Skin deposition and permeation of finasteride in vitro: effects of propylene glycol, ethanol and sodium lauryl sulfate

References

• Libecco JF, Bergfeld WF. Finasteride in the treatment of alopecia. Expert Opin Pharmacother 2004;5:933–940
   PubMed Web of Science ®Google Scholar
• Sintov A, Serafimovich S, Gilhar A. New topical antiandrogenic formulations can stimulate hair growth in human bald scalp grafted onto mice. Int J Pharm 2000;194:125–134
   PubMed Web of Science ®Google Scholar
• Drake L, Hordinsky M, Fiedler V, et al. The effect of finasteride on scalp skin and serum androgen levels in men with androgenetic alopecia. J Am Acad Dermatol 1999;41:550–554
   PubMed Web of Science ®Google Scholar
• Mazzarella F, Loconsole F, Cammisa A, et al. Topical finasteride in the treatment of andrognic alopecia. Preliminary evaluations after a 16-month therapy course. J Dermatol Treat 1997;8:189–192
   Web of Science ®Google Scholar
• Ye F, Imamura K, Imanishi N, et al. Effects of topical antiandrogen and 5-alpha-reductase inhibitors on sebaceous glands in male fuzzy rats. Skin Pharmacol 1997;10:288–297
   PubMedGoogle Scholar
• Rao Y, Zheng F, Zhang X, et al. In Vitro percutaneous permeation and skin accumulation of finasteride using vesicular ethosomal carriers. AAPS PharmSciTech 2008;9:860–865
   PubMed Web of Science ®Google Scholar
• Kalia YN, Guy RH. Modeling transdermal drug release. Adv Drug Deliv Rev 2001;48:159–172
   PubMed Web of Science ®Google Scholar
• Barry BW. Lipid-protein-partitioning theory of skin penetration enhancement. J Control Release 1991;15:237–248
   Web of Science ®Google Scholar
• Williams AC, Barry BW. Penetration enhancers. Adv Drug Deliv Rev 2004;56:603–618
   PubMed Web of Science ®Google Scholar
• Tabbakhian M, Tavakoli N, Jaafari MR, Daneshamouz S. Enhancement of follicular delivery of finasteride by liposomes and niosomes: 1. In vitro permeation and in vivo deposition studies using hamster flank and ear models. Int J Pharm 2006;323:1–10
   PubMed Web of Science ®Google Scholar
• Javadzadeh Y, Shokri J, Hallaj-Nezhadi S, et al. Enhancement of percutaneous absorption of finasteride by cosolvents, cosurfactant and surfactants. Pharm Dev Technol 2010;15:619–625
   PubMed Web of Science ®Google Scholar
• Caon T, Porto LC, Granada A, et al. Chitosan-decorated polystyrene-b-poly(acrylic acid) polymersomes as novel carriers for topical delivery of finasteride. Eur J Pharm Sci 2014;52:165–172
   PubMed Web of Science ®Google Scholar
• Daneshamouz S, Tabbakhian M, Tavakoli N, Jaafari MR. Influence of liposomes and niosomes on the in vitro permeation and skin retention of finasteride. Iran J Pharm Sci 2005;1:119–130
   Google Scholar
• Biruss B, Valenta C. Skin permeation of different steroid hormones from polymeric coated liposomal formulations. Eur J Pharm Biopharm 2006;62:210–219
   PubMed Web of Science ®Google Scholar
• Tuntiyasawasdikul S, Limpongsa E, Jaipakdee N, Sripanidkulchai B. Transdermal permeation of kaempferia parviflora methoxyflavones from isopropyl myristate-based vehicles. AAPS PharmSciTech 2014;15:947–955
   PubMed Web of Science ®Google Scholar
• Borràs-Blasco J, López A, Morant MJ, et al. Influence of sodium lauryl sulphate on the in vitro percutaneous absorption of compounds with different lipophilicity. Eur J Pharm Sci 1997;5:15–22
   Web of Science ®Google Scholar
• Herkenne C, Naik A, Kalia, YN, et al. Effect of propylene glycol on ibuprofen absorption into human skin in vivo. J Pharm Sci 2008;97:185–197
   PubMed Web of Science ®Google Scholar
• Nokhodchi A, Shokri J, Dashbolaghi A, et al. The enhancement effect of surfactants on the penetration of lorazepam through rat skin. Int J Pharm 2003;250:359–369
   PubMed Web of Science ®Google Scholar
• Panchagnula R, Salve PS, Thomas NS, et al. Transdermal delivery of naloxane: effect of water, propylene glycol, ethanol and their binary combinations on permeation through rat skin. Int J Pharm 2001;219:95–105
   PubMed Web of Science ®Google Scholar
• Watkinson RM, Guy RH, Hadgraft J, Lane ME. Optimisation of cosolvent concentration for topical drug delivery – II: influence of propylene glycol on ibuprofen permeation. Skin Pharmacol Physiol 2009;22:225–230
   PubMed Web of Science ®Google Scholar
• Watkinson RM, Herkenne C, Guy RH, et al. Influence of ethanol on the solubility, ionization and permeation characteristics of ibuprofen in silicone and human skin. Skin Pharmacol Physiol 2009;22:15–21
