randomized sequential allocation study to determine the minimum effective analgesic concentration of levobupivacaine and ropivacaine in patients receiving epidural analgesia for labor Anesthesiology 2003 99 1383 1386 14639153
  • Camorcia M Capogna G Columb MO Minimum local analgesic doses of ropivacaine, levobupivacaine, and bupivacaine for intrathecal labor analgesia Anesthesiology 2005 102 646 650 15731605
  • Lee YY Ngan Kee WD Fong SY Liu JT Gin T The median effective dose of bupivacaine, levobupivacaine, and ropivacaine after intrathecal injection in lower limb surgery Anesth Analg 2009 109 1331 1334 19762766
  • Simpson D Curran MP Oldfield V Keating GM Ropivacaine: a review of its use in regional anaesthesia and acute pain management Drugs 2005 65 2675 2717 16392884
  • McGlade DP Kalpokas MV Mooney PH Comparison of 0.5% ropivacaine and 0.5% bupivacaine in lumbar epidural anaesthesia for lower limb orthopaedic surgery Anaesth Intensive Care 1997 25 262 266 9209608
  • Lee BB Ngan Kee WD Plummer JL Karmakar MK Wong AS The effect of the addition of epinephrine on early systemic absorption of epidural ropivacaine in humans Anesth Analg 2002 95 1402 1407 12401633
  • Lee BB Ngan Kee WD Wong EL Liu JY Dose-response study of epidural ropivacaine for labor analgesia Anesthesiology 2001 94 767 772 11388526
  • Karmakar MK Ho AM Law BK Wong AS Shafer SL Gin T Arterial and venous pharmacokinetics of ropivacaine with and without epinephrine after thoracic paravertebral block Anesthesiology 2005 103 704 711 16192762
  • Chen S Chen Z Jin Y Pharmacokinetics and efficacy of ropivacaine in Chinese patients following intra-articular administration Int J Clin Pharmacol Ther 2013 51 393 400 23458229
  • Karmakar MK Aun CS Wong EL Wong AS Chan SK Yeung CK Ropivacaine undergoes slower systemic absorption from the caudal epidural space in children than bupivacaine Anesth Analg 2002 94 259 265 11812681
  • Kitayama M Wada M Hashimoto H Kudo T Yakoshi C Hirota K Plasma ropivacaine concentrations after ultrasound-guided transversus abdominis plane block for open retropubic prostatectomy J Anesth Epub 12 18 2013
  • Emanuelsson BM Persson J Alm C Heller A Gustafsson LL Systemic absorption and block after epidural injection of ropivacaine in healthy volunteers Anesthesiology 1997 87 1309 1317 9416714
  • Simon MJ Veering BT Vletter AA Stienstra R van Kleef JW Burm AG The effect of age on the systemic absorption and systemic disposition of ropivacaine after epidural administration Anesth Analg 2006 102 276 282 16368843
  • Burm AG Stienstra R Brouwer RP Emanuelsson BM van Kleef JW Epidural infusion of ropivacaine for postoperative analgesia after major orthopedic surgery: pharmacokinetic evaluation Anesthesiology 2000 93 395 403 10910488
  • Ekström G Gunnarsson UB Ropivacaine, a new amide-type local anesthetic agent, is metabolized by cytochromes P450 1A and 3A in human liver microsomes Drug Metab Dispos 1996 24 955 961 8886604
  • Tucker GT Pharmacokinetics of local anaesthetics Br J Anaesth 1986 58 717 731 3524638
  • Whiteside JB Wildsmith JA Developments in local anaesthetic drugs Br J Anaesth 2001 87 27 35 11460810
  • Halldin MM Bredberg E Angelin B Metabolism and excretion of ropivacaine in humans Drug Metab Dispos 1996 24 962 968 8886605
  • Li M Cai HW Ren F Chen JH Sun B Epidural anesthesia with ropivacaine by computerized infusion pump Zhong Nan Da Xue Xue Bao Yi Xue Ban 2007 32 351 354 Chinese 17478952
