From micro- to nanostructured implantable device for local anesthetic delivery

References

• EdgcombeHHockingG[webpage on the Internet]. Local anaesthetic pharmacologyWorld Anaesth Tutor Week2005125127 Available from: http://www.frca.co.uk/documents/la.pdfAccessed April 8, 2016
   Google Scholar
• ShiptonEANew formulations of local anaesthetics-part IAnesthesiol Res Pract2012201254640922190922
   PubMedGoogle Scholar
• AndreaeMHAndreaeDALocal anaesthetics and regional anaesthesia for preventing chronic pain after surgeryCochrane Database Syst Rev2012107CD00710523076930
   PubMedGoogle Scholar
• BrennanFCarrDBCousinsMPain management: a fundamental human rightAnesth Analg2007105120522117578977
   PubMed Web of Science ®Google Scholar
• SentürkMOzcanPETaluGKThe effects of three different analgesia techniques on long-term postthoracotomy painAnesth Analg2002941111511772793
   PubMed Web of Science ®Google Scholar
• KroinJSBuvanendranAWattsDESahaCTumanKJUpregulation of cerebrospinal fluid and peripheral prostaglandin E2 in a rat postoperative pain modelAnesth Analg20061032334343 table of contents16861414
   PubMed Web of Science ®Google Scholar
• GuptaAFavaiosSPerniolaAMagnusonABerggrenLA meta-analysis of the efficacy of wound catheters for post-operative pain managementActa Anaesthesiol Scand201155778579621615349
   PubMedGoogle Scholar
• Galindo AriasMLEVOBUPIVACAINE – a long acting local anaesthetic, with less cardiac and neurotoxicityUpdate Anaesth2002142325
   Google Scholar
• TanJPKTanMBHTamMKCApplication of nanogel systems in the administration of local anestheticsLocal Reg Anesth2010319310022915875
   PubMedGoogle Scholar
• CovinoBGGiddonDBPharmacology of local anesthetic agentsJ Dent Res1981608145414596942010
   PubMedGoogle Scholar
• McLureHARubinAPReview of local anaesthetic agentsMinerva Anestesiol2005713597415714182
   PubMedGoogle Scholar
• LeeKJYangSYRyuWHControlled release of bupivacaine HCl through microchannels of biodegradable drug delivery deviceBiomed Microdevices201214358359322374474
   PubMedGoogle Scholar
• StevensRAChesterWLSchubertABrandonDGrueterJAZumrickJpH-adjustment of 2-chloroprocaine quickens the onset of epidural anaesthesiaCan J Anaesth19893655155182551520
   PubMedGoogle Scholar
• WeinigerCFGolovanevskiLDombAJIckowiczDExtended release formulations for local anaesthetic agentsAnaesthesia201267890691622607613
   PubMedGoogle Scholar
• GuayJAdverse events associated with intravenous regional anesthesia (Bier block): a systematic review of complicationsJ Clin Anesth200921858559420122591
   PubMed Web of Science ®Google Scholar
• BrownDLRansomDMHallJALeichtCHSchroederDROffordKPRegional anesthesia and local anesthetic-induced systemic toxicity: seizure frequency and accompanying cardiovascular changesAnesth Analg19958123213287618723
   PubMed Web of Science ®Google Scholar
• KuhnertBRKuhnertPMPhilipsonEHSyracuseCDKaineCJChang-hyonYThe half-life of 2-chloroprocaineAnesth Analg19866532732783954093
   PubMed Web of Science ®Google Scholar
• FredholtKLarsenDHLarsenCModification of in vitro drug release rate from oily parenteral depots using a formulation approachEur J Pharm Sci200011323123711042229
   PubMedGoogle Scholar
• LarsenDHFredholtKLarsenCAssessment of rate of drug release from oil vehicle using a rotating dialysis cellEur J Pharm Sci200011322322911042228
   PubMedGoogle Scholar
• LarsenSWØstergaardJFriberg-JohansenHJessenMNBLarsenCIn vitro assessment of drug release rates from oil depot formulations intended for intra-articular administrationEur J Pharm Sci200629534835416920337
   PubMedGoogle Scholar
