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Research Article

Evaluation of physico-mechanical properties of drug-excipients agglomerates obtained by crystallization

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Pages 243-249 | Received 20 Oct 2009, Accepted 11 Jan 2010, Published online: 22 Feb 2010

References

  • Chelakara LV, Sushrut KK, Dhanashri RK. Spherical agglomeration of mefenamic acid and nabumetone to improve micromeritics and solubility. AAPS. PharmSciTech. 2006;7(2):1–8.
  • Maghsoodi M, Hassan-zadeh D, Barzegar-jalali M, Nokhodchi A, Martin G. Improved compaction and packing properties of naproxen agglomerated crystals obtained by spherical crystallization technique. Drug Dev Ind Pharm. 2007;33:1216–1224.
  • Venkadarirammohan G, Sprinivas M, Madhobhai MP, Girish KJ. Spherical crystals of celecoxib to improve solubility, dissolution rate and micromeritic properties. Acta Pharm. 2007;57:173–184.
  • Kawashima Y, Lin Y, Ogawa M, HanDA T, Takenaka H. Prolonged release microcapsules of indomethacin through spherical crystallization technique. J Pharm Sci. 1985;74:1152–1156.
  • Guillaume F, Guyothermann AM, Guyot JC. Spherical crystallization of meprobamate. Farmaco. 1993;48:473–485.
  • Di Martino P, Barthelemy C, Piva F, Joiris E, Palmieri GE, Martelli S. Improved dissolution behavior of fenobufen by spherical crystallization. Drug Dev Ind Pharm. 1999;25: 1073–1081.
  • Kadam SS, Mahadik KR, Paradkar AR. A process for making agglomerates for use as or in a drug delivery system. Indian patent. 183036; 1997.
  • Kadam SS, Mahandik KR, Paradkar AR. A process for making agglomerates for use as or in a drug delivery system. Indian patent. 183481; 1997.
  • Maghsoodi M, Taghizadeh O, Martin G, Nokhodchi A. Particle design of naproxen-disintegrant agglomerates for direct compression by a crystallo-co-agglomeration technique. Int J Pharm. 2008;351:45–54.
  • Nokhodchi A, Maghsoodi M, Hassan-Zadeh D, Barzegar-Jalali M. Preparation of agglomerated crystals for improving flowability and compactibility of poorly flowable and compatible drugs and excipients. Powder Technol. 2007;175:73–81.
  • Pilpel N. The flow properties of magnesia. J Pharm Pharmacol. 1964;16:705–716.
  • Carr RL. Evaluation flow properties of solids. Chem Eng. 1965; 72:163–168.
  • Carr RL. Classify flow properties of solids. Chem Eng. 1965; 72:69–72.
  • Kawashima Y, Handa T, Takeuchi H, Okumara M, Katou H, Nagata O. Crystal modification of phenytoin with polyethylene glycol for improving mechanical strength, dissolution rate and bioavailability by spherical crystallization technique. Chem Pharm Bull. 1986;34:3376–3383.
  • Kawashima Y, Handa T, Takeuchi H, Okumura M. Effect of polyethylene glycol on size of agglomerated crystals of phenytoin prepared by the spherical crystallization technique. Chem Pharm Bull. 1986;34: 3403–3407.
  • Morishima K, Kawashima Y, Takeuchi H, Niwa T, Hino T. Micromeritic characteristics and agglomeration mechanisms in the spherical crystallization of bucillamine by the spherical agglomeration and the emulsion solvent diffusion methods. Powder Technol. 1993;76:57–64.
  • Paradkar AR, Pawar AP, Chordiya JK. Spherical crystallization of celecoxib. Drug Dev Ind Pharm. 2002;28:1213–1220.
  • Morishima K, Kawashima Y, Takeuchi H, Niwa T, Hino T. Spherical crystallization of celecoxib to improve solubility, dissolution rate and micromeritic properties. Acta Pharm. 2007:57:173–184.
  • Sethia S, Squillante E. Physicochemical characterization of solid dispersions of carbamazepine formulated by supercritical carbon dioxide and conventional solvent evaporation method. J Pharm Sci. 2002;91:1984–1957.
  • Krahn FU, Mielck JB. Relations between several polymorphic forms and the dihydrate of carbamazepine. Pharm Acta Helv. 1987;62:248–254.
  • Lowes MMJ, Caira MR, Lo”ter AP, Van Der Watt JG. Physico-chemical properties and X-ray structure studies of the trigonal polymorph of carbamazepine. J Pharm Sci. 1987;76:744–752.
  • Rustichelli C, Gamberini G, Ferioli V, Gamberini MC, Ficarra R, Tommasini S. Solid-state of polymorphic drug: Carbamazepine. J Pharm Biomed Anal. 2000;23:41–54.
  • Edwards AD, Shekunov BY, Kordikowski A, Forbes RT, York P. Crystallization of pure anhydrous polymorphs of carbamazepine by solution enhanced dispersion with supercritical fluids (SEDSe). J Pharm Sci. 2001;90:1115–1124.
  • Zhao N, Augsburger L. The influence of product brand-to-brand variability on superdisintegrant performance: A case study with croscarmellose sodium. Pharm Dev Technol. 2006;11:79–185.
  • Shah U, Augsburger L. Evaluation of the functional equivalence of crospovidone NF from different sources. II Standard performance test. Pharm Dev Technol. 2001;6:419–430.
  • Lopez-Solisa J, Villafuerte-Roblesa L. Effect of disintegrants with different hygroscopicity on dissolution of norfloxacin: Pharmatose DCL 11 tablets. Int J Pharm. 2001;216:127–135.
  • Gordon MS, Chowhan ZT. Effect of tablet solubility and hygroscopicity on disintegrant efficiency in direct compression tablets intem of dissolution. J Pharm Sci. 1987;76:907–909.
  • Johnson JR, Wang LH, Gordon MS, Chowhan ZT. Effect of formulation solubility and hygroscopicity on desentegration efficiency in tablet prepared by wet granulation intem of dissolution. J Pharm Sci. 1991;80:469–471.
  • Jbiilou M, Ettabia A, Gguyot-Hermann AM, Guyot JC. Ibuprofen agglomerates preparation by phase sepration. Drug Dev Ind Pharm. 1999;25:297–305.
  • Kobayashi Y, Ito S, Itai S, Yamamoto K. Physicochemical properties and bioavailability of carbamazepine polymorphs and dehydrate. Int J Pharm. 2000;193:137–146.
  • Tian F, Sandler N, Aaltonen J, Lang C, Saville DJ, Gordon KC, Strachan CJ, Rantanen J, Rades T. Influence of polymorphic form, morphology, and excipient interactions on the dissolution of carbamazepine compacts. J Pharm Sci. 2007;96(3):584–594.

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