Permeability enhancing lipid-based co-solvent and SEDDS formulations of SQ641, an antimycobacterial agent

References

• Zalavadiya P, Tala S, Akbari J, Joshi H. Multi-component synthesis of dihydropyrimidines by iodine catalyst at ambient temperature and in-vitro antimycobacterial activity. Arch Pharm (Weinheim) 2009;342:469–475
   PubMed Web of Science ®Google Scholar
• The WHO/IUATLD Global Project on Anti-tuberculosis Drug Resistance Surveillance 1999–2002: Anti-tuberculosis Drug Resistance in the World; Report No. 3. Available from: http://whqlibdoc.who.int/publications/2004/9241562854_foreword_summary.pdf [last accessed 8 May 2013]
   Google Scholar
• Koga T, Fukuoka T, Doi N, et al. Activity of capuramycin analogues against Mycobacterium tuberculosis, Mycobacterium avium and Mycobacterium intracellulare in vitro and in vivo. J Antimicrob Chemother 2004;54:755–760
   PubMed Web of Science ®Google Scholar
• Reddy VM, Einck L, Nacy CA. In vitro antimycobacterial activities of capuramycin analogues. Antimicrob Agents Chemother 2008;52:719–721
   PubMed Web of Science ®Google Scholar
• Aungst BJ. Novel formulation strategies for improving oral bioavailability of drugs with poor membrane permeation or presystemic metabolism. J Pharm Sci 1993;82:979–987
   PubMed Web of Science ®Google Scholar
• Kommuru TR, Gurley B, Khan MA, Reddy IK. Self-emulsifying drug delivery systems (SEDDS) of coenzyme Q10: formulation development and bioavailability assessment. Int J Pharm 2001;212:233–246
   PubMed Web of Science ®Google Scholar
• Robinson JR. Introduction: semi-solid formulations for oral drug delivery. Bull Tech Gattefosse 1996;89:11–13
   Google Scholar
• Vasconcelos T, Sarmento B, Costa P. Solid dispersions as strategy to improve oral bioavailability of poor water soluble drugs. Drug Discov Today 2007;12:1068–1075
   PubMed Web of Science ®Google Scholar
• Gursoy RN, Benita S. Self-emulsifying drug delivery systems (SEDDS) for improved oral delivery of lipophilic drugs. Biomed Pharmacother 2004;58:173–182
   PubMed Web of Science ®Google Scholar
• Kang BK, Lee JS, Chon SK, et al. Development of self-microemulsifying drug delivery systems (SMEDDS) for oral bioavailability enhancement of simvastatin in beagle dogs. Int J Pharm 2004;274:65–73
   PubMed Web of Science ®Google Scholar
• Patel AR, Vavia PR. Preparation and in vivo evaluation of SMEDDS (self-microemulsifying drug delivery system) containing fenofibrate. AAPS J 2007;9:E344–E352
   PubMed Web of Science ®Google Scholar
• Pouton CW, Outon CW. Formulation of self-emulsifying drug delivery systems. Adv Drug Deliv Rev 1997;25:47–58
   Web of Science ®Google Scholar
• Pouton CW. Lipid formulations for oral administration of drugs: non-emulsifying, self-emulsifying and ‘self-microemulsifying’ drug delivery systems. Eur J Pharm Sci 2000;11:S93–S98
   PubMed Web of Science ®Google Scholar
• Tarr BD, Yalkowsky SH. Enhanced intestinal absorption of cyclosporine in rats through the reduction of emulsion droplet size. Pharm Res 1989;6:40–43
   PubMed Web of Science ®Google Scholar
• Lundin PD, Bojrup M, Ljusberg-Wahren H, et al. Enhancing effects of monohexanoin and two other medium-chain glyceride vehicles on intestinal absorption of desmopressin (dDAVP). J Pharmacol Exp Ther 1997;282:585–590
   PubMed Web of Science ®Google Scholar
• Swenson ES, Curatolo WJ. Means to enhance penetration. Adv Drug Deliv Rev 1992;8:39–42
   Web of Science ®Google Scholar
• Constantinides PP. Lipid microemulsions for improving drug dissolution and oral absorption: physical and biopharmaceutical aspects. Pharm Res 1985;12:161–172
   Google Scholar
• Prabhu S, Ortega M, Ma C. Novel lipid-based formulations enhancing the in vitro dissolution and permeability characteristics of a poorly water-soluble model drug, piroxicam. Int J Pharm 2005;301:209–216
   PubMedGoogle Scholar
• Lindmark T, Nikkila T, Artursson P. Mechanisms of absorption enhancement by medium chain fatty acids in intestinal epithelial Caco-2 cell monolayers. J Pharmacol Exp Ther 1995;275:958–964
   PubMed Web of Science ®Google Scholar
• Sha X, Yan G, Wu Y, et al. Effect of self-microemulsifying drug delivery systems containing Labrasol on tight junctions in Caco-2 cells. Eur J Pharm Sci 2005;24:477–486
   PubMed Web of Science ®Google Scholar
• Lo YL, Hsu CY, Huang JD. Comparison of effects of surfactants with other MDR reversing agents on intracellular uptake of epirubicin in Caco-2 cell line. Anticancer Res 1998;18:3005–3009
   PubMed Web of Science ®Google Scholar
• Nerurkar MM, Burton PS, Borchardt RT. The use of surfactants to enhance the permeability of peptides through Caco-2 cells by inhibition of an apically polarized efflux system. Pharm Res 1996;13:528–534
   PubMed Web of Science ®Google Scholar
• Yu L, Bridgers A, Polli J, et al. Vitamin E-TPGS increases absorption flux of an HIV protease inhibitor by enhancing its solubility and permeability. Pharm Res 1999;16:1812–1817
   PubMed Web of Science ®Google Scholar
• Hotoda H, Daigo M, Furukawa M, et al. Synthesis and antimycobacterial activity of capuramycin analogues. Part 2: Acylated derivatives of capuramycin-related compounds. Bioorg Med Chem Lett 2003;13:2833–2836
   PubMed Web of Science ®Google Scholar
• Giron D. Contribution of thermal methods and related techniques to the rational development of pharmaceuticals – Part 1. Pharm Sci Technol Today 1998;1:191–199
   Google Scholar
• Bond L, Allen S, Davies MC, et al. Differential scanning calorimetry and scanning thermal microscopy analysis of pharmaceutical materials. Int J Pharm 2002;243:71–82
   PubMed Web of Science ®Google Scholar
• Craig DQM, Barker SA, Banning D, Booth SW. An investigation into the mechanisms of self-emulsification using particle size analysis and low frequency dielectric spectroscopy. Int J Pharm 1995;114:103–110
   Web of Science ®Google Scholar
• Ungell AL, Nylander S, Bergstrand S, et al. Membrane transport of drugs in different regions of the intestinal tract of the rat. J Pharm Sci 1998;87:360–366
   PubMed Web of Science ®Google Scholar
• Balimane PV, Chong S, Morrison RA. Current methodologies used for evaluation of intestinal permeability and absorption. J Pharmacol Toxicol Methods 2000;44:301–312
   PubMed Web of Science ®Google Scholar