• LarsenSWFrostABØstergaardJMarcherHLarsenCOn the mechanism of drug release from oil suspensions in vitro using local anesthetics as model drug compoundsEur J Pharm Sci2008341374418374550
   PubMedGoogle Scholar
• ThingMLarsenCØstergaardJJensenHLarsenSWIn vitro release from oil injectables for intra-articular administration: importance of interfacial area, diffusivity and partitioningEur J Pharm Sci201245335135722178293
   PubMedGoogle Scholar
• DubnikaALocaDBerzina-CimdinaLFunctionalized hydroxyapatite scaffolds coated with sodium alginate and chitosan for controlled drug deliveryProc Est Acad Sci2012613193
   Google Scholar
• SalmaIPilmaneMSkagersAEarly morphofunctional response of contact tissue after intraosal implantation in rabbit jaw of pure synthetic hydroxyapatite (HAp) bioceramic materials and HAp saturated with lidocaineStomatologija200911411311820179398
   PubMedGoogle Scholar
• KumarswamyAMorettiAPaquetteDPadillaREverettENaresSIn vivo assessment of osseous wound healing using a novel bone putty containing lidocaine in the surgical management of tooth extractionsInt J Dent2012201218
   Google Scholar
• LiuDZSheuMTChenCHYangYRHoHORelease characteristics of lidocaine from local implant of polyanionic and polycationic hydrogelsJ Control Release2007118333333917292505
   PubMed Web of Science ®Google Scholar
• SobankoJFMillerCJAlsterTSTopical anesthetics for dermatologic procedures: a reviewDermatologic Surg2012385709721
   PubMed Web of Science ®Google Scholar
• PetrisorGIonRMBrachaisCHCouvercelleJ-PChambinODesigning medical devices based on silicon polymeric material with controlled release of local anestheticsJ Macromol Sci Part A2012495439444
   Web of Science ®Google Scholar
• GeeverLMCooneyCCLyonsJGCharacterisation and controlled drug release from novel drug-loaded hydrogelsEur J Pharm Biopharm20086931147115918502627
   PubMedGoogle Scholar
• FuYKaoWJDrug release kinetics and transport mechanisms from semi-interpenetrating networks of gelatin and poly(ethylene glycol) diacrylatePharm Res20092699971003
   Google Scholar
• MakinoKIdenumaRMurakamiTOhshimaHDesign of a rate- and time-programming drug release device using a hydrogel: pulsatile drug release from kappa-carrageenan hydrogel device by surface erosion of the hydrogelColloids Surf B Biointerfaces200120435535911166546
   PubMed Web of Science ®Google Scholar
• KloseDSiepmannFElkharrazKSiepmannJPLGA-based drug delivery systems: importance of the type of drug and device geometryInt J Pharm20083541–29510318055140
   PubMed Web of Science ®Google Scholar
• BlancoMDBernardoMVGómezCMuñizETeijónJMBupivacaine- loaded comatrix formed by albumin microspheres included in a poly(lactide-co-glycolide) film: in vivo biocompatibility and drug release studiesBiomaterials199920201919192410514068
   PubMedGoogle Scholar
• ChenP-CParkYJChangL-CInjectable microparticle-gel system for prolonged and localized lidocaine release. I. In vitro characterizationJ Biomed Mater Res A2004704341241915293314
   PubMedGoogle Scholar
• CurleyJCastilloJHotzJProlonged regional nerve blockade. Injectable biodegradable bupivacaine/polyester microspheresAnesthesiology1996846140114108669682
   PubMedGoogle Scholar
• KohaneDSSmithSELouisDNProlonged duration local anesthesia from tetrodotoxin-enhanced local anesthetic microspheresPain20031041–241542112855352
   PubMedGoogle Scholar
• HuangYYChungTWTzengTWA method using biodegradable polylactides/polyethylene glycol for drug release with reduced initial burstInt J Pharm199918219310010332078
   PubMedGoogle Scholar
• ChenP-CKohaneDSParkYJBartlettRHLangerRYangVCInjectable microparticle-gel system for prolonged and localized lidocaine release. II. In vivo anesthetic effectsJ Biomed Mater Res A200470345946615293320
   PubMedGoogle Scholar
