4,906
Views
91
CrossRef citations to date
0
Altmetric
Research Article

Preparation of curcumin self-micelle solid dispersion with enhanced bioavailability and cytotoxic activity by mechanochemistry

, , , , , , & show all
Pages 198-209 | Received 03 Nov 2017, Accepted 25 Dec 2017, Published online: 05 Jan 2018

Keep up to date with the latest research on this topic with citation updates for this article.

Read on this site (9)

Junying Zhang, Yiwen Zhang, Hufang Wang, Wenlin Chen, Aiyu Lu, Hailiang Li, Lifeng Kang & Chunyong Wu. (2023) Solubilisation and Enhanced Oral Absorption of Curcumin Using a Natural Non-Nutritive Sweetener Mogroside V. International Journal of Nanomedicine 18, pages 1031-1045.
Read now
Dabu Zhu, Qiuqin Zhang, Yifang Chen, Minghua Xie, Jianbo Li, Shen Yao, Ming Li, Zhao Lou, Yue Cai & Xuanrong Sun. (2022) Mechanochemical preparation of triptolide-loaded self-micelle solid dispersion with enhanced oral bioavailability and improved anti-tumor activity. Drug Delivery 29:1, pages 1398-1408.
Read now
Shiqi Liu, Han Liu, Lulu Zhang, Chao Ma & A. M. Abd El-Aty. (2022) Edible pentacyclic triterpenes: A review of their sources, bioactivities, bioavailability, self-assembly behavior, and emerging applications as functional delivery vehicles. Critical Reviews in Food Science and Nutrition 0:0, pages 1-17.
Read now
Yelda Komesli & Ercument Karasulu. (2022) Permeability of olmesartan medoxomil from lipid based and suspension formulations using an optimized HDM-PAMPA model. Pharmaceutical Development and Technology 27:6, pages 749-757.
Read now
Bing Chen, Xuewen Wang, Yanyan Zhang, Kangping Huang, Hao Liu, Dafen Xu, Shaoguang Li, Qicai Liu, Jianyong Huang, Hong Yao & Xinhua Lin. (2020) Improved solubility, dissolution rate, and oral bioavailability of main biflavonoids from Selaginella doederleinii extract by amorphous solid dispersion. Drug Delivery 27:1, pages 309-322.
Read now
Yuzhen Hou, Hui Wang, Fan Zhang, Fengyuan Sun, Meng Xin, Mengshuang Li, Jun Li & Xianggen Wu. (2019) Novel self-nanomicellizing solid dispersion based on rebaudioside A: a potential nanoplatform for oral delivery of curcumin. International Journal of Nanomedicine 14, pages 557-571.
Read now
Fengyuan Sun, Zhou Zheng, Jie Lan, Xuefei Li, Mengshuang Li, Kaichao Song & Xianggen Wu. (2019) New micelle myricetin formulation for ocular delivery: improved stability, solubility, and ocular anti-inflammatory treatment. Drug Delivery 26:1, pages 575-585.
Read now
Pinggang Ding, Hongxue Shen, Jianan Wang & Jianming Ju. (2018) Improved oral bioavailability of magnolol by using a binary mixed micelle system. Artificial Cells, Nanomedicine, and Biotechnology 46:sup2, pages 668-674.
Read now

Articles from other publishers (82)

Debadatta Mohapatra, Dulla Naveen Kumar, Singh Shreya, Vivek Pandey, Pawan K. Dubey, Ashish Kumar Agrawal & Alakh N Sahu. (2023) Quality by design–based development and optimization of fourth-generation ternary solid dispersion of standardized Piper longum extract for melanoma therapy. Drug Delivery and Translational Research 13:12, pages 3094-3131.
Crossref
Mohammad Banazadeh, Behzad Behnam, Narges Ashraf Ganjooei, B.H. Jaswanth Gowda, Prashant Kesharwani & Amirhossein Sahebkar. (2023) Curcumin-based nanomedicines: A promising avenue for brain neoplasm therapy. Journal of Drug Delivery Science and Technology 89, pages 105040.
