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Research Article

Investigation of different emulsion systems for dermal delivery of nicotinamide

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Pages 1417-1423 | Received 30 Apr 2012, Accepted 05 Sep 2012, Published online: 06 Jun 2013

References

  • Shalita AR, Smith JG, Parish LC, Sofman MS, Chalker DK. Topical nicotinamide compared with clindamycin gel in the treatment of inflammatory acne vulgaris. Int J Dermatol 1995;34:434–437.
  • Lawrence MJ, Rees GD. Microemulsion-based media as novel drug delivery systems. Adv Drug Deliv Rev 2000;45:89–121.
  • Bissett DL. Method of reducing cellulite in mammalian skin United States Patent 5962482, 5 October, 1999.
  • Namazi MR. Nicotinamide as a potential addition to the anti-atopic dermatitis armamentarium. Int Immunopharmacol 2004;4:709–712.
  • Hakozaki T, Minwalla L, Zhuang J, Chhoa M, Matsubara A, Miyamoto K et al. The effect of niacinamide on reducing cutaneous pigmentation and suppression of melanosome transfer. Br J Dermatol 2002;147:20–31.
  • Gensler HL. Prevention of photoimmunosuppression and photocarcinogenesis by topical nicotinamide. Nutr Cancer 1997;29:157–162.
  • Nicoli S, Zani F, Bilzi S, Bettini R, Santi P. Association of nicotinamide with parabens: effect on solubility, partition and transdermal permeation. Eur J Pharm Biopharm 2008;69:613–621.
  • Tenjarla S. Microemulsions: an overview and pharmaceutical applications. Crit Rev Ther Drug Carrier Syst 1999;16:461–521.
  • Yuan Y, Li SM, Mo FK, Zhong DF. Investigation of microemulsion system for transdermal delivery of meloxicam. Int J Pharm 2006;321:117–123.
  • Gasco MR, Gallarate M, Pattarino F. In vitro permeation of azelaic acid from viscosized microemulsions. Int J Pharm 1991;69:193–196.
  • Peltola S, Saarinen-Savolainen P, Kiesvaara J, Suhonen TM, Urtti A. Microemulsions for topical delivery of estradiol. Int J Pharm 2003;254:99–107.
  • Baroli B, López-Quintela MA, Delgado-Charro MB, Fadda AM, Blanco-Méndez J. Microemulsions for topical delivery of 8-methoxsalen. J Control Release 2000;69:209–218.
  • Schmalfuss U, Neubert R, Wohlrab W. Modification of drug penetration into human skin using microemulsions. J Control Release 1997;46:279–285.
  • Delgado-Charro MB, Iglesias-Vilas G, Blanco-Méndez J, Lopez Quintela MA, Merty JP, Guy RH. Delivery of a hydrophilic solute through the skin from novel microemulsion systems. Eur J Pharm Biopharm 1997;43:37–42.
  • Trotta M, Pattarino F, Gasco MR. Transdermal permeation of apomorphine through hairless mouse skin from microemulsions. Pharm Acta Helv 1996;71:135–140.
  • Kreilgaard M, Kemme MJ, Burggraaf J, Schoemaker RC, Cohen AF. Influence of a microemulsion vehicle on cutaneous bioequivalence of a lipophilic model drug assessed by microdialysis and pharmacodynamics. Pharm Res 2001;18:593–599.
  • Kreilgaard M. Dermal pharmacokinetics of microemulsion formulations determined by in vivo microdialysis. Pharm Res 2001;18:367–373.
  • Lehmann L, Keipert S, Gloor M. Effects of microemulsions on the stratum corneum and hydrocortisone penetration. Eur J Pharm Biopharm 2001;52:129–136.
  • Kreilgaard M, Pedersen EJ, Jaroszewski JW. NMR characterisation and transdermal drug delivery potential of microemulsion systems. J Control Release 2000;69:421–433.
  • Ozer O, Baloglu E, Ertan G, Muguet V, Yazan Y. The effect of the type and the concentration of the lipophilic surfactant on the stability and release kinetics of the W/O/W multiple emulsions. Int J Cosmet Sci 2000;22:459–470.
  • Khan AY, Talegaonkar S, Iqbal Z, Ahmed FJ, Khar RK. Multiple emulsions: an overview. Curr Drug Deliv 2006;3:429–443.