• ChungTWHuangYYLiuYZEffects of the rate of solvent evaporation on the characteristics of drug loaded PLLA and PDLLA microspheresInt J Pharm2001212216116911165073
   PubMed Web of Science ®Google Scholar
• ZhangHLuYZhangGGaoSSunDZhongYBupivacaine-loaded biodegradable poly(lactic-co-glycolic) acid microspheres. I. Optimization of the drug incorporation into the polymer matrix and modelling of drug releaseInt J Pharm20083511–224424918024022
   PubMedGoogle Scholar
• McAlvinJBReznorGShankarappaSAStefanescuCFKohaneDSLocal toxicity from local anesthetic polymeric microparticlesAnesth Analg2013116479480323460564
   PubMedGoogle Scholar
• HuangYYChungTWTzengTWDrug release from PLA/PEG microparticulatesInt J Pharm19971561915
   Google Scholar
• BragagniMBeneitezCMartínCDe La OssaDHPMuraPAGil-AlegreMESelection of PLA polymers for the development of injectable prilocaine controlled release microparticles: usefulness of thermal analysisInt J Pharm20134411–246847523164705
   PubMedGoogle Scholar
• PedersenJLLillesøJHammerNABupivacaine in microcapsules prolongs analgesia after subcutaneous infiltration in humans: a dose-finding studyAnesth Analg200499391291815333431
   PubMedGoogle Scholar
• Le CorrePEstèbeJPClémentRSpray-dryed bupivacaine-loaded microspheres: in vitro evaluation and biopharmaceutics of bupivacaine following brachial plexus administration in sheepInt J Pharm20022381–219120311996823
   PubMedGoogle Scholar
• EstebeJPLe CorrePDu PlessisLThe pharmacokinetics and pharmacodynamics of bupivacaine-loaded microspheres on a brachial plexus block model in sheepAnesth Analg2001932447455 4th contents page11473878
   PubMed Web of Science ®Google Scholar
• MontanariLCilurzoFSelminFPoly(lactide-co-glycolide) microspheres containing bupivacaine: comparison between gamma and beta irradiation effectsJ Control Release200390328129012880695
   PubMedGoogle Scholar
• YinWYatesMZEncapsulation and sustained release from biodegradable microcapsules made by emulsification/freeze drying and spray/freeze dryingJ Colloid Interface Sci2009336115516119423128
   PubMed Web of Science ®Google Scholar
• HolgadoMAAriasJLCózarMJAlvarez-FuentesJGañán-CalvoAMFernández-ArévaloMSynthesis of lidocaine-loaded PLGA microparticles by flow focusing. Effects on drug loading and release propertiesInt J Pharm20083581–2273518372128
   PubMed Web of Science ®Google Scholar
• XuQHashimotoMDangTTPreparation of monodisperse biodegradable polymer microparticles using a microfluidic flow-focusing device for controlled drug deliverySmall20095131575158119296563
   PubMed Web of Science ®Google Scholar
• VladisavljevićGTShahmohamadiHDasDBEkanemEETauanovZSharmaLGlass capillary microfluidics for production of monodispersed poly (DL-lactic acid) and polycaprolactone microparticles: experiments and numerical simulationsJ Colloid Interface Sci201441816317024461831
   PubMed Web of Science ®Google Scholar
• KloseDSiepmannFWillartJFDescampsMSiepmannJDrug release from PLGA-based microparticles: effects of the “microparticle:bulk fluid” ratioInt J Pharm20103831–212313119748558
   PubMed Web of Science ®Google Scholar
• KranzHBodmeierRStructure formation and characterization of injectable drug loaded biodegradable devices: in situ implants versus in situ microparticlesEur J Pharm Sci2008342–316417218501569
   PubMed Web of Science ®Google Scholar
• KranzHYilmazEBrazeauGABodmeierRIn vitro and in vivo drug release from a novel in situ forming drug delivery systemPharm Res20082561347135417968634
   PubMedGoogle Scholar
• KohaneDSLippMKinneyRCBiocompatibility of lipid–protein–sugar particles containing bupivacaine in the epineuriumJ Biomed Mater Res200259345045911774302
