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Research Article

THA—A Review of the Literature and Its Use in Treatment of Five Overdose Patients

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Pages 269-281 | Published online: 25 Sep 2008

References

  • Slovis T. L., Ott J. E., Teitelbaum D. T., Lipscomb W. Physostigmine therapy in acute tricyclic antidepressant poisoning. Clin. Toxicol. 1972; 4: 451
  • Bernards W. Case History H74: Reversal of phenothiazine coma with physostigmine. Anesth. Analg. 1973; 52: 938
  • Brown M. L., Gershon S., Lang W. J., Korol B. Effects of psychomimetric response to Ditran in dogs. Arch. Int. Pharmacodyn. 1966; 160: 407
  • Burks J. S., Walker J. E., Rumack B. H., Ott J. E. Tricyclic antidepressant poisoning: Reversal of coma, choreoathetosis, and myoclonus by physostigmine. J. Am. Med. Assoc. 1974; 230: 1405
  • Coppolino C. A. Incidence of postanesthetic delirium in community hospital: A statistical study. Mil. Med. 1963; 28: 238
  • Crowell E. B., Ketchum J. S. Treatment of scopolamine‐induced delirium by physostigmine. Clin. Pharmacol. Therap. 1967; 8: 409
  • El‐Yousef M. K., Janowsky D., Davis J. M., Senkenke H. J. Reversal of anti‐Parkinsonian drug toxicity by physostigmine. Am. J. Psychiatry 1973; 130: 141
  • Granacher R. P., Baldessarine R. Physostigmine‐Its use in acute anticholinergic syndrome with antidepressant and anti‐Parkinson drugs. Arch. Gen. Psychiatry 1975; 32: 375
  • Heiser J. F., Gillin J. C. The reversal of anticholinergic drug induced delirium and coma with physostigmine. Am. J. Psychiatry 1971; 127: 1050
  • Heiser J. F., Wilbert D. E. Reversal of delirium induced by tricyclic antidepressant drugs with physostigmine. Am. J. Psychiatry 1974; 131: 1275
  • Janowsky D. S., Davis J. M., El‐Yousef M. K., Senkenke H. J. Combined anticholinergic agents and atropine‐like delirium. Am. J. Psychiatry 1972; 129: 360
  • Newton R. W. Physostigmine salicylate in the treatment of tricyclic antidepressant overdose. J. Am. Med. Assoc. 1975; 231: 941
  • Rasmussen J. Poisoning by amitriptyline, imipramine, and nortriptyline. Dan. Med. Bull. 1966; 13: 201
  • Rumack B. H. Anticholinergic poisoning treatment with physostigmine. Pediatrics 1972; 53: 449
  • Pharmacological Basis of Therapeutics5th ed., L. S. Goodman, A. Gilman. Macmillan, New York 1975
  • Vance M. A., Ross S. M., Millington W. R., Blumberg J. B. Potentiation of tricyclic antidepressant toxicity by physostigmine in mice. Clin. Toxicol. 1977; 11: 413
  • Bell C., Gershon S., Carrol B., Holan G. Behavioral antagonism to a new psychomimetic: JB‐329. Arch. Int. Pharmacodyn. 1964; 147: 9
  • Bell C., Gershon S. Experimental anticholinergic psychotomimetics: Antagonism of yohimbine and tecrine (THA). Med. Exp. 1964; 10: 15
  • Gershon S., Newbauer H., Sundland D. M. Ditran and its antagonistics in a mixed psychiatric population. J. Nerv. Ment. Dis. 1966; 142: 265
  • Gershon S. Behavioral effects of anticholinergic psychotomimetics and their antagonists in man and animals. Rec. Adv. Biol. Psychi. 1966; 13: 141
  • Itil T. M., Fink M. Anticholinergic drug induced delirium: Experimental modification, quantitative EEG, and behavioral correlation. J. Nerv. Ment. 1966; 143: 492
  • Itil T. M. Quantitative EEG changes induced by anticholinergic drugs and their behavioral correlates in man. Recent Adv. Biol. Psychiatry 1966; 13: 151
  • Gershon S., Olaria J. J.B.‐329‐A new psychotomimetic, its antagonism by tetrahydro aminoacridine and its comparison with LSD, mescaline, and sernyl. J. Neuropsychiatry 1960; 1: 283
  • Summers W. K. A clinical method for estimating risk of drug induced delirium. Life Sci. 1978; 22: 1511
  • Shaw F. H., Bentley G. Some aspects of the pharmacology of morphine with special reference to its antagonism by 5‐aminoacridine (THA) and other chemically related compounds. Med. J. Aust. 1949; 2: 868
  • Shaw F. H., Bentley G. A. Pharmacology of some new anticholinesterases. Aust. J. Exp. Biol. Med. Sci. 1953; 31: 573
  • Shaw F. H., Schulman A. Treatment of intractable pain with large doses of morphine and diamine phenylthiazole. Br. Med. J. 1955; 1: 1367