  • Abrams K, Harvell JD, Shriner D, Wertz P, Maibach H, Maibach HI et al. Effect of organic solvents on in vitro human skin water barrier function. J Invest Dermatol 1993;101:609–613.
  • Gao S, Singh J. Effect of oleic/ethanol and oleic acid/propylene glycol on the in vitro percutaneous absorption of 5-fluorouracil and tamoxifen and the macroscopic barrier property of porcine epidermis. Int J Pharm 1998;165:45–55.
  • Senyigit T, Tekmen I, Sönmez U, Santi P, Ozer O. Deoxycholate hydrogels of betamethasone-17-valerate intended for topical use: In vitro and in vivo evaluation. Int J Pharm 2011;403:123–129.
  • Levin J, Maibach H. The correlation between transepidermal water loss and percutaneous absorption: an overview. J Control Release 2005;103:291–299.
  • Sintov A, Ze’evi A, Uzan R, Nyska A. Influence of pharmaceutical gel vehicles containing oleic acid/sodium oleate combinations on hairless mouse skin, a histological evaluation. Eur J Pharm Biopharm 1999;47:299–303.
  • Ozer O, Ozyazici M, Tedajo M, Taner MS, Köseoglu K. W/O/W multiple emulsions containing nitroimidazole derivates for vaginal delivery. Drug Deliv 2007;14:139–145.
  • Zhao X, Liu JP, Zhang X, Li Y. Enhancement of transdermal delivery of theophylline using microemulsion vehicle. Int J Pharm 2006;327:58–64.
  • Djordjevic L, Primorac M, Stupar M. In vitro release of diclofenac diethylamine from caprylocaproyl macrogolglycerides based microemulsions. Int J Pharm 2005;296:73–79.
  • Draelos ZD, Matsubara A, Smiles K. The effect of 2% niacinamide on facial sebum production. J Cosmet Laser Ther 2006;8:96–101.
  • U.S. Pharmacopeia XXII, Official Monographs, Niacinamide, 944.
  • Validation of analytical procedures. Proceedings of International Conference on Harmonisation (ICH). Commission of European Communities, 1996.
  • Touitou E, Godin B, Karl Y, Bujanover S, Becker Y. Oleic acid, a skin penetration enhancer, affects Langerhans cells and corneocytes. J Control Release 2002;80:1–7.
  • Fang JY, Leu YL, Wang YY, Tsai YH. In vitro topical application and in vivo pharmacodynamic evaluation of nonivamide hydrogels using Wistar rat as an animal model. Eur J Pharm Sci 2002;15:417–423.
  • Kreilgaard M. Influence of microemulsions on cutaneous drug delivery. Adv Drug Deliv 2002;1:77–98.
  • Chen H, Chang X, Weng T, Zhao X, Gao Z, Yang Y et al. A study of microemulsion systems for transdermal delivery of triptolide. J Control Release 2004;98:427–436.
  • Kale NJ, Allen Jr. LV. Studies o microemulsions using Brij 96 as surfactant and glycerin, ethylene glycol and propylene glycol as cosurfactants. Int J Pharm 1989;57:87–93.
  • Ayannides CA, Ktistis G. A rheological study on microemulsion gels of isopropyl myristate, polysorbate 80, glycerol and water. J Cosmet Sci 1999;50:1–7.
  • Yue Y, San-Ming L, Pan D, Da-Fang Z. Physicochemical properties and evaluation of microemulsion systems for transdermal delivery of meloxicam. Chem Res Chinese 2007;23:81–86.
  • Lin SS, Hsleh AL, Min DBS, Chang SS. A study of the color stability of commercial oleic acid. J Am Oil Chem Soc 1976;53:157–161.
  • Tanno O, Ota Y, Kitamura N, Katsube T, Inoue S. Nicotinamide increases biosynthesis of ceramides as well as other stratum corneum lipids to improve the epidermal permeability barrier. Br J Dermatol 2000;143:524–531.
  • Soma Y, Kashima M, Imaizumi A, Takahama H, Kawakami T, Mizoguchi M. Moisturizing effects of topical nicotinamide on atopic dry skin. Int J Dermatol 2005;44:197–202.
  • Tanojo H, Boelsma E, Junginger HE, Ponec M, Boddé HE. In vivo human skin permeability enhancement by oleic acid: a laser Doppler velocimetry study. J Control Release 1999;58:97–104.

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