  • Liu J Jiang Y Pang D Xi H Liu Y Li W Associations between single-nucleotide polymorphisms and epidural ropivacaine consumption in patients undergoing breast cancer surgery Genet Test Mol Biomarkers 2013 17 489 493 23577780
  • Wang G Sun Y Luo GJ Lin PC Liu PQ Effect of perioperative continuous epidural morphine administration on plasma D-dimer in patients undergoing total hip replacement Nan Fang Yi Ke Da Xue Xue Bao 2006 26 523 525 Chinese 16624773
  • Cai J Guo QL Zou WY Clinical anesthetic effects of epidural ropivacaine with tramadol Zhong Nan Da Xue Xue Bao Yi Xue Ban 2004 29 218 220 Chinese 16145920
  • Wan XH Huang QQ Su MX Wan LJ Huang HQ Security evaluation of bupivacaine, ropivacaine combined with fentanyl in postoperative continuous epidural analgesia Zhonghua Wai Ke Za Zhi 2006 44 1200 1202 Chinese 17147867
  • Crosby E Sandler A Finucane B Comparison of epidural anaesthesia with ropivacaine 0.5% and bupivacaine 0.5% for caesarean section Can J Anaesth 1998 45 1066 1071 10021954
  • Bjornestad E Smedvig JP Bjerkreim T Narverud G Kollerøs D Bergheim R Epidural ropivacaine 7.5 mg/mL for elective Caesarean section: a double-blind comparison of efficacy and tolerability with bupivacaine 5 mg/mL Acta Anaesthesiol Scand 1999 43 603 608 10408812
  • Kampe S Tausch B Paul M Epidural block with ropivacaine and bupivacaine for elective caesarean section: maternal cardiovascular parameters, comfort and neonatal well-being Curr Med Res Opin 2004 20 7 12 14741065
  • Hillyard SG Bate TE Corcoran TB Paech MJ O’Sullivan G Extending epidural analgesia for emergency Caesarean section: a meta-analysis Br J Anaesth 2011 107 668 678 21997149
  • Pouzeratte Y Delay JM Brunat G Patient-controlled epidural analgesia after abdominal surgery: ropivacaine versus bupivacaine Anesth Analg 2001 93 1587 1592 11726450
  • Casati A Santorsola R Aldegheri G Intraoperative epidural anesthesia and postoperative analgesia with levobupivacaine for major orthopedic surgery: a double-blind, randomized comparison of racemic bupivacaine and ropivacaine J Clin Anesth 2003 15 126 131 12719052
  • Leone S Di Cianni S Casati A Fanelli G Pharmacology, toxicology, and clinical use of new long acting local anesthetics, ropivacaine and levobupivacaine Acta Biomed 2008 79 92 105 18788503
  • Geng ZY Wang DX Wu XM Minimum effective local anesthetic dose of intrathecal hyperbaric ropivacaine and bupivacaine for cesarean section Chin Med J (Engl) 2011 124 509 513 21362272
  • Chen XZ Chen H Lou AF Lü CC Dose-response study of spinal hyperbaric ropivacaine for cesarean section J Zhejiang Univ Sci B 2006 7 992 997 17111469
  • Lee YY Ngan Kee WD Muchhal K Chan CK Randomized double-blind comparison of ropivacaine-fentanyl and bupivacaine-fentanyl for spinal anaesthesia for urological surgery Acta Anaesthesiol Scand 2005 49 1477 1482 16223393
  • Lee YY Ngan Kee WD Chang HK So CL Gin T Spinal ropivacaine for lower limb surgery: a dose response study Anesth Analg 2007 105 520 523 17646516
  • Gautier PE De Kock M Van Steenberge A Intrathecal ropivacaine for ambulatory surgery Anesthesiology 1999 91 1239 1245 10551572
  • McDonald SB Liu SS Kopacz DJ Stephenson CA Hyperbaric spinal ropivacaine: a comparison to bupivacaine in volunteers Anesthesiology 1999 90 971 977 10201665
  • Malinovsky JM Charles F Kick O Intrathecal anesthesia: ropivacaine versus bupivacaine Anesth Analg 2000 91 1457 1460 11094000
  • Camorcia M Capogna G Berritta C Columb MO The relative potencies for motor block after intrathecal ropivacaine, levobupivacaine, and bupivacaine Anesth Analg 2007 104 904 907 17377104
