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Original Articles: Clinical

A phase 1 trial of the HDAC inhibitor AR-42 in patients with multiple myeloma and T- and B-cell lymphomas

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Pages 2310-2318 | Received 13 Sep 2016, Accepted 16 Feb 2017, Published online: 07 Mar 2017

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R. Kundu, S. Banerjee, S.K. Baidya, N. Adhikari & T. Jha. (2022) A quantitative structural analysis of AR-42 derivatives as HDAC1 inhibitors for the identification of promising structural contributors. SAR and QSAR in Environmental Research 33:11, pages 861-883.
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Nour Ghazzaui, Mélissa Ferrad, Hussein Issaoui, Sandrine Lecardeur, Jeanne Cook-Moreau, Justine Pollet, Sandrine Le Noir & Yves Denizot. (2021) HDAC recruitment in the IgH locus 3’ regulatory region is different between mature B-cells and mature B-cell lymphomas. Leukemia & Lymphoma 62:14, pages 3511-3515.
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Sophia G. Liva, Christopher C. Coss, Jiang Wang, William Blum, Rebecca Klisovic, Bhavana Bhatnagar, Katherine Walsh, Susan Geyer, Qiuhong Zhao, Ramiro Garzon, Guido Marcucci, Mitch A. Phelps & Alison R. Walker. (2020) Phase I study of AR-42 and decitabine in acute myeloid leukemia. Leukemia & Lymphoma 61:6, pages 1484-1492.
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