Synthesis of N-Arylinosines

Tokumi Maruyama Faculty of Pharmaceutical Sciences, Tokushima Bunri University, Yamashiro-cho, Tokushima, 770, JAPAN

Yoshiko Sato Faculty of Pharmaceutical Sciences, Tokushima Bunri University, Yamashiro-cho, Tokushima, 770, JAPAN

Takeshi Goto Faculty of Pharmaceutical Sciences, Tokushima Bunri University, Yamashiro-cho, Tokushima, 770, JAPAN

Mitsutoshi Fukuhara Faculty of Pharmaceutical Sciences, Tokushima Bunri University, Yamashiro-cho, Tokushima, 770, JAPAN

Abstract

2′,3′,5′-Tri-O(tetrahydropyran-2-yl)inosine 1 was treated with iodobenzene or 2-bromopyridine in the presence of cuprous oxide in pyridines to give the N¹ -aryl derivatives 2a, b. Deprotection of the products afforded N¹ -arylinosines 3a, b.

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Synthesis of N-Arylinosines

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Synthesis of N-Arylinosines

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