  • McNamee DA McClelland AM Scott S Milligan KR Westman L Gustafsson U Spinal anaesthesia: comparison of plain ropivacaine 5 mg mL(−1) with bupivacaine 5 mg mL(−1) for major orthopaedic surgery Br J Anaesth 2002 89 702 706 12393766
  • Whiteside JB Burke D Wildsmith JA Comparison of ropivacaine 0.5% (in glucose 5%) with bupivacaine 0.5% (in glucose 8%) for spinal anaesthesia for elective surgery Br J Anaesth 2003 90 304 308 12594141
  • Cappelleri G Aldegheri G Danelli G Spinal anesthesia with hyperbaric levobupivacaine and ropivacaine for outpatient knee arthroscopy: a prospective, randomized, double-blind study Anesth Analg 2005 101 77 82 15976210
  • Khaw KS Ngan Kee WD Wong EL Liu JY Chung R Spinal ropivacaine for cesarean section: a dose-finding study Anesthesiology 2001 95 1346 1350 11748390
  • Khaw KS Ngan Kee WD Wong M Ng F Lee A Spinal ropivacaine for cesarean delivery: a comparison of hyperbaric and plain solutions Anesth Analg 2002 94 680 685 11867397
  • Liisanantti O Luukkonen J Rosenberg PH High-dose bupivacaine, levobupivacaine and ropivacaine in axillary brachial plexus block Acta Anaesthesiol Scand 2004 48 601 606 15101856
  • Altintas F Gumus F Kaya G Interscalene brachial plexus block with bupivacaine and ropivacaine in patients with chronic renal failure: diaphragmatic excursion and pulmonary function changes Anesth Analg 2005 100 1166 1171 15781539
  • Beaulieu P Babin D Hemmerling T The pharmacodynamics of ropivacaine and bupivacaine in combined sciatic and femoral nerve blocks for total knee arthroplasty Anesth Analg 2006 103 768 774 16931694
  • Casati A Borghi B Fanelli G Interscalene brachial plexus anesthesia and analgesia for open shoulder surgery: a randomized, double-blinded comparison between levobupivacaine and ropivacaine Anesth Analg 2003 96 253 259 12505962
  • Casati A Borghi B Fanelli G A double-blinded, randomized comparison of either 0.5% levobupivacaine or 0.5% ropivacaine for sciatic nerve block Anesth Analg 2002 94 987 990 11916809
  • Palmisani S Arcioni R Di Benedetto P De Blasi RA Mercieri M Ronconi P Ropivacaine and levobupivacaine for bilateral selective ankle block in patients undergoing hallux valgus repair Acta Anaesthesiol Scand 2008 52 841 844 18477086
  • Casati A Vinciguerra F Cappelleri G Levobupivacaine 0.2% or 0.125% for continuous sciatic nerve block: a prospective, randomized, double-blind comparison with 0.2% ropivacaine Anesth Analg 2004 99 919 923 15333432
  • Di Donato A Fontana C Lancia F Celleno D Efficacy and comparison of 0.5% levobupivacaine with 0.75% ropivacaine for peribulbar anaesthesia in cataract surgery Eur J Anaesthesiol 2006 23 487 490 16507188
  • Olmez G Cakmak SS Caca I Unlu MK Intraocular pressure and quality of blockade in peribulbar anesthesia using ropivacaine or lidocaine with adrenaline: a double-blind randomized study Tohoku J Exp Med 2004 204 203 208 15502419
  • Belyamani L Kriet M Laktaoui A Peribulbar anesthesia: comparing 1% ropivacaine and a mixture of 0.5% bupivacaine – 2% lidocaine J Fr Ophtalmol 2003 26 953 956 French 14631279
  • Borazan M Karalezli A Oto S Algan C Aydin Akova Y Comparison of a bupivacaine 0.5% and lidocaine 2% mixture with levobupivacaine 0.75% and ropivacaine 1% in peribulbar anaesthesia for cataract surgery with phacoemulsification Acta Ophthalmol Scand 2007 85 844 847 17662095
  • Cline E Franz D Polley RD Maye J Burkard J Pellegrini J Analgesia and effectiveness of levobupivacaine compared with ropivacaine in patients undergoing an axillary brachial plexus block AANA J 2004 72 339 345 15529729
