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Organic Preparations and Procedures International
The New Journal for Organic Synthesis
Volume 34, 2002 - Issue 5
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OPPI BRIEFS

A SIMPLIFIED SYNTHESIS OF ETHYL 5-CHLORO-4-FLUORO-1H-INDOLE-2-CARBOXYLATE AND ETHYL 5-CHLORO-6-FLUORO-1H-H-INDOLE-2-CARBOXYLATE

Romano Silvestri Dipartimento di Studi Farmaceutici, Università di Roma “La Sapienza”, Box 36-Roma 62, P.le Aldo Moro 5, I-00185, Roma, Italy
,
Gabriella De Martino Dipartimento di Studi Farmaceutici, Università di Roma “La Sapienza”, Box 36-Roma 62, P.le Aldo Moro 5, I-00185, Roma, Italy
&
Gianluca Sbardella Dipartimento di Scienze Farmaceutiche, Università di Salerno, Via Ponte Don Melillo, I-84084, Fisciano (Salerno), Italy Phone: +39 06 49913800 E-mail: [email protected]
Pages 517-520 | Received 03 Dec 2001, Published online: 11 Feb 2009

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Matiur Rahman, Monoranjan Ghosh, Alakananda Hajra & Adinath Majee. (2013) A simple and efficient approach for the sulfonylation of indoles catalyzed by CuI. Journal of Sulfur Chemistry 34:4, pages 342-346.
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Francesco Piscitelli, Giuseppe La Regina & Romano Silvestri. (2008) AN IMPROVED SYNTHESIS OF ETHYL 5-CHLORO-4-FLUORO-1H-INDOLE-2-CARBOXYLATE. Organic Preparations and Procedures International 40:2, pages 204-208.
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Articles from other publishers (6)

Valeria Famiglini & Romano Silvestri. (2018) Indolylarylsulfones, a fascinating story of highly potent human immunodeficiency virus type 1 non-nucleoside reverse transcriptase inhibitors. Antiviral Chemistry and Chemotherapy 26, pages 204020661775344.
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Benjamin A. MayesNarayan C. ChaudhuriChristopher P. HenckenFrederic JeannotG. Mark LathamSteven MathieuF. Patrick McGarryAlistair J. StewartJingyang WangAdel Moussa. (2010) Robust Synthesis of Methyl 5-Chloro-4-fluoro-1 H -indole-2-carboxylate: A Key Intermediate in the Preparation of an HIV NNRTI Candidate . Organic Process Research & Development 14:5, pages 1248-1253.
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Giuseppe La ReginaAntonio ColucciaFrancesco PiscitelliAlberto BergaminiAnna SinistroAntonella CavazzaGiovanni MagaAlberta SamueleSamantha ZanoliEttore NovellinoMarino ArticoRomano Silvestri. (2007) Indolyl Aryl Sulfones as HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors:  Role of Two Halogen Atoms at the Indole Ring in Developing New Analogues with Improved Antiviral Activity. Journal of Medicinal Chemistry 50:20, pages 5034-5038.
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Devendrapratap U. Singh, Pankajkumar R. Singh & Shriniwas D. Samant. (2004) Fe-pillared bentonite—an efficient catalyst for sulfonylation of arenes using aryl and alkyl sulfonyl chlorides. Tetrahedron Letters 45:49, pages 9079-9082.
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J.S. Yadav, B.V.S. Reddy, A.D. Krishna & T. Swamy. (2003) InBr3-catalyzed sulfonation of indoles: a facile synthesis of 3-sulfonyl indoles. Tetrahedron Letters 44:32, pages 6055-6058.
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Romano Silvestri, Gabriella De Martino & Gianluca Sbardella. (2010) A Simplified Synthesis of Ethyl 5‐Chloro‐4‐fluoro‐1H‐indole‐2‐carboxylate and Ethyl 5‐Chloro‐6‐fluoro‐1H‐indole‐2‐carboxylate.. ChemInform 33:52, pages 113-113.
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