References
- Smyth DG, Nagamatsu A, Fruton JS. Some reactions of N-ethylmaleimide. J Am. Chem Soc 1960;82:4600–4804.
- Han KK, Delacourte A, Hemon B. Chemical modification of thiol group(s) in protein: Application to the study of anti-microtubular drugs binding. Comp Biochem Physiol, B 1987;88:1057–1065.
- Shaw E. Cysteinyl proteinases and their selective inactivation. Adv Enzymol Relat Areas Mol Biol 1990;63:271–347.
- Matuszak N, Muccioli GG, Labar G, Lambert DM. Synthesis and in vitro evaluation of N-substituted maleimide derivatives as selective monoglyceride lipase inhibitors. J Med Chem 2009;52:7410–7420.
- Takatori K, Hasegawa T, Nakano S, Kitamura J, Kato N. Antifungal activities of N-substituted maleimide derivatives. Microbiol Immunol 1985;29:1237–1241.
- Igarashi Y, Yagami K, Imai R, Watanabe S. Antimicrobial activities of some N-aklylmaleimides. J Industr Microbiol 1990;6:223–225.
- Zentz F, Valla A, Le Guillou R, Labia R, Mathot AG, Sirot D. Synthesis and antimicrobial activities of N-substituted imides. Farmaco 2002;57:421–426.
- Sortino M, Cechinel Filho V, Corrêa R, Zacchino S. N-Phenyl and N-phenylalkyl-maleimides acting against Candida spp.: Time-to-kill, stability, interaction with maleamic acids. Bioorg Med Chem 2008;16:560–568.
- López SN, Castelli MV, de Campos F, Corrêa R, Cechinel Filho V, Yunes RA, Zamora MA, Enriz RD, Ribas JC, Furlán RL, Zacchino SA. In vitro antifungal properties structure-activity relationships and studies on the mode of action of N-phenyl, N-aryl, N-phenylalkyl maleimides and related compounds. Arzneimittelforschung 2005;55:123–132.
- Shults EE, Shakirov MM, Tolstikov GA, Kalinin VN, Schmidhammer G. Thebaine adducts with maleimides. Synthesis and transformations. Russian J Org Chem 2005;41:1132–1144.
- Coyle JD, Bryant LRB. Synthesis of diazaheterocycles with a bridgehead nitrogen by photocyclisation of N-substituted alicyclic imides. J Chem Soc Perkin Trans I 1983;2857–2865.
- Tetko IV, Tanchuk VY. Application of associative neural networks for prediction of lipophilicity in ALOGPS 2.1 program. J Chem Inf Comput Sci 2002;42:1136–1145.
- National Committee for Clinical Laboratory Standards. (2002). Reference method for broth dilution antifungal susceptibility testing of yeasts, 2nd edn. Approved standard M27-A2. Wayne, PA: NCCLS.
- Kippert F, Lloyd D. The aniline blue fluorochrome specifically stains the septum of both live and fixed Schizosaccharomyces pombe cells. FEMS Microbiol Lett 1995;132:215–219.
- Cabib E, Kang MS. Fungal 1,3-β-glucan synthase. Meth Enzymol 1987;138:637–642.
- Shedletzky E, Unger C, Delmer DP. A microtiter-based fluorescence assay for (1,3)-β-glucan synthases. Anal Biochem 1997;249:88–93.
- Munro CA, Schofield DA, Gooday GW, Gow NA. Regulation of chitin synthesis during dimorphic growth of Candida albicans. Microbiology (Reading, Engl) 1998;144:391–401.
- Bulawa CE, Slater M, Cabib E, Au-Young J, Sburlati A, Adair WL Jr, Robbins PW. The S. cerevisiae structural gene for chitin synthase is not required for chitin synthesis in vivo. Cell 1986;46:213–225.
- Gregory JD. The stability of N-ethylmaleimide and its reaction with sulfhydryl groups. J Am Chem Soc 1955;77:3922–3923.
- Niyaz Khan M. Kinetics and mechanism of the alkaline hydrolysis of maleimide. J Pharm Sci 1984;73:1767–1771.
- Georgopapadakou NH, Walsh TJ. Antifungal agents: Chemotherapeutic targets and immunologic strategies. Antimicrob Agents Chemother 1996;40:279–291.
- Bang KH, Lee DW, Park HM, Rhee YH. Inhibition of fungal cell wall synthesizing enzymes by trans-cinnamaldehyde. Biosci Biotechnol Biochem 2000;64:1061–1063.
- Frost DJ, Brandt K, Kaufmann T, Goldman R. Interaction of sulfhydryl reactive reagents with components involved in (1,3)-β-glucan synthesis from Candida albicans. Can J Microbiol 1995;41:692–698.
- Douglas CM. Fungal beta(1,3)-d-glucan synthesis. Med Mycol 2001;39 Suppl 1:55–66.
- Latgé JP. The cell wall: A carbohydrate armour for the fungal cell. Mol Microbiol 2007;66:279–290.
- López SN, Castelli MV, Zacchino SA, Domínguez JN, Lobo G, Charris-Charris J, Cortés JC, Ribas JC, Devia C, Rodríguez AM, Enriz RD. In vitro antifungal evaluation and structure-activity relationships of a new series of chalcone derivatives and synthetic analogues, with inhibitory properties against polymers of the fungal cell wall. Bioorg Med Chem 2001;9:1999–2013.
- Łącka I, Konieczny MT, Bułakowska A, Rzymowski T, Milewski, S. Antifungal action of the oxathiolone-fused chalcone derivative. Mycoses 2011 (in press). Available at: http://onlinelibrary.wiley.com/doi/10.1111/j.1439-0507.2010.01936.x/pdf
- Garcia-Effron G, Park S, Perlin DS. Correlating echinocandin MIC and kinetic inhibition of fks1 mutant glucan synthases for Candida albicans: Implications for interpretive breakpoints. Antimicrob Agents Chemother 2009;53:112–122.
- Friedmann E, Marrian DH, Simonreuss I. Antimitotic action of maleimide and related substances. Br J Pharmacol Chemother 1949;4:105–108.
- Matsui S, Yamazoe H, Watanabe I, Hayashi E, Konya K. [Studies on the experimental chemotherapy for dermatomycosis and candidiasis. IX. On the antifungal activity of various maleimide and succinimide compounds]. Yakugaku Zasshi 1984;104:1198–1206.