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Research Article

The molecular basis of the structure and function of the 5-HT 3 receptor: a model ligand-gated ion channel (Review)

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Pages 11-26 | Published online: 09 Jul 2009

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Francesca De Rienzo, Arménio J. Moura Barbosa, Marta A.S. Perez, Pedro A. Fernandes, Maria J. Ramos & Maria Cristina Menziani. (2012) The extracellular subunit interface of the 5-HT3 receptors: a computational alanine scanning mutagenesis study. Journal of Biomolecular Structure and Dynamics 30:3, pages 280-298.
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Tamme W. Goecke, Arif B. Ekici, Beate Niesler, Christian R. Loehberg, Christian Hammer, Gudrun Rappold, Denny Schanze, Verica Straub, Hans-Harald Altmann, Pamela Strissel, Reiner Strick, Matthias W. Beckmann & Peter A. Fasching. (2010) Two naturally occurring variants of the serotonin receptor gene HTR3C are associated with nausea in pregnancy. Acta Obstetricia et Gynecologica Scandinavica 89:1, pages 7-14.
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E Anthony Jones. (2008) Pruritus and fatigue associated with liver disease: is there a role for ondansetron?. Expert Opinion on Pharmacotherapy 9:4, pages 645-651.
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Andrew J Thompson & Sarah CR Lummis. (2007) The 5-HT3 receptor as a therapeutic target. Expert Opinion on Therapeutic Targets 11:4, pages 527-540.
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Nora L. Sullivan, Nora L. Sullivan, Andrew J. Thompson, Kerry L. Price & Sarah C. R. Lummis. (2006) Defining the roles of Asn-128, Glu-129 and Phe-130 in loop A of the 5-HT3 receptor. Molecular Membrane Biology 23:5, pages 442-451.
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Shiva Amiri, Kaihsu Tai, Oliver Beckstein, Philip C. Biggin & Mark S. P. Sansom. (2005) The α7 nicotinic acetylcholine receptor: Molecular modelling, electrostatics, and energetics. Molecular Membrane Biology 22:3, pages 151-162.
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BL Fiebich, RS Akundi, M Seidel, V Geyer, U Haus, W Müller, T Stratz & E Candelario‐Jalil. (2004) Expression of 5‐HT3A receptors in cells of the immune system. Scandinavian Journal of Rheumatology 33:sup119, pages 9-11.
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Robert Luedtke, Cathy Bell-Horner, Michael Volk, Manfred Reinecke & Glenn Dillon. (2004) Pharmacological Survey of Medicinal Plants for Activity at Ligand-Gated Ion Channels: Selective Interaction with 5-HT3 Receptors. Pharmaceutical Biology 42:1, pages 73-82.
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