Enhanced bioavailability and anthelmintic efficacy of mebendazole in redispersible microparticles with low-substituted hydroxypropylcellulose

References

• Hemphill A Müller J Alveolar and cystic echinococcosis: towards novel chemotherapeutical treatment options J Helminthol 2009 83 2 99 111 19296876
   PubMed Web of Science ®Google Scholar
• Dayan AD Albendazole, mebendazole and praziquantel. Review of non-clinical toxicity and pharmacokinetics Acta Trop 2003 86 2–3 141 159 12745134
   PubMed Web of Science ®Google Scholar
• Sievens-Figueroa L Bhakay A Jerez-Rozo JI Preparation and characterization of hydroxypropyl methyl cellulose films containing stable BCS Class II drug nanoparticles for pharmaceutical applications Int J Pharm 2012 423 2 496 508 22178619
   PubMed Web of Science ®Google Scholar
• Loh GOK Tan YT Peh KK Hydrophilic polymer solubilization on norfloxacin solubility in preparation of solid dispersion Powder Technology 2014 256 462 469
   Web of Science ®Google Scholar
• Onoue S Sato H Ogawa K Improved dissolution and pharmacokinetic behavior of cyclosporine. A using high-energy amorphous solid dispersion approach Int J Pharm 2010 399 1–2 94 101 20705124
   PubMed Web of Science ®Google Scholar
• Lim SC Paech MJ Sunderland B Liu Y In vitro and in vivo evaluation of a sublingual fentanyl water formulation Drug Des Devel Ther 2013 7 317 324
   Web of Science ®Google Scholar
• Dinunzio JC Brough C Hughey JR Miller DA Williams RO McGinity JW Fusion production of solid dispersions containing a heat-sensitive active ingredient by hot melt extrusion and Kinetisol dispersing Eur J Pharm Biopharm 2010 74 2 340 351 19818402
   PubMed Web of Science ®Google Scholar
• Usha AN Mutalik S Reddy MS Ranjith AK Kushtagi P Udupa N Preparation and, in vitro, preclinical and clinical studies of aceclofenac spherical agglomerates Eur J Pharm Biopharm 2008 70 2 674 683 18606224
   PubMed Web of Science ®Google Scholar
• Kawabata Y Yamamoto K Debari K Onoue S Yamada S Novel crystalline solid dispersion of tranilast with high photostability and improved oral bioavailability Eur J Pharm Biopharm 2010 39 4 256 262
   Google Scholar
• Molina-Berríos A Campos-Estrada C Lapier M Benznidazole prevents endothelial damage in an experimental model of Chagas disease Acta Trop 2013 127 1 6 13 23529066
   PubMed Web of Science ®Google Scholar
• Matadamas-Martínez F Nogueda-Torres B Hernández-Campos A Analysis of the effect of a 2-(trifluoromethyl)-1H-benzimidazole derivative on Trichinella spiralis muscle larvae Vet Parasitol 2013 194 2–4 193 207 23462252
   PubMed Web of Science ®Google Scholar
• Daniel-Mwambete K Torrado S Cuesta-Bandera C Ponce-Gordo F Torrado JJ The effect of solubilization on the oral bioavailability of three benzimidazole carbamate drugs Int J Pharm 2004 272 1–2 29 36 15019066
   PubMed Web of Science ®Google Scholar
• Swanepoel E Liebenberg W Villiers MM Quality evaluation of generic drugs by dissolution test: changing the USP dissolution medium to distinguish between active and non-active mebendazole polymorphs Eur J Pharm Biopharm 2003 55 3 345 349 12754010
   PubMed Web of Science ®Google Scholar
• Cirri M Maestrelli F Mennini N Mura P Influence of the preparation method on the physical-chemical properties of ketoprofen-cyclodextrin-phosphatidylcholine ternary Systems J Pharm Biomed Anal 2009 50 5 690 694 19097721
   PubMed Web of Science ®Google Scholar