Crossref
RENI AGUSTINA & DEWI SETYANINGSIH. (2023) SOLID DISPERSION AS A POTENTIAL APPROACH TO IMPROVE DISSOLUTION AND BIOAVAILABILITY OF CURCUMIN FROM TURMERIC (CURCUMA LONGA L.). International Journal of Applied Pharmaceutics, pages 37-47.
Crossref
Jai Bharti Sharma, Shailendra Bhatt, Abhishek Tiwari, Varsha Tiwari, Manish Kumar, Ravinder Verma, Deepak Kaushik, Tarun Virmani, Girish Kumar, Omkulthom Al kamaly, Asmaa Saleh, Mohammed Khalid Parvez & Abdulsalam Alhalmi. (2023) Statistical optimization of tetrahydrocurcumin loaded solid lipid nanoparticles using Box Behnken design in the management of streptozotocin-induced diabetes mellitus. Saudi Pharmaceutical Journal 31:9, pages 101727.
Crossref
Dan Shen, Tingyu Jin, Yin Xiao, Xingyi Zhu & Yunfen Hua. (2023) Preparation of pazopanib-fumarate disodium glycyrrhizinate nanocrystalline micelles by liquid-assisted ball milling. European Journal of Pharmaceutical Sciences 188, pages 106530.
Crossref
Esha S. Attar, Vanashree H. Chaudhari, Chaitanya G. Deokar, Sathish Dyawanapelly & Padma V. Devarajan. (2023) Nano Drug Delivery Strategies for an Oral Bioenhanced Quercetin Formulation. European Journal of Drug Metabolism and Pharmacokinetics 48:5, pages 495-514.
Crossref
Jian-Hong Qi, Dong-Chuan Xu, Xiao-Long Wang, Ding-Yuan Cai, Yi Wang & Wei Zhou. (2023) Micro-simulation insights into the functional and mechanistic understanding of glycyrrhizin against asthma. Frontiers in Pharmacology 14.
Crossref
Nasim Shadmani, Sepehr Gohari, Azin Kadkhodamanesh, Parivash Ghaderinia, Maryam Hassani & Motahare Sharifyrad. (2023) The synthesis and development of poly(ε-caprolactone) conjugated polyoxyethylene sorbitan oleate-based micelles for curcumin drug release: an in vitro study on breast cancer cells . RSC Advances 13:34, pages 23449-23460.
Crossref
Maria N. Lvova, Denis V. Ponomarev, Alena A. Tarasenko, Anna V. Kovner, Galina A. Minkova, Michail A. Tsyganov, Meijun Li, Yan Lou, Veronica I. Evseenko, Alexander V. Dushkin, Irina V. Sorokina, Tatiana G. Tolstikova, Viatcheslav A. Mordvinov & Damira F. Avgustinovich. (2023) Curcumin and Its Supramolecular Complex with Disodium Glycyrrhizinate as Potential Drugs for the Liver Fluke Infection Caused by Opisthorchis felineus. Pathogens 12:6, pages 819.
Crossref
Xiaoshun Jia, Jinfeng Chen, Hongqing Cheng, Xinxin Pan, Yixin Ke, Tingming Fu, Hongzhi Qiao, Xiaobing Cui, Wen Li, Lisi Zou, Jianming Cheng & Junsong Li. (2023) Use of surfactant-based amorphous solid dispersions for BDDCS class II drugs to enhance oral bioavailability: A case report of resveratrol. International Journal of Pharmaceutics 641, pages 123059.
Crossref
Tahir Mahmood, Rai M. SarfrazAsmara IsmailMuhammad AliAbdur Rauf Khan. (2023) Pharmaceutical Methods for Enhancing the Dissolution of Poorly Water-Soluble Drugs. ASSAY and Drug Development Technologies 21:2, pages 65-79.
Crossref
Enas Elmowafy, Marwa O. El-Derany, Luca Casettari, Mahmoud E. Soliman & Riham I. El-Gogary. (2023) Gamma oryzanol loaded into micelle-core/chitosan-shell: from translational nephroprotective potential to emphasis on sirtuin-1 associated machineries. International Journal of Pharmaceutics 631, pages 122482.
