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Xenobiotica
the fate of foreign compounds in biological systems
Volume 30, 2000 - Issue 10
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Research Article

Metabolism of 7-benzyloxy-4-trifluoromethylcoumarin by human hepatic cytochrome P450 isoforms

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Pages 955-969 | Published online: 22 Sep 2008

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Charles Awortwe, Vamshi K. Manda, Cristina Avonto, Shabana I. Khan, Ikhlas A. Khan, Larry A. Walker, Patrick J. Bouic & Bernd Rosenkranz. (2015) Echinacea purpurea up-regulates CYP1A2, CYP3A4 and MDR1 gene expression by activation of pregnane X receptor pathway. Xenobiotica 45:3, pages 218-229.
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Abidemi J. Akindele, Erika A. Eksioglu, Jason C. Kwan, Olufunmilayo O. Adeyemi, Chen Liu, Hendrik Luesch & Margaret O. James. (2011) Biological effects of Byrsocarpus coccineus in vitro. Pharmaceutical Biology 49:2, pages 152-160.
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Claudia Mariana Gómez-Gutiérrez & Graciela Guerra-Rivas. (2010) Uptake and biochemical response to B[a]P in the sea anemone Anthopleura elegantissima . Journal of Environmental Science and Health, Part A 45:1, pages 42-48.
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N. J. Proctor, G. T. Tucker & A. Rostami-Hodjegan. (2004) Predicting drug clearance from recombinantly expressed CYPs: intersystem extrapolation factors. Xenobiotica 34:2, pages 151-178.
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Slobodan Rendic. (2002) Summary of information on human CYP enzymes: human P450 metabolism data. Drug Metabolism Reviews 34:1-2, pages 83-448.
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A. B. Renwick, G. Lavignette, P. D. Worboys, B. Williams, D. Surry, D. F. V. Lewis, R. J. Price, B. G. Lake & D. C. Evans. (2001) Evaluation of 7-benzyloxy-4-trifluoromethylcoumarin, some other 7-hydroxy-4-trifluoromethylcoumarin derivatives and 7-benzyloxyquinoline as fluorescent substrates for rat hepatic cytochrome P450 enzymes. Xenobiotica 31:12, pages 861-878.
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A. B. Renwick, D. F. V. Lewis, S. Fulford, D. Surry, B. Williams, P. D. Worboys, X. Cai, R. W. Wang, R. J. Price, B. G. Lake & D. C. Evans. (2001) Metabolism of 2,5-bis(trifluoromethyl)-7-benzyloxy-4-trifluoromethylcoumarin by human hepatic CYP isoforms: evidence for selectivity towards CYP3A4. Xenobiotica 31:4, pages 187-204.
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