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Original Article

Radiosensitization Efficacy of KU-2285, RP-170 and Etanidazole at Low Radiation Doses: Assessment by in Vitro Cytokinesis-block Micronucleus Assay

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Pages 473-478 | Received 26 Jun 1991, Accepted 10 Oct 1991, Published online: 03 Jul 2009

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Yuta Shibamoto, Chikao Sugie, Hiroyuki Ogino & Natsuo Tomita. 2015. Intensity-Modulated Radiation Therapy. Intensity-Modulated Radiation Therapy 43 57 .
Yuta SHIBAMOTO, Shinya OTSUKA, Hiromitsu IWATA, Chikao SUGIE, Hiroyuki OGINO & Natsuo TOMITA. (2012) Radiobiological Evaluation of the Radiation Dose as Used in High-precision Radiotherapy: Effect of Prolonged Delivery Time and Applicability of the Linear-quadratic Model. Journal of Radiation Research 53:1, pages 1-9.
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Tomoaki YAHIRO, Shigeki MASUI, Nobuo KUBOTA, Koji YAMADA, Ataru KOBAYASHI & Kenichi KISHII. (2005) Effects of Hypoxic Cell Radiosensitizer Doranidazole (PR-350) on the Radioresponse of Murine and Human Tumor Cells in vitro and in vivo. Journal of Radiation Research 46:3, pages 363-372.
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Yuta Shibamoto, Masato Ito, Chikao Sugie, Hiroyuki Ogino & Masaki Hara. (2004) Recovery from sublethal damage during intermittent exposures in cultured tumor cells: implications for dose modification in radiosurgery and imrt. International Journal of Radiation Oncology*Biology*Physics 59:5, pages 1484-1490.
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J. M. Akudugu, J. P. Slabbert, A. Serafin & L. Bohm. (2000) Frequency of Radiation-Induced Micronuclei in Neuronal Cells Does Not Correlate with Clonogenic Survival. Radiation Research 153:1, pages 62-67.
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Yuta Shibamoto, Masaji Takahashi & Mitsuyuki Abe. (1996) A Phase I study of a hypoxic cell sensitizer KU-2285 in combination with conventional radiotherapy. Radiotherapy and Oncology 40:1, pages 55-58.
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Toru Shibata, Yuta Shibamoto, Keisuke Sasai, Natsuo Oya, Rumi Murata, Takehisa Takagi, Masahiro Hiraoka & Mitsuyuki Abe. (2005) Comparison of in vivo Efficacy of Hypoxic Cytotoxin Tirapazamine and Hypoxic Cell Radiosensitizer KU‐2285 in Combination with Single and Fractionated Irradiation . Japanese Journal of Cancer Research 87:1, pages 98-104.
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Natsuo Oya, Yuta Shibamoto, Keisuke Sasai, Toru Shibata, Rumi Murata, Takehisa Takagi, Hiroyuki Iwai, Toshimitsu Suzuki & Mitsuyuki Abe. (1995) Optical isomers of a new 2-nitroimidazole nucleoside analog (PR-350 series): Radiosensitization efficiency and toxicity. International Journal of Radiation Oncology*Biology*Physics 33:1, pages 119-127.
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Toru Shibata, Yuta Shibamoto, Keisuke Sasai, Natsuo Oya, Takehisa Takagi, Rumi Murata & Mitsuyuki Abe. (1995) Assessment of micronucleus induction in SCCVII cells treated with bioreductive agents, WIN 59075 (SR 4233) and mitomycin C, under aerobic and hypoxic conditions. Mutation Research/Genetic Toxicology 342:3-4, pages 171-177.
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Natsuo Oya, Yuta Shibamoto, Toru Shibata, Keisuke Sasai, Taketoshi Sugiyama & Mitsuyuki Abe. (1994) Combined cytokinesis-block micronucleus and chromosomal aberration assay for the evaluation of radiosensitizers at low radiation doses. International Journal of Radiation Oncology*Biology*Physics 30:5, pages 1153-1159.
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Natsuo Oya, Yuta Shibamoto, Toru Shibata, Rumi Murata, Hiroyuki Iwai, Taketoshi Sugiyama & Mitsuyuki Abe. (1994) KIN-804 vs. KU-2285 as a radiosensitizer for clinical use. International Journal of Radiation Oncology*Biology*Physics 29:3, pages 595-600.
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Hiroyuki Iwai, Etsuko Matsuno, Keisuke Sasai, Yuta Shibamoto & Mitsuyuki Abe. (1994) Radiosensitizing activity and pharmacokinetics of multiple dose administered KU-2285 in peripheral nerve tissue in mice. International Journal of Radiation Oncology*Biology*Physics 29:3, pages 591-594.
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Toru Shibata, Yuta Shibamoto, Natsuo Oya, Keisuke Sasai, Rumi Murata, Takashi Ishigaki & Mitsuyuki Abe. (1994) Comparison of radiosensitizing effect of KU-2285 and SR-2508 at low drug concentrations and doses. International Journal of Radiation Oncology*Biology*Physics 29:3, pages 587-590.
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Keisuke Sasai, Hiroyuki Iwai, Toru Yoshizawa, Sei-Ichi Nishimoto, Yuta Shibamoto, Natsuo Oya, Toru Shibata & Mitsuyuki Abe. (1994) Fluorinated 2-nitroimidazole derivative hypoxic cell radiosensitizers: Radiosensitizing activities and pharmacokinetics. International Journal of Radiation Oncology*Biology*Physics 29:3, pages 579-582.
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Kirsten A. Skov & Susan Macphail. (1994) Low concentrations of nitroimidazoles: Effective radiosensitizers at low doses. International Journal of Radiation Oncology*Biology*Physics 29:1, pages 87-93.
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Natsuo Oya, Yuta Shibamoto, Keisuke Sasai, Taketoshi Sugiyama & Mitsuyuki Abe. (1993) In vivo radiosensitization efficacy of KU-2285 and etanidazole at clinically relevant low radiation doses. International Journal of Radiation Oncology*Biology*Physics 27:5, pages 1113-1119.
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