• Cirri M Maestrelli F Mennini N Mura P Physical-chemical characterization of binary and ternary systems of ketoprofen with cyclodextrins and phospholipids J Pharm Biomed Anal 2009 50 5 683 689 19095391
   PubMed Web of Science ®Google Scholar
• Vo CL Park C Lee BJ Current trends and future perspectives of solid dispersions containing poorly water-soluble drugs Eur J Pharm Biopharm 2013 85 3 Pt B 799 813 24056053
   PubMed Web of Science ®Google Scholar
• García-Rodríguez JJ Torre-Iglesias PM Vegas-Sánchez MC Torrado-Durán S Bolás-Fernández F Torrado-Santiago S Changed crystallinity of mebendazole solid dispersion: Improved anthelmintic activity Int J Pharm 2011 403 1–2 23 28 20934497
   PubMed Web of Science ®Google Scholar
• Torrado S López ML Torrado G Bolás F Torrado S Cadórniga R A novel formulation of albendazole solution: oral bioavailability and efficacy evaluation Int J Pharm 1997 156 181 187
   Web of Science ®Google Scholar
• Beinborn NA Dua J Wiederhold NP Smyth HD Williams RO3rd Dry powder insufflation of crystalline and amorphous voriconazole formulations produced by thin film freezing to mice Eur J Pharm Biopharm 2012 81 3 600 608 22569473
   PubMed Web of Science ®Google Scholar
• García JJ Bolás F Torrado JJ Bioavailability and efficacy characteristics of two different oral liquid formulations of albendazole Int J Pharm 2003 250 2 351 358 12527162
   PubMed Web of Science ®Google Scholar
• Wakelin D Lloyd M Accelerated expulsion of adult Trichinella spiralis in mice given lymphoid cells and serum from infected donors Parasitology 1976 72 3 307 315 967521
   PubMed Web of Science ®Google Scholar
• Cerdeira AM Mazzotti M Gander B Formulation and drying of miconazole and itraconazole nanosuspensions Int J Pharm 2013 443 1–2 209 220 23291552
   PubMed Web of Science ®Google Scholar
• Karavas E Georgarakis E Sigalas MP Avgoustakis K Bikiaris D Investigation of the release mechanism of a sparingly water-soluble drug from solid dispersions in hydrophilic carriers based on physical state of drug, particle size distribution and drug–polymer interactions Eur J Pharm Biopharm 2007 66 3 334 347 17267194
   PubMed Web of Science ®Google Scholar
• Jana S Maji N Nayak AK Sen KK Basu SK Development of chitosan-based nanoparticles through inter-polymeric complexation for oral drug delivery Carbohydr Polym 2013 98 1 870 876 23987423
   PubMed Web of Science ®Google Scholar
• De Villiers MM Terblanche RJ Liebenberg W Swanepoel E Dekker TG Song M Variable-temperature X-ray powder diffraction analysis of the crystal transformation of the pharmaceutically preferred polymorph C of mebendazole J Pharm Biomed Anal 2005 38 3 435 441 15925244
   PubMed Web of Science ®Google Scholar
• Mura P Manderioli A Bramanti G Furlanetto S Pinzauti S Utilization of differential scanning calorimetry as a screening technique to determine the compatibility of ketoprofen with excipients Int J Pharm 1995 119 71 79
   Web of Science ®Google Scholar
• Pani NR Nath LK Acharya S Bhuniya B Application of DSC, IST, and FTIR study in the compatibility testing of nateglinide with different pharmaceutical excipients J Therm Anal Calorim 2012 108 1 219 226
   Web of Science ®Google Scholar
• Damian F Blaton N Naessens L Physicochemical characterization of solid dispersions of the antiviral agent UC-781 with polyethylene glycol 6000 and Gelucire 44/14 Eur J Pharm Sci 2000 10 4 311 322 10838021