Crossref
Xingxing Dai, Yuyao Liao, Cuiting Yang, Yingying Zhang, Minfang Feng, Yuting Tian, Qingsong Qu, Mengke Sheng, Zhixun Li, Xinhui Peng, Shuai Cen & Xinyuan Shi. (2022) Diammonium Glycyrrhizinate-Based Micelles for Improving the Hepatoprotective Effect of Baicalin: Characterization and Biopharmaceutical Study. Pharmaceutics 15:1, pages 125.
Crossref
Olga Yu. Selyutina, Simon V. Babenko, Alexander I. Kruppa, Tatyana V. Leshina & Nikolay E. Polyakov. (2022) Photostabilization of ketoprofen by inclusion in glycyrrhizin micelles and gel nanoparticles. New Journal of Chemistry 46:37, pages 17865-17873.
Crossref
Yin Xiao, Tingyu Jin, Xuerong Geng & Xingyi Zhu. (2022) Azilsartan-nicotinamide cocrystal: Preparation, characterization and in vitro / vivo evaluation. European Journal of Pharmaceutical Sciences 176, pages 106241.
Crossref
Suchiwa Pan-On, Piyameth Dilokthornsakul & Waree Tiyaboonchai. (2022) Trends in advanced oral drug delivery system for curcumin: A systematic review. Journal of Controlled Release 348, pages 335-345.
Crossref
Shichang Zhang, Yiwei Zhao, Liangjun Tan, Sheng Wu, Qing Zhang, Boxin Zhao & Guofeng Li. (2022) A Novel Berberine–Glycyrrhizic Acid Complex Formulation Enhanced the Prevention Effect to Doxorubicin-Induced Cardiotoxicity by Pharmacokinetic Modulation of Berberine in Rats. Frontiers in Pharmacology 13.
Crossref
Shasha Yang, Zhihuan Zhao, Yiliang Xie, Jianying Lin, Bing Zhang & Jimin Fan. (2022) Engineering Bio-MOF/polydopamine as a biocompatible targeted theranostic system for synergistic multi-drug chemo-photothermal therapy. International Journal of Pharmaceutics 623, pages 121912.
Crossref
Min Lu, Wei Wei, Wenhao Xu, Nikolay E. Polyakov, Alexandr V. Dushkin & Weike Su. (2022) Preparation of DNC Solid Dispersion by a Mechanochemical Method with Glycyrrhizic Acid and Polyvinylpyrrolidone to Enhance Bioavailability and Activity. Polymers 14:10, pages 2037.
Crossref
Alaa F. Bakr, Ping Shao & Mohamed A. Farag. (2022) Recent advances in glycyrrhizin metabolism, health benefits, clinical effects and drug delivery systems for efficacy improvement; a comprehensive review. Phytomedicine 99, pages 153999.
Crossref
Zh. F. Ziyavitdinov, U. Zh. Ishimov, N. Sh. Berdiev, I. Z. Zhumaev, Yu. I. Oshchepkova, P. B. Usmanov & Sh. I. Salikhov. (2022) Supramolecular Complex of Lappaconitine Hydrobromide and the Monoammonium Salt of Glycyrrhizic Acid: Synthesis, Physicochemical Characteristics, and Antiarrhythmic Activity. Pharmaceutical Chemistry Journal 56:2, pages 167-173.
Crossref
Qihong Zhang, Chen Su, Zhaohui Lu, Hui Wang, Zongmiao Feng, Alexandr V. Dushkin & Weike Su. (2022) Preparation, physicochemical and pharmacological study of 10-hydroxycamptothecin solid dispersion with complexation agent – xylan-nonanoic acid amphiphilic conjugates. International Journal of Biological Macromolecules 204, pages 224-233.
Crossref
Jiwei Cui, Yuanxin Xu, Haiyan Tu, Huacong Zhao, Honglan Wang, Liuqing Di & Ruoning Wang. (2022) Gather wisdom to overcome barriers: Well-designed nano-drug delivery systems for treating gliomas. Acta Pharmaceutica Sinica B 12:3, pages 1100-1125.
