161
Views
5
CrossRef citations to date
0
Altmetric
Research Article

Solid-state compatibility screening of excipients suitable for development of indapamide sustained release solid-dosage formulation

, &
Pages 481-489 | Received 04 May 2012, Accepted 27 Jul 2012, Published online: 24 Sep 2012

References

  • Gombás A, Szabó-Revész P, Kata M, Regdon G, Erõs I. Quantitative determination of crystallinity of α-lactose monohydrate by DSC. J Therm Anal Calorim 2002;68:503–510.
  • Medeiros ACD, Correia LP, Simões MOS, Macêdo RO. Technological quality determination of pharmaceutical disintegrant by DSC cooling and DCS photovisual. J Therm Anal Calorim 2007;88:311–315.
  • Gandhi R, Pillai O, Thilagavathi R, Gopalakrishnan B, Kaul CL, Panchagnula R. Characterization of azithromycin hydrates. Eur J Pharm Sci 2002;16:175–184.
  • Ramos LA, Cavalheiro ÉTG. Thermal behaviour of loratadine. J Therm Anal Calorim 2007;87:831–834.
  • Venkataram S, Khohlokwane M, Wallis SH. Differential scanning calorimetry as a quick scanning technique for solid state stability studies. Drug Dev Ind Pharm 1995;21:847–855.
  • Martini A, Kume S, Crivellente M, Artico R. Use of subambient differential scanning calorimetry to monitor the frozen-state behavior of blends of excipients for freeze-drying. PDA J Pharm Sci Technol 1997;51:62–67.
  • Wesolowski M. Thermoanalytical methods in pharmaceutical technology. J Therm Anal 1992;38:2239–2245.
  • Blanco M, Valdés D, Bayod MS, Fernández-Mari F, Llorente I. Characterization and analysis of polymorphs by near-infrared spectrometry. Anal Chim Acta 2004;502:221–227.
  • Rodionova OY, Houmøller LP, Pomerantsev AL, Geladi P, Burger J, Dorofeyev VL, Arzamastsev AP. NIR spectrometry for counterfeit drug detection: A feasibility study. Anal Chim Acta 2005;549:151–158.
  • Pollanen K, Hakkinen A, Huhtanen M, Satu-Pia R, Karjalainen M, Rantanen J, Louhi-Kultanen M, Nystrom L. DRIFT-IR for quantitative characterization of polymorphic composition of sulfathiazole. Anal Chim Acta 2005;544:108–117.
  • Petruševski G, Ugarkovic S, Makreski P. Solid-state transformation of the pseudopolymorphic forms of codeine phosphate hemihydrate and codeine phosphate sesquihydrate monitored by vibrational spectroscopy and thermal analysis. J Mol Struct 2011;993:328–335.
  • Petrusevski G, Naumov P, Jovanovski G, Bogoeva-Gaceva G, Ng SW. Solid-state forms of sodium valproate, active component of the anticonvulsant drug epilim. Chem Med Chem 2008;3:1377–1386.
  • Naumov P, Petruševski G, Jovanovski G. Vibrational spectra of calcium, strontium and barium valproates. Selfassembly of valproate nanostrands in aqueous solution and in the solid state. Cryst Eng Comm 2010;12:2325–2331.
  • Narang AS, Rao VM, Raghavan KS. Developing Solid Oral Dosage Forms: Pharmaceutical Theory and Practice. Elsevier Inc, 2009:125–145.
  • Cunha-Filho MS, Martínez-Pacheco R, Landín M. Compatibility of the antitumoral beta-lapachone with different solid dosage forms excipients. J Pharm Biomed Anal 2007;45:590–598.
  • Siepmann J, Peppas NA. Modeling of drug release from delivery systems based on hydroxypropyl methylcellulose (HPMC). Adv Drug Deliv Rev 2001;48:139–157.
  • Ambrosioni E, Safar M, Degaute JP, Malin PL, MacMahon M, Pujol DR et al. Low-dose antihypertensive therapy with 1.5 mg sustained-release indapamide: results of randomised double-blind controlled studies. European study group. J Hypertens 1998;16:1677–1684.
  • Leonetti G. Clinical positioning of indapamide sustained release 1.5mg in management protocols for hypertension. Drugs 2000;59 Suppl 2:27–38; discussion 39.
  • Hauschild K, Picker-Freyer KM. Evaluation of tableting and tablet properties of Kollidon SR: the influence of moisture and mixtures with theophylline monohydrate. Pharm Dev Technol 2006;11:125–140.
  • Kotler K, Karl M, Nalawade S, Rottman N. Hot-melt extrusion with BASF pharma polymers, extrusion compendium. 2010, BASF SE, Pharma Ingredients & Services, 67056 Ludwigshafen, Germany.
  • Schachter D, Schmitt R, Mitchell S, Tirol G. Solid solution of a poorly soluble model drug in a phase-separated polymer matrix: melt-prepared dispersions based on Polyox WSR. 30th Annual Meeting of the Controlled Release Society, Glasgow, Scotland, July 19–23, 2003.
  • Rus LM, Tomuta I, Iuga C, Maier C, Kacso I, Borodi G, Bratu I, Bojita M. Indapamide slow release tablet preformulation: interactions with excipients analysis. Clujul Medical, 2011; 84, 550–555.
  • DiFeo TJ, Shuster JE. Analytical profiles of drug substances and excipients, Academic Press, Inc. 1994;23:229–268.

Reprints and Corporate Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

To request a reprint or corporate permissions for this article, please click on the relevant link below:

Academic Permissions

Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?

Obtain permissions instantly via Rightslink by clicking on the button below:

If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.