   PubMed Web of Science ®Google Scholar
• Froehlich PE Gasparotto FS Mebendazol: identificação das formas polimórficas em diferentes matérias-primas e medicamentos (referência e genéricos) disponíveis no mercado nacional. [Mebendazole: identification of polymorphic forms in different raw materials and drugs (reference and generics) available domestically] Rev Ciênc Farm Básica Apl 2005 26 3 205 210 Portuguese
   Google Scholar
• Moes J Koolen S Huitema A Schellens J Beijnen J Nuijen B Development of an oral solid dispersion formulation for use in low-dose metronomic chemotherapy of paclitaxel Eur J Pharm Biopharm 2013 83 1 87 94 23085332
   PubMed Web of Science ®Google Scholar
• Karmwar P Graeser K Gordon KC Strachan CJ Rades T Investigation of properties and recrystallisation behaviour of amorphous indomethacin samples prepared by different methods Int J Pharm 2011 417 1–2 94 100 21182910
   PubMed Web of Science ®Google Scholar
• Mura P Bettinetti GP Cirri M Maestrelli F Sorrenti M Catenacci L Solid-state characterization and dissolution properties of Naproxen–Arginine–Hydroxypropyl-β-cyclodextrin ternary system Eur J Pharm Biopharm 2005 59 1 99 106 15567306
   PubMed Web of Science ®Google Scholar
• Chadha R Bala M Arora P Jain DV Pissurlenkar RRS Coutinho EC Valsartan inclusion by methyl-β-cyclodextrin: Thermodynamics, molecular modelling, Tween 80 effect and evaluation Carbohydr Polym 2014 103 15 300 309 24528733
   PubMed Web of Science ®Google Scholar
• Krishnaiah YS Veer RP Dinesh KB Satyanarayana V Karthiekeyan RS Bhaskar P Pharmacokinetic evaluation of guar gum-based colon-targeted drug delivery systems of mebendazole in healthy volunteers J Control Release 2003 88 1 95 103 12586507
   PubMed Web of Science ®Google Scholar
• Zhang M Li H Lang B Formulation and delivery of improved amorphous fenofibrate solid dispersions prepared by thin film freezing Eur J Pharm Biopharm 2012 82 3 534 544 22974985
   PubMed Web of Science ®Google Scholar
• Yang W Johnston KP Williams RO3rd Comparison of bioavailability of amorphous versus crystalline itraconazole nanoparticles via pulmonary administration in rats Eur J Pharm Biopharm 2010 75 1 33 41 20102737
   PubMed Web of Science ®Google Scholar
• Hess JA Chandrasekar PH Mortiere M Molinari JA Comparative Efficacy of Ketoconazole and Mebendazole in Experimental Trichinosis Antimicrob Agents Chemother 1986 30 6 953 954 3813518
   PubMed Web of Science ®Google Scholar
• de-la-Rosa JL Alvarez N Gomez-Priego A Study of the reproductive capacity of Trichinella spiralis recovered from experimentally infected mice under-dosed with albendazole or mebendazole Trop Biomed 2007 24 2 93 97 18209715
   PubMed Web of Science ®Google Scholar
• Maki J Yanagisawa T Comparative efficacy of flubendazole and mebendazole on encysted larvae of Trichinella spiralis (USA strain) in the diaphragm of mice and rats J Helminthol 1988 62 1 35 39 3372977
   PubMed Web of Science ®Google Scholar
• Zardi EM Petrarca V Pozio E Uwechie V Tamburrini A Laghi V A case from India of neurocysticercosis responsive to albendazole treatment Parasite 2000 7 1 54 56 10743650
   PubMed Web of Science ®Google Scholar
• Yépez-Mulia L Morales-Hurtado R Viveros-Guzmán N Evaluation of albendazole prodrugs in experimental trichinellosis Arch Med Res 1999 30 5 368 374 10596455
   PubMed Web of Science ®Google Scholar