   PubMed Web of Science ®Google Scholar
• FundueanuGConstantinMAscenziPPoly(N-isopropylacrylamide-co-acrylamide) cross-linked thermoresponsive microspheres obtained from preformed polymers: influence of the physico-chemical characteristics of drugs on their release profilesActa Biomater20095136337318723416
   PubMedGoogle Scholar
• FundueanuGConstantinMOaneaIHarabagiuVAscenziPSimionescuBCPrediction of the appropriate size of drug molecules that could be released by a pulsatile mechanism from pH/thermoresponsive microspheres obtained from preformed polymersActa Biomater2012831281128921945634
   PubMed Web of Science ®Google Scholar
• FundueanuGConstantinMAsmarandeiIHarabagiuVAscenziPSimionescuBCThe thermosensitivity of pH/thermoresponsive microspheres activated by the electrostatic interaction of pH-sensitive units with a bioactive compoundJ Biomed Mater Res – Part A2013101616611669
   Google Scholar
• SivakumaranDMaitlandDHoareTInjectable microgel-hydrogel composites for prolonged small-molecule drug deliveryBiomacromolecules201112114112412022007750
   PubMed Web of Science ®Google Scholar
• PatenaudeMHoareTInjectable, mixed natural-synthetic polymer hydrogels with modular propertiesBiomacromolecules201213236937822251304
   PubMedGoogle Scholar
• SivakumaranDMaitlandDOszustowiczTHoareTTuning drug release from smart microgel-hydrogel composites via cross-linkingJ Colloid Interface Sci2013392142243023137903
   PubMedGoogle Scholar
• GangulySDashAKA novel in situ gel for sustained drug delivery and targetingInt J Pharm20042761–2839215113617
   PubMed Web of Science ®Google Scholar
• FoleyPLUleryBDKanHMA chitosan thermogel for delivery of ropivacaine in regional musculoskeletal anesthesiaBiomaterials201334102539254623321347
   PubMed Web of Science ®Google Scholar
• RadinSChenTDucheynePThe controlled release of drugs from emulsified, sol gel processed silica microspheresBiomaterials200930585085819010531
   PubMed Web of Science ®Google Scholar
• CostacheMCVaughanADQuHDucheynePDevoreDITyrosine-derived polycarbonate-silica xerogel nanocomposites for controlled drug deliveryActa Biomater2013956544655223395749
   PubMed Web of Science ®Google Scholar
• CuiDCLuWLSaEAGuMJLuXJFanTYPoly(acrylic acid) microspheres loaded with lidocaine: preparation and characterization for arterial embolizationInt J Pharm20124361–252753522820132
   PubMedGoogle Scholar
• GautierHChamblainVWeissPMerleCBoulerJMIn vitro characterisation of calcium phosphate biomaterials loaded with lidocaine hydrochloride and morphine hydrochlorideJ Mater Sci Mater Med201021123141315021046202
   PubMedGoogle Scholar
• VerronEGauthierOJanvierPAnalgesic properties of calcium phosphate apatite loaded with bupivacaine on postoperative painJ Biomed Mater Res – Part B Appl Biomater2010941899620524182
   PubMedGoogle Scholar
• MendesLPDelgadoJMFCostaADBiodegradable nanoparticles designed for drug delivery: the number of nanoparticles impacts on cytotoxicityToxicol Vitr20152912681274
   PubMed Web of Science ®Google Scholar
• ShangLNienhausKNienhausGUEngineered nanoparticles interacting with cells: size mattersJ Nanobiotechnology2014121524491160
   PubMed Web of Science ®Google Scholar
• VermaAStellacciFEffect of surface properties on nanoparticle-cell interactionsSmall201061122119844908
   PubMed Web of Science ®Google Scholar
• De PaulaECeredaCMSTofoliGRFranz-MontanMFracetoLFde AraújoDRDrug delivery systems for local anestheticsRecent Pat Drug Deliv Formul201041233419807683
   PubMedGoogle Scholar
• WeinigerCFGolovanevskiMSokolsky-PapkovMDombAJReview of prolonged local anesthetic actionExpert Opin Drug Deliv20107673775220408748
   PubMed Web of Science ®Google Scholar