Crossref
Qihong Zhang, Zongmiao Feng, Wei Ren, Yunchun Zhao, Alexandr V. Dushkin & Weike Su. (2021) Preparation of olmesartan medoxomil solid dispersion with sustained release performance by mechanochemical technology. Drug Delivery and Translational Research 12:3, pages 589-602.
Crossref
Zhuomin Xu, Shanshan Zheng, Xin Gao, Yulu Hong, Yue Cai, Qiuqin Zhang, Jiani Xiang, Dehui Xie, Fuxing Song, Huawei Zhang, Hong Wang & Xuanrong Sun. (2021) Mechanochemical preparation of chrysomycin A self-micelle solid dispersion with improved solubility and enhanced oral bioavailability. Journal of Nanobiotechnology 19:1.
Crossref
A.V. Kim, E.A. Shelepova, V.I. Evseenko, A.V. Dushkin, N.N. Medvedev & N.E. Polyakov. (2021) Mechanism of the enhancing effect of glycyrrhizin on nifedipine penetration through a lipid membrane. Journal of Molecular Liquids 344, pages 117759.
Crossref
Qin Shen, Yongjie Jiang, Jing Chen, Xueling Wang & Jiao Zheng. (2021) A Novel Curcumin-Based Drug Powder Inhalation Medicine for Chronic Obstructive Pulmonary Disease. Bioinorganic Chemistry and Applications 2021, pages 1-9.
Crossref
Hui Yang, Qilong Cao, Zhixin Yuan, Xianggen Wu & Mengshuang Li. (2021) Enhanced therapeutic efficacy of a novel self-micellizing nanoformulation-loading fisetin against acetaminophen-induced liver injury. Nanomedicine 16:27, pages 2431-2448.
Crossref
Shuang Li, Jueshuo Guo, Zonghua Tian, Jing Chen, Guojing Gou, Yang Niu, Li Li & Jianhong Yang. (2021) Piperine-Loaded Glycyrrhizic Acid- and PLGA-Based Nanoparticles Modified with Transferrin for Antitumor. AAPS PharmSciTech 22:7.
Crossref
Qihong Zhang, Hui Wang, Zongmiao Feng, Zhaohui Lu, Chen Su, Yunchun Zhao, Jingbo Yu, Alexandr V. Dushkin & Weike Su. (2021) Preparation of pectin-tannic acid coated core-shell nanoparticle for enhanced bioavailability and antihyperlipidemic activity of curcumin. Food Hydrocolloids 119, pages 106858.
Crossref
Mohamed Elbadawy, Kimika Hayashi, Hiromi Ayame, Yusuke Ishihara, Amira Abugomaa, Makoto Shibutani, Shim-Mo Hayashi, Shoichi Hazama, Hiroko Takenouchi, Masao Nakajima, Ryouichi Tsunedomi, Nobuaki Suzuki, Hiroaki Nagano, Yuta Shinohara, Masahiro Kaneda, Hideyuki Yamawaki, Tatsuya Usui & Kazuaki Sasaki. (2021) Anti-cancer activity of amorphous curcumin preparation in patient-derived colorectal cancer organoids. Biomedicine & Pharmacotherapy 142, pages 112043.
Crossref
Gamze Ergin Kızılçay & Sıdıka Ertürk Toker. (2021) Effect of glycyrrhizic acid on the bioavailability of resveratrol after oral administration in rabbit plasma using HPLC with fluorescence detection. Microchemical Journal 168, pages 106360.
Crossref
Hasriadi, Peththa Wadu Dasuni Wasana, Opa Vajragupta, Pornchai Rojsitthisak & Pasarapa Towiwat. (2021) Mechanistic Insight into the Effects of Curcumin on Neuroinflammation-Driven Chronic Pain. Pharmaceuticals 14:8, pages 777.
Crossref
Keyvan Khazei, Nasrin Mohajeri, Esat Bonabi, Zeynep Turk & Nosratollah Zarghami. (2021) New Insights Toward Nanostructured Drug Delivery of Plant-Derived Polyphenol Compounds: Cancer Treatment and Gene Expression Profiles. Current Cancer Drug Targets 21:8, pages 689-701.