  • Mageswaran R Choy YC Comparison of 0.5% ropivacaine and 0.5% levobupivacaine for infraclavicular brachial plexus block Med J Malaysia 2010 65 300 303 21901950
  • Borgeat A Kalberer F Jacob H Ruetsch YA Gerber C Patient-controlled interscalene analgesia with ropivacaine 0.2% versus bupivacaine 0.15% after major open shoulder surgery: the effects on hand motor function Anesth Analg 2001 92 218 223 11133631
  • Borghi B Facchini F Agnoletti V Pain relief and motor function during continuous interscalene analgesia after open shoulder surgery: a prospective, randomized, double-blind comparison between levobupivacaine 0.25%, and ropivacaine 0.25% or 0.4% Eur J Anaesthesiol 2006 23 1005 1009 16824239
  • Borgeat A Aguirre J Marquardt M Mrdjen J Blumenthal S Continuous interscalene analgesia with ropivacaine 0.2% versus ropivacaine 0.3% after open rotator cuff repair: the effects on postoperative analgesia and motor function Anesth Analg 2010 111 1543 1547 20889941
  • Liu SS Richman JM Thirlby RC Wu CL Efficacy of continuous wound catheters delivering local anesthetic for postoperative analgesia: a quantitative and qualitative systematic review of randomized controlled trials J Am Coll Surg 2006 203 914 932 17116561
  • Liu YY Yeh CN Lee HL Local anesthesia with ropivacaine for patients undergoing laparoscopic cholecystectomy World J Gastroenterol 2009 15 2376 2380 19452582
  • Chan SK Lai PB Li PT The analgesic efficacy of continuous wound instillation with ropivacaine after open hepatic surgery Anaesthesia 2010 65 1180 1186 20958277
  • Liu HL Ma CH Zhang XQ Yang Y Song XL Guo XY Combined efficacy of parecoxib and incisional ropivacaine infiltration on pain management after diagnostic hysteroscopy and laparoscopy Beijing Da Xue Xue Bao 2013 45 901 905 Chinese 24343071
  • Mulroy MF Burgess FW Emanuelsson BM Ropivacaine 0.25% and 0.5%, but not 0.125%, provide effective wound infiltration analgesia after outpatient hernia repair, but with sustained plasma drug levels Reg Anesth Pain Med 1999 24 2 136 141 10204899
  • Pettersson N Berggren P Larsson M Westman B Hahn RG Pain relief by wound infiltration with bupivacaine or high-dose ropivacaine after inguinal hernia repair Reg Anesth Pain Med 1999 24 569 575 10588564
  • Manfè AZ Marchesini M Bortolato A Feltracco P Lumachi F Ropivacaine versus levobupivacaine for minor breast surgery in outpatients: inversion of postoperative pain relief efficacy In Vivo 2012 26 1075 1077 23160696
  • Marret E Gentili M Bonnet MP Bonnet F Intra-articular ropivacaine 0.75% and bupivacaine 0.50% for analgesia after arthroscopic knee surgery: a randomized prospective study Arthroscopy 2005 21 313 316 15756185
  • Ngan Kee WD Ng FF Khaw KS Lee A Gin T Determination and comparison of graded dose-response curves for epidural bupivacaine and ropivacaine for analgesia in laboring nulliparous women Anesthesiology 2010 113 445 453 20613484
  • Chan L Lee BB Ngan Kee WD A randomised double-blinded controlled trial of the effect of diluent volume on the efficacy of a single dose of epidural ropivacaine for labour analgesia Int J Obstet Anesth 2006 15 201 205 16798444
  • Lee BB Ngan Kee WD Ng FF Lau TK Wong EL Epidural infusions of ropivacaine and bupivacaine for labor analgesia: a randomized, double-blind study of obstetric outcome Anesth Analg 2004 98 1145 1152 15041615
  • Beilin Y Guinn NR Bernstein HH Zahn J Hossain S Bodian CA Local anesthetics and mode of delivery: bupivacaine versus ropivacaine versus levobupivacaine Anesth Analg 2007 105 756 763 17717236