• JunghannsJUAHMüllerRHNanocrystal technology, drug delivery and clinical applicationsInt J Nanomedicine20083329530918990939
   PubMed Web of Science ®Google Scholar
• RangasamyMNano technology : a reviewJ Appl Pharm Sci20110102816
   Google Scholar
• MoreyTEVarshneyMFlintJARajasekaranSShahDODennisDMTreatment of local anesthetic-induced cardiotoxicity using drug scavenging nanoparticlesNano Lett20044475775926321882
   PubMedGoogle Scholar
• CohenRKanaanHGrantGJBarenholzYProlonged analgesia from Bupisome and Bupigel formulations: from design and fabrication to improved stabilityJ Control Release2012160234635222233969
   PubMedGoogle Scholar
• Fernandes FracetoLDe Matos Alves PintoLFranzoniLSpectroscopic evidence for a preferential location of lidocaine inside phospholipid bilayersBiophys Chem200299322924312408938
   PubMedGoogle Scholar
• GrantGJPiskounBBansinathMAnalgesic duration and kinetics of liposomal bupivacaine after subcutaneous injection in miceClin Exp Pharmacol Physiol2003301296696814678238
   PubMedGoogle Scholar
• GrantGJBarenholzYBolotinEMA novel liposomal bupivacaine formulation to produce ultralong-acting analgesiaAnesthesiology2004101113313715220782
   PubMed Web of Science ®Google Scholar
• CabeçaLFFernandesSAde PaulaEMarsaioliAJTopology of a ternary complex (proparacaine-beta-cyclodextrin-liposome) by STD NMRMagn Reson Chem200846983283718642398
   PubMedGoogle Scholar
• De AraujoDRCeredaCMSBrunettoGBPharmacological and local toxicity studies of a liposomal formulation for the novel local anaesthetic ropivacaineJ Pharm Pharmacol200860111449145718957165
   PubMed Web of Science ®Google Scholar
• De AraujoDRCeredaCMSBrunettoGBPintoLMSantanaMHde PaulaEEncapsulation of mepivacaine prolongs the analgesia provided by sciatic nerve blockade in miceCan J Anaesth200451656657215197119
   PubMedGoogle Scholar
• ToongsuwanSLiLCEricksonBKChangHCFormulation and characterization of bupivacaine lipospheresInt J Pharm20042801–2576515265547
   PubMedGoogle Scholar
• KohaneDSLippMKinneyRCLotanNLangerRSciatic nerve blockade with lipid-protein-sugar particles containing bupivacainePharm Res200017101243124911145230
   PubMedGoogle Scholar
• ColomboGPaderaRLangerRKohaneDSProlonged duration local anesthesia with lipid-protein-sugar particles containing bupivacaine and dexamethasoneJ Biomed Mater Res – Part A2005752458464
   Google Scholar
• Zur MühlenASchwarzCMehnertWSolid lipid nanoparticles (SLN) for controlled drug delivery – drug release and release mechanismEur J Pharm Biopharm19984521491559704911
   PubMed Web of Science ®Google Scholar
• SchwarzCMehnertWFreeze-drying of drug-free and drug-loaded solid lipid nanoparticles (SLN)Int J Pharm1997157217117910477814
   PubMed Web of Science ®Google Scholar
• PietkiewiczJSznitowskaMPlaczekMThe expulsion of lipophilic drugs from the cores of solid lipid microspheres in diluted suspensions and in concentratesInt J Pharm20063101–2647116413712
   PubMedGoogle Scholar
• GörnerTGrefRMichenotDSommerFTranMNDellacherieELidocaine-loaded biodegradable nanospheres. I. Optimization of the drug incorporation into the polymer matrixJ Control Release19995732592689895413
   PubMed Web of Science ®Google Scholar
• PolakovicMGornerTGrefRDellacherieELidocaine-loaded biodegradable nanospheres. II. Modeling of drug releaseJ Control Release1999602–316917710425323
   PubMedGoogle Scholar
• MoraesCMDe MatosAPDe LimaRRosaAHDe PaulaEFracetoLFInitial development and characterization of PLGA nanospheres containing ropivacaineJ Biol Phys2007335–645546119669531
   PubMedGoogle Scholar
• Ramos CamposEVSilva de MeloNFGuilhermeVAPreparation and characterization of poly(ε-caprolactone) nanospheres containing the local anesthetic lidocaineJ Pharm Sci2013102121522623108693