Crossref
Aibibai Amuti, Xue Wang, Mingyang Zan, Shaojun Lv & Zhanzhong Wang. (2021) Formulation and characterization of curcumin-loaded microemulsions: Evaluation of antioxidant stability and in vitro release. Journal of Molecular Liquids 336, pages 116881.
Crossref
Wenjing Su, Nikolay E. Polyakov, Wenhao Xu & Weike Su. (2021) Preparation of astaxanthin micelles self-assembled by a mechanochemical method from hydroxypropyl β-cyclodextrin and glyceryl monostearate with enhanced antioxidant activity. International Journal of Pharmaceutics 605, pages 120799.
Crossref
Qihong Zhang, Zongmiao Feng, Hui Wang, Chen Su, Zhaohui Lu, Jingbo Yu, Alexandr V. Dushkin & Weike Su. (2021) Preparation of camptothecin micelles self-assembled from disodium glycyrrhizin and tannic acid with enhanced antitumor activity. European Journal of Pharmaceutics and Biopharmaceutics 164, pages 75-85.
Crossref
Helmy Yusuf, Nina Wijiani, Rizka Arifa Rahmawati, Riesta Primaharinastiti, M. Agus Syamsur Rijal & Dewi Isadiartuti. (2021) Analytical method for the determination of curcumin entrapped in polymeric micellar powder using HPLC. Journal of Basic and Clinical Physiology and Pharmacology 32:4, pages 867-873.
Crossref
Yuyao Liao, Zhixun Li, Qing Zhou, Mengke Sheng, Qingsong Qu, Yanshuang Shi, Jiaqi Yang, Lijing Lv, Xingxing Dai & Xinyuan Shi. (2021) Saponin surfactants used in drug delivery systems: A new application for natural medicine components. International Journal of Pharmaceutics 603, pages 120709.
Crossref
Sana Rubab, Komal Naeem, Isra Rana, Namrah Khan, Maryam Afridi, Izhar Ullah, Fawad Ali Shah, Sadia Sarwar, Fakhar ud Din, Ho-Ik Choi, Cheol-Ho Lee, Chang-Wan Lim, Abir Abdullah Alamro, Jin-Ki Kim & Alam Zeb. (2021) Enhanced neuroprotective and antidepressant activity of curcumin-loaded nanostructured lipid carriers in lipopolysaccharide-induced depression and anxiety rat model. International Journal of Pharmaceutics 603, pages 120670.
Crossref
Lei Zheng, Chen Sun, Xingyi Zhu, Wenhao Xu, Jingbo Yu, Qihong Zhang, Alexandr V. Dushkin & Weike Su. (2021) Inositol hexanicotinate self-micelle solid dispersion is an efficient drug delivery system in the mouse model of non-alcoholic fatty liver disease. International Journal of Pharmaceutics 602, pages 120576.
Crossref
Blake C. Walker, Srijan Adhikari & Sandeep Mittal. 2021. Gliomas. Gliomas 139 150 .
Jai Bharti SharmaShailendra Bhatt, Vipin SainiManish Kumar. (2021) Pharmacokinetics and Pharmacodynamics of Curcumin-Loaded Solid Lipid Nanoparticles in the Management of Streptozotocin-Induced Diabetes Mellitus: Application of Central Composite Design. ASSAY and Drug Development Technologies 19:4, pages 262-279.
Crossref
Wenhao Xu, Wenjing Su, Zhencheng Xue, Faxiang Pu, Zhangfu Xie, Kongliang Jin, Nikolay E. Polyakov, Alexander V. Dushkin & Weike Su. (2021) Research on Preparation of 5-ASA Colon-Specific Hydrogel Delivery System without Crosslinking Agent by Mechanochemical Method. Pharmaceutical Research 38:4, pages 693-706.
Crossref
Wei Wei, Veronica I. Evseenko, Mikhail V. Khvostov, Sergey A. Borisov, Tatyana G. Tolstikova, Nikolay E. Polyakov, Aleksandr V. Dushkin, Wenhao Xu, Lu Min & Weike Su. (2021) Solubility, Permeability, Anti-Inflammatory Action and In Vivo Pharmacokinetic Properties of Several Mechanochemically Obtained Pharmaceutical Solid Dispersions of Nimesulide. Molecules 26:6, pages 1513.