  • Bang EC Lee HS Kang YI Cho KS Kim SY Park H Onset of labor epidural analgesia with ropivacaine and a varying dose of fentanyl: a randomized controlled trial Int J Obstet Anesth 2012 21 45 50 22153132
  • Werdehausen R Fazeli S Braun S Apoptosis induction by different local anaesthetics in a neuroblastoma cell line Br J Anaesth 2009 103 711 718 19700777
  • Yamashita A Matsumoto M Matsumoto S Itoh M Kawai K Sakabe T A comparison of the neurotoxic effects on the spinal cord of tetracaine, lidocaine, bupivacaine, and ropivacaine administered intrathecally in rabbits Anesth Analg 2003 97 512 519 12873946
  • Takenami T Wang G Nara Y Intrathecally administered ropivacaine is less neurotoxic than procaine, bupivacaine, and levobupivacaine in a rat spinal model Can J Anaesth 2012 59 456 465 22383086
  • Arlock P Actions of three local anaesthetics: lidocaine, bupivacaine and ropivacaine on guinea pig papillary muscle sodium channels (Vmax) Pharmacol Toxicol 1988 63 96 104 2847132
  • Knudsen K Beckman Suurküla M Blomberg S Sjövall J Edvardsson N Central nervous and cardiovascular effects of iv infusions of ropivacaine, bupivacaine and placebo in volunteers Br J Anaesth 1997 78 507 514 9175963
  • Scott DB Lee A Fagan D Bowler GM Bloomfield P Lundh R Acute toxicity of ropivacaine compared with that of bupivacaine Anesth Analg 1989 69 563 569 2679230
  • Markham A Faulds D Ropivacaine. A review of its pharmacology and therapeutic use in regional anaesthesia Drugs 1996 52 429 449 8875132
  • Naropin® (ropivacaine HCl) injection; prescribing information (Canada) AstraZeneca Available from: http://www.astrazeneca.ca/cs/BlobServer?blobcol=pdffile&blobheader=application%2F-pdf&blobheadername1=Content-Disposition&blobheadername2=MDT-Type&blobheadervalue1=inline%3B+filename%3DProduct-Monograph.pdf&blobheadervalue2=abinary%3B+charset%3DUTF-8&blobkey=id&blobnocache=true&blobtable=AZ_FixedURLPDF&blobwhere=1285585474170&ssbinary=true Accessed August 28, 2014
  • Wong JO Tan TD Leung PO Tseng KF Cheu NW Tang CS Comparison of the effect of two different doses of 0.75% glucose-free ropivacaine for spinal anesthesia for lower limb and lower abdominal surgery Kaohsiung J Med Sci 2004 20 423 430 15506554
  • Simon MJ Veering BT Stienstra R van Kleef JW Burm AG The effects of age on neural blockade and hemodynamic changes after epidural anesthesia with ropivacaine Anesth Analg 2002 94 1325 1330 11973214
  • Dresner M Freeman J Calow C Quinn A Bamber J Ropivacaine 0.2% versus bupivacaine 0.1% with fentanyl: a double blind comparison for analgesia during labour Br J Anaesth 2000 85 826 829 11732513
  • Fernández-Guisasola J Serrano ML Cobo B A comparison of 0.0625% bupivacaine with fentanyl and 0.1% ropivacaine with fentanyl for continuous epidural labor analgesia Anesth Analg 2001 92 1261 1265 11323358
  • Messina M Magrin S Bignami E Prospective randomized, blind comparison of ropivacaine and levobupivacaine for superficial plexus anesthesia in carotid endoarterectomy Minerva Anestesiol 2009 75 7 12 19172143
  • Purdie NL McGrady EM Comparison of patient-controlled epidural bolus administration of 0.1% ropivacaine and 0.1% levobupivacaine, both with 0.0002% fentanyl, for analgesia during labour Anaesthesia 2004 59 133 137 14725515
  • Gutton C Bellefleur JP Puppo S Lidocaine versus ropivacaine for perineal infiltration post-episiotomy Int J Gynaecol Obstet 2013 122 33 36 23579103
  • Liu J Yuan W Wang X Peripheral nerve blocks versus general anesthesia for total knee replacement in elderly patients on the postoperative quality of recovery Clin Interv Aging 2014 9 341 350 24600214