   PubMedGoogle Scholar
• GovenderTRileyTEhtezaziTDefining the drug incorporation properties of PLA-PEG nanoparticlesInt J Pharm200019919511010794931
   PubMed Web of Science ®Google Scholar
• BilatiUAllémannEDoelkerEDevelopment of a nanoprecipitation method intended for the entrapment of hydrophilic drugs into nanoparticlesEur J Pharm Sci2005241677515626579
   PubMed Web of Science ®Google Scholar
• GovenderTStolnikSGarnettMCIllumLDavisSSPLGA nanoparticles prepared by nanoprecipitation: drug loading and release studies of a water soluble drugJ Control Release19995721711859971898
   PubMed Web of Science ®Google Scholar
• MoraesCMDe LimaRRosaAHDe PaulaEFracetoLFEncapsulation of local anesthetic bupivacaine in biodegradable poly(DL-lactide-co-glycolide) nanospheres: factorial design, characterization and cytotoxicity studiesMacromol Symp20092811106112
   Google Scholar
• MoraesCMDe PaulaERosaAHFracetoLFPhysicochemical stability of poly(lactide-co-glycolide) nanocapsules containing the local anesthetic bupivacaineJ Braz Chem Soc20102169951000
   Google Scholar
• GarciaXEscribanoEDomenechJQueraltJFreixesJIn vitro characterization and in vivo analgesic and anti-allodynic activity of PLGA-bupivacaine nanoparticlesJ Nanoparticle Res201113522132223
   Google Scholar
• MoraesCMde MatosAPde PaulaERosaAHFracetoLFBenzocaine loaded biodegradable poly-(d,l-lactide-co-glycolide) nanocapsules: factorial design and characterizationMater Sci Eng B Solid-State Mater Adv Technol20091653243246
   Google Scholar
• Silva de MeloNFde AraújoDRGrilloRBenzocaine-loaded polymeric nanocapsules: study of the anesthetic activitiesJ Pharm Sci201210131157116522105694
   PubMedGoogle Scholar
• De MeloNFSGrilloRGuilhermeVAPoly(lactide-co-glycolide) nanocapsules containing benzocaine: influence of the composition of the oily nucleus on physico-chemical properties and anesthetic activityPharm Res20112881984199421472490
   PubMed Web of Science ®Google Scholar
• WeldonCBTsuiJHShankarappaSAElectrospun drug-eluting sutures for local anesthesiaJ Control Release2012161390390922609349
   PubMed Web of Science ®Google Scholar
• MocanuAPascaRDTomoaiaGNew procedure to synthesize silver nanoparticles and their interaction with local anestheticsInt J Nanomedicine201383867387424143090
   PubMed Web of Science ®Google Scholar
• TanJPKGohCHTamKCComparative drug release studies of two cationic drugs from pH-responsive nanogelsEur J Pharm Sci2007324–534034817950583
   PubMedGoogle Scholar
• TanJPKZengAQChangCCTamKCRelease kinetics of procaine hydrochloride (PrHy) from pH-responsive nanogels: theory and experimentsInt J Pharm20083571–230531318358651
   PubMedGoogle Scholar
• TanJPKWangQTamKCControl of burst release from nanogels via layer by layer assemblyJ Control Release2008128324825418457895
   PubMed Web of Science ®Google Scholar
• HoareTYoungSLawlorMWKohaneDSThermoresponsive nanogels for prolonged duration local anesthesiaActa Biomater20128103596360522732383
   PubMed Web of Science ®Google Scholar
• HoareTSivakumaranDStefanescuCFLawlorMWKohaneDSNanogel scavengers for drugs: local anesthetic uptake by thermoresponsive nanogelsActa Biomater2012841450145822244983
   PubMedGoogle Scholar
• YaghmurARappoltMOøstergaardJLarsenCLarsenSWCharacterization of bupivacaine-loaded formulations based on liquid crystalline phases and microemulsions: the effect of lipid compositionLangmuir20122852881288922247936
   PubMed Web of Science ®Google Scholar
• GrilloRde MeloNFSde AraújoDRde PaulaERosaAHFracetoLFPolymeric alginate nanoparticles containing the local anesthetic bupivacaineJ Drug Target201018968869920196632
   PubMed Web of Science ®Google Scholar