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Journal of Receptor Research Volume 8, 1988 - Issue 6
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Research Article

Method for Comparing Selectivities of Unlabeled Subpopulation-Selective Ligands: Application to Muscarinic Receptors

John Ellis Neuroscience Research Unit, Department of Psychiatry, University of Vermont, Burlington, VT, 05405, USA
Pages 885-900 | Published online: 26 Sep 2008

References

  • Ellis J., Lenox R. H. Quaternary forms of classical muscarinic antagonists distinguish subpopulations of muscarinic receptors: Correlation with gallamine-defined subpopulations. Biochem. Bioph. Res. Com. 1985; 126: 1242–1250
  • Ellis J., Seidenberg M. Interactions between gallamine and muscarinic receptors: allosterism and subpopulation specificity are separate phenomena. Eur. J. Pharmacol. 1987; 144: 39–44
  • Vanderheyden P., Ebinger G., Vauquelin G. Different agonist binding properties of M1 and M2 muscarinic receptors in calf brain cortex membranes. Biochem. Pharmacol. 1987; 36: 4119–4124
  • Feldman H. A. Mathematical theory of complex ligand-binding systems at equilibrium: some methods for parameter fitting. Anal. Biochem. 1972; 48: 317–338
  • Knott G. D. MLAB - Mathematical modeling tool. Comput. Prog. Biomed. 1979; 10: 271–280
  • Ellis J., Hoss W. Analysis of regional variations in the affinities of muscarinic agonists in rat brain. Brain Res. 1980; 193: 189–190
  • Ellis J., Lenox R. H. Characterization of the interactions of gallamine with muscarinic receptors from brain. Biochem. Pharmacol. 1985; 34: 2214–2217
  • Stockton J. M., Birdsall N. J.M., Burgen A. S.V., Hulme E. C. Modification of the binding properties of muscarinic receptors by gallamine. Mol. Pharmacol. 1983; 23: 551–557
  • Gillard M., Waelbroeck M., Christophe J. In vitro effects of gallamine on dissociation kinetics of (3H)N-methylscopolamine and (3H)pirenzepine from rat brain muscarinic receptors. J. Rec. Res. 1986; 6: 47–61
  • Watson M., Roeske W. R., Yamamura H. I. [3H]Pirenzepine and (-)-[3H]quinuclidinyl benzilate binding to rat cerebral cortical and cardiac muscarinic cholinergic sites. II. Characterization and regulation of antagonist binding to putative muscarinic subtypes. J. Pharmacol. Exp. Ther. 1986; 237: 419–427
  • Watson M., Yamamura H. I, Roeske W. R. [3H]Pirenzepine and (-)-[3H]quinuclidinyl benzilate binding to rat cerebral cortical and cardiac muscarinic cholinergic sites. I. Characterization and regulation of agonist binding to putative muscarinic subtypes. J. Pharmacol. Exp. Ther. 1986; 237: 411–418

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