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Research Article

Thermal solvent-free synthesis of chromonyl chalcones, pyrazolines and their in vitro antibacterial, antifungal activities

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Pages 84-91 | Received 11 Dec 2010, Accepted 29 Mar 2011, Published online: 25 May 2011

References

  • Oliveira RDR, Maffei CML, Martinez R. Infecção urinária hospitalar por leveduras do gênero Candida. Rev Assoc Med Bras 2001;47:231–235.
  • Diekema DJ, BootsMiller BJ, Vaughn TE, Woolson RF, Yankey JW, Ernst EJ et al. Antimicrobial resistance trends and outbreak frequency in United States hospitals. Clin Infect Dis 2004;38:78–85.
  • Georgopapadakou NH. Infectious disease 2001: drug resistance, new drugs. Drug Resist Updat 2002;5:181–191.
  • Zhang W, Berberov EM, Freeling J, He D, Moxley RA, Francis DH. Significance of heat-stable and heat-labile enterotoxins in porcine colibacillosis in an additive model for pathogenicity studies. Infect Immun 2006;74:3107–3114.
  • Shaheen HI, Khalil SB, Rao MR, Abu Elyazeed R, Wierzba TF, Peruski LF Jr et al. Phenotypic profiles of enterotoxigenic Escherichia coli associated with early childhood diarrhea in rural Egypt. J Clin Microbiol 2004;42:5588–5595.
  • Puerto AS, Fernández JG, del Castillo Jde D, Pino MJ, Angulo GP. In vitro activity of beta-lactam and non-beta-lactam antibiotics in extended-spectrum beta-lactamase-producing clinical isolates of Escherichia coli. Diagn Microbiol Infect Dis 2006;54:135–139.
  • Nolan CM, Chalhub EG, Nash DG, Yamauchi T. Treatment of bacterial meningitis with intravenous amoxicillin. Antimicrob Agents Chemother 1979;16:171–175.
  • Harbottle H, Thakur S, Zhao S, White DG. Genetics of antimicrobial resistance. Anim Biotechnol 2006;17:111–124.
  • Berger S. Incidence of severe side effects during therapy with sulfonylurea and biguanides. Horm Metab Res 1985;17:111–115.
  • Barton D, Ollis WD. (1979). Comprehensive Organic Chemistry,vol 1–6. Oxford: Pergamon.
  • Chemler YY, Leonard E, Koffas MAG. Combinatorial mutasynthesis of flavonoid analogues from acrylic acids in microorganisms. Org Lett 2007;9:1855–1858.
  • Prakash O, Kumar R, Parkash V. Synthesis and antifungal activity of some new 3-hydroxy-2-(1-phenyl-3-aryl-4-pyrazolyl) chromones. Eur J Med Chem 2008;43:435–440.
  • Kuroda M, Uchida S, Watanabe K, Mimaki Y. Chromones from the tubers of Eranthis cilicica and their antioxidant activity. Phytochemistry 2009;70:288–293.
  • Larget R, Lockhart B, Renard P, Largeron M. A convenient extension of the Wessely-Moser rearrangement for the synthesis of substituted alkylaminoflavones as neuroprotective agents in vitro. Bioorg Med Chem Lett 2000;10:835–838.
  • Yu D, Chen CH, Brossi A, Lee KH. Anti-AIDS agents. 60. Substituted 3′R,4′R-di-O-(-)-camphanoyl-2′,2′-dimethyldihydropyrano[2,3-f]chromone (DCP) analogues as potent anti-HIV agents. j Med Chem 2004;47:4072–4082.
  • Valenti P, Bisi A, Rampa A, Belluti F, Gobbi S, Zampiron A et al. Synthesis and biological activity of some rigid analogues of flavone-8-acetic acid. Bioorg Med Chem 2000;8:239–246.
  • Horton DA, Bourne GT, Smythe ML. The combinatorial synthesis of bicyclic privileged structures or privileged substructures. Chem Rev 2003;103:893–930.
  • Nowaskowska Z. A review of anti-infective and anti-inflammatory chalcones. Eur J Med Chem 2007;42:125–137.
  • Acharya BN, Saraswat D, Tiwari M, Shrivastava AK, Ghorpade R, Bapna S et al. Synthesis and antimalarial evaluation of 1, 3, 5-trisubstituted pyrazolines. Eur J Med Chem 2010;45:430–438.
  • Tanaka K, Toda F. Solvent-free organic synthesis. Chem Rev 2000;100:1025–1074.
  • Cave GW, Raston CL, Scott JL. Recent advances in solventless organic reactions: towards benign synthesis with remarkable versatility. Chem Commun (Camb) 2001;2159:2169.
  • Toda F. (2005). Solid State Reaction topics in Current Organic Chemistry. Berlin, Heidelberg, New York: Springer.
  • Wang GW. (2004). Fullerene Mechanochemistry. In: Nalwa HS, ed. Encyclopedia of Nanoscience and Nanotechnology, vol. 3. Stevenson Ranch: American Scientific Publishers, 557.
  • Nohara A, Umetani T, Sanno Y. A facile synthesis of 4-oxo-4H-1-benzopyran-3- carboxaldehydes by vilsmeier reagents. Tetrahedron 1974;30:3353–3561.
  • Singh SP, Sehgal S, Tarar LS, Dhawan SN. Synthesis of 2-[3-methyl or trifluromethyl-5-(2-thienyl)-pyrazol-1-yl]thiazol and benzothiazoles. Indian J Chem 1990;29B:310–314.
  • Jursic BS, Neumann DM. Preparation of 5-formyl and 5-acetyl barbituric acids, including the corresponding Schiff bases and phenyl hydrazones. Tetrahedron Lett 2001;42:8435–8439.
  • Cruickshank R, Duguid JP, Marmion BP, Swain RHA. (1975). Medicinal Microbiology. 12th edn, vol. II, London: Churchill Livingstone, 196–202.
  • Collins AH. (1976). In: Microbiological Methods, second edn. London: Butterworth.
  • Khan ZK. In vitro and vivo screening techniques for bioactivity screening and evaluation, Proc Int Workshop UNIDO-CDRI 1997:210–211.
  • Varma RS.(1998). Antifungal Agents: Past, Present and Future prospects. Lucknow, India: National Academy of Chemistry & Biology.
  • Wiley RH, Jarboe CH. The Chemistry of Heterocyclic compounds. Interscience, NY: 1967;22:183.

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