Crossref
Ping Ying, Jingbo Yu & Weike Su. (2021) Liquid‐Assisted Grinding Mechanochemistry in the Synthesis of Pharmaceuticals. Advanced Synthesis & Catalysis 363:5, pages 1246-1271.
Crossref
Dong-Wei Wang, Shu-Juan Li, Xue-Ying Tan, Jin-Hui Wang, Ying Hu, Zeng Tan, Jing Liang, Jing-Bo Hu, Yan-Guo Li & Yu-Fen Zhao. (2021) Engineering of stepwise-targeting chitosan oligosaccharide conjugate for the treatment of acute kidney injury. Carbohydrate Polymers 256, pages 117556.
Crossref
Olga Yu. Selyutina, Anna V. Mastova, Ekaterina A. Shelepova & Nikolay E. Polyakov. (2021) pH-Sensitive Glycyrrhizin Based Vesicles for Nifedipine Delivery. Molecules 26:5, pages 1270.
Crossref
Fan Zhang, Huabo Chen, Jie Lan, Kaichao Song & Xianggen Wu. (2021) Preparation and in vitro/in vivo evaluations of novel ocular micelle formulations of hesperetin with glycyrrhizin as a nanocarrier. Experimental Eye Research 202, pages 108313.
Crossref
Jie Gao, Kenza Mamouni, Lei Zhang & Bal L. Lokeshwar. 2021. Evolutionary Diversity as a Source for Anticancer Molecules. Evolutionary Diversity as a Source for Anticancer Molecules 275 308 .
A. I. Varlamova, I. A. Arkhipov, S. S. Khalikov, K. M. Sadov & T. Yu. Degtyarevskaya. (2021) Praziquantel Efficacy Increased Using Mechanical Technology and Supramolecular Targeted Delivery System for Treatment of Cestodiasis. Pharmaceutical Chemistry Journal 54:10, pages 1075-1078.
Crossref
Huanhuan Luo, Tianyang Jie, Li Zheng, Chenglong Huang, Gang Chen & Wenguo Cui. 2021. Bio-Nanomedicine for Cancer Therapy. Bio-Nanomedicine for Cancer Therapy 163 190 .
Elisa Panzarini, Stefania Mariano, Stefano Tacconi, Elisabetta Carata, Ada Maria Tata & Luciana Dini. (2020) Novel Therapeutic Delivery of Nanocurcumin in Central Nervous System Related Disorders. Nanomaterials 11:1, pages 2.
Crossref
Blake C. Walker & Sandeep Mittal. (2020) Antitumor Activity of Curcumin in Glioblastoma. International Journal of Molecular Sciences 21:24, pages 9435.
Crossref
Zhenqi Liu, John D. Smart & Ananth S. Pannala. (2020) Recent developments in formulation design for improving oral bioavailability of curcumin: A review. Journal of Drug Delivery Science and Technology 60, pages 102082.
Crossref
Igor Lomovskiy, Aleksey Bychkov, Oleg Lomovsky & Tatiana Skripkina. (2020) Mechanochemical and Size Reduction Machines for Biorefining. Molecules 25:22, pages 5345.
Crossref
Phuong H.L. Tran & Thao T.D. Tran. (2020) Developmental Strategies of Curcumin Solid Dispersions for Enhancing Bioavailability. Anti-Cancer Agents in Medicinal Chemistry 20:16, pages 1874-1882.
Crossref
Kaichao Song, Meixing Yan, Mengshuang Li, Yiwan Geng & Xianggen Wu. (2020) Preparation and in vitro–in vivo evaluation of novel ocular nanomicelle formulation of thymol based on glycyrrhizin. Colloids and Surfaces B: Biointerfaces 194, pages 111157.
Crossref
Jun Young Park, Ga Eul Chu, Sanghyo Park, Chaewon Park, Susmita Aryal, Won Jun Kang, Won Gil Cho