  • Stone V., Moon W., Shaw F. H. Treatment of intractable pain with morphine and THA. Br. Med. J. 1961; 1: 471
  • Rees J. M. H. Anticurare activity of tacrine (THA). J. Pharm. Pharmacol. 1966; 18: 289
  • McCaul K., Robinson G. D. Suxamethonium extension by tetrahydroaminoacrine. Br. J. Anaest. 1967; 39: 629
  • Ho A. K., Freeman S. E. Anticholinesterase activity by tetrahydroaminoacrine and succinylcholine hydrosis. Nature 1965; 205: 1118
  • Albin M. S., Orr M. D., Bunegin L. B., Henderson P. A. tetrahydroaminoacridine antagonism to narcotic addiction. Exp. Neurol. 1975; 46: 644
  • Albin M. S., Bunegin L., Massopust L. C., Jannetta P. J. Ketamine‐induced post‐anesthetic delirium attenuated by tetrahydroaminoacridine. Exp. Neurol. 1974; 44: 126
  • Albin M. S., Bunegin L., Jannetta P. J., Massopust L. C. tetrahydroaminoacridine (THA) I. Effect on post‐anesthetic emergence responses and anesthesia sleep‐time after ketamine, phencyclidine, and thiamylal in animals. Excerpta Med. Int. Congr. Ser. 1974; 347: 143
  • Maryani S., Weinstein H., Cohen S. Acetylcholine‐like molecular arrangement in psychotomimetic anticholinergic drugs. Proc. Natl. Acad. Sci. U.S. 1973; 70: 3103
  • Maryani S., Weinstein H., Ben‐Zue N., Cohen S., Sokolovsky M. Psychotomimetics as anticholinergic agents I. Cyclohexylpiperidine derivatives: Anticholinesterase activity and antagonistic activity to acetylcholine. Biochem. Pharmacol. 1974; 23: 1263
  • De La Lande I. S., Bentley G. The action of morphine and antagonists of the narcotic action of morphine on acetylcholine synthesis in brain. Aust. J. Exp. Biol. Med. Sci. 1955; 33: 555
  • De La Lande I. S., Porter R. S. The actions of tacrine (THA) and aminphenazole on acetylcholine metabolism in the guinea pig ileum. Aust. J. Exp. Biol. Med. Sci. 1963; 41: 149
  • Porter R. B. Some actions of tacrine on slow muscles of the toad (Bufo marinus) and the chick. Br. J. Pharmacol. 1965; 25: 179
  • Howland J. C., Carter M. K. The diuretic activity of tetrahydroaminoacridine in rats (34825). Proc. Soc. Exp. Biol. Med. 1970; 134: 513
  • Albert A. Improved synthesis of amino acridines. J. Soc. Chem. Ind. (Chem.) 1945; 65: 169
  • Heilbronn E. Inhibition of cholinesterases by tetrahydroaminoacridine. Acta Chem. Scand. 1961; 15: 1386
  • Kaul P. N. Enzyme inhibiting action of tetrahydroaminoacridine and its structural fragments. J. Pharm. Pharmacol. 1962; 14: 243
  • Hunter A. R. Tetrahydroaminoacridine in anesthesia. Br. J. Anaest. 1965; 37: 505
  • Rubbo S. D. Influence of chemical constitution on toxicity. Br. J. Exp. Pathol. 1947; 28: 1
  • Ungar J., Robinson F. A. Investigation of antibacterial and toxic actions of certain acridine derivatives. J. Pharmacol. Exp. Ther. 1944; 80: 217
  • Brodie D. E., Way E. L., Lowenhaupt E. Studies on 9‐aminoacridine antagonism of morphine and related drugs. Arch. Int. Pharmacodyn. 1952; 89: 1
  • Cristie G., Gershon S., Gray R., Shaw F. H., McCance I., Bruce D. W. Treatment of certain side effects of morphine. Br. Med. J. 1958; 1: 675
  • Crankshaw T. P. A Suxamethonium Potentiator. Presented at the Second World Congress of Anaesthesiologists, Toronto. 1960
  • Gordh T., Wahlin A. Potentiation of the neuromuscular effect of succinylcholine by tetrahydroaminoacridine. Acta Anaesthesiol. Scand. 1961; 5: 55
  • Gershon S., Shaw F. H. Tetrahydroaminoacrine as a decurarising agent. J. Pharm. Sci. 1958; 10: 638
  • Hunter A. R. An appraisal of tacrine‐extended suxamethonium. Br. J. Anaesth. 1970; 42: 155
  • Jones C. R., Davis M. Replacement drug for edrophonium bromide. Med. J. Aust. 1975; 2: 650
  • Albin M. S., Aguirre E. M., Albin R. L. Tetrahydroaminoacridine (THA) II. Modifications of post‐anesthetic emergence responses and anesthesia sleep‐time after ketamine hydrochloride (KH) in the human. Excerpta Med. Int. Congr. Ser. 1974; 347: 147
  • Mendelson G. Central anticholinergic syndrome reversed by tetrahydroaminoacrine (THA). Med. J. Aust. 1975; 1: 906

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