   PubMed Web of Science ®Google Scholar
• Bhatia KS, Gao S, Singh J. Effect of penetration enhancers and iontophoresis on the FT-IR spectroscopy and LHRH permeability through porcine skin. J Control Release 1997;47:81–89
   Web of Science ®Google Scholar
• Tseng RL, Wu FC, Juang RS. Characteristics and applications of the Lagergren’s first-order equation for adsorption kinetics. J Taiwan Inst Chem Eng 2010;41:661–669
   Web of Science ®Google Scholar
• Anissimov YG, Roberts MS. Diffusion modeling of percutaneous absorption kinetics: 4. Effects of a slow equilibration process within stratum corneum on absorption and desorption kinetics. J Pharm Sci 2009;98:772–781
   PubMed Web of Science ®Google Scholar
• Cestari AR, Vieira EFS, Matos JDS, dos Anjos DSC. Determination of kinetic parameters of Cu(II) interaction with chemically modified thin chitosan membranes. J Colloid Interface Sci 2005;285:288–295
   PubMed Web of Science ®Google Scholar
• Mitragotri S, Anissimov YG, Bunge AL, et al. Mathematical model of skin permeability: an overview. Int J Pharm 2011;418:115–129
   PubMed Web of Science ®Google Scholar
• Hansch C, Leo A, Hoekman D. In exploring QSAR: hydrophobic, electronic and steric constants. Washington, DC: American Chemical Society; 1995
   Google Scholar
• Florence AT, Attwood D. Physicochemical principles of pharmacy. 4th ed. London: Pharmaceutical Press; 2006
   Google Scholar
• Rowe RC, Sheskey PJ, Quinn ME. Handbook of pharmaceutical excipients. 6th ed. Gurnee (IL): Pharmaceutical Press; 2009
   Google Scholar
• Bolzinger M-A, Briançon S, Pelletier J, Chevalier Y. Penetration of drugs through skin, a complex rate-controlling membrane. Curr Opin Colloid In 2012;17:156–165
   Web of Science ®Google Scholar
• Shen L-N, Zhang Y-T, Wang Q, et al. Enhanced in vitro and in vivo skin deposition of apigenin delivered using ethosomes. Int J Pharm 2014;460:280–288
   PubMed Web of Science ®Google Scholar
• Yang Z, Teng Y, Wang H, Hou H. Enhancement of skin permeation of bufalin by limonene via reservoir type transdermal patch: formulation design and biopharmaceutical evaluation. Int J Pharm 2013;447:231–240
   PubMed Web of Science ®Google Scholar
• Valia KH, Chien YW, Shinal EC. Long-term skin permeation kinetics of estradiol (I): effect of drug solubilizer-polyethylene glycol 400. Drug Dev Ind Pharm 1984;10:951–981
   Web of Science ®Google Scholar
• Addicks WJ, Flynn GL, Weiner ND, Curl RL. Drug delivery from topical formulations: theoretical prediction and experimental assessment. In: Osborne DW, Amann AH, eds. Topical drug delivery formulations. New York: Marcel Dekker; 1990:221–244
   Google Scholar
• Bommannan D, Potts RO, Guy RH. Examination of the effect of ethanol on human stratrum corneum in vivo using infrared spectroscopy. J Control Release 1991;16:299–304
   Web of Science ®Google Scholar
• Pershing LK, Silver BS, Krueger GG, et al. Feasibility of measuring the bioavailability of topical betamethaosne dipropionate in commercial formulations using drug content in skin and skin blanching assay. Pharm Res 1992;9:45–51
   PubMed Web of Science ®Google Scholar
• Ribaud C, Garson JC, Doucet J, Lévêque JL. Organization of stratum corneum lipids in relation to permeability: influence of sodium lauryl sulfate and preheating. Pharm Res 1994;11:1414–1418
   PubMed Web of Science ®Google Scholar
• Van der Merwe D, Riviere JE. Effect of vehicles and sodium lauryl sulphate on xenobiotic permeability and stratum corneum partitioning in porcine skin. Toxicology 2005;206:325–335
   PubMed Web of Science ®Google Scholar
• Méndez-Díaz JD, Prados-Joya G, Rivera-Utrilla J, et al. Kinetic study of the adsorption of nitroimidazole antibiotics on activated carbons in aqueous phase. J Colloid Interface Sci 2010;345:481–490
   PubMed Web of Science ®Google Scholar
• Lee CK, Uchida T, Kazuhisa K, et al. Skin permeability of various drugs with different lipophilicity. J Pharm Sci 1994;83:562–565
   PubMed Web of Science ®Google Scholar
• Gibbs S, Vietsch H, Meier U, Ponec M. Effect of skin barrier competence on SLS and water-induced IL-1α expression. Exp Dermatol 2002;11:217–223
   PubMed Web of Science ®Google Scholar
• Lee CH, Maibach HI. Sodium lauryl sulfate. In: Chew A-L, Maibach HI, eds. Irritant dermatitis. Berlin: Springer-Verlag; 2006:257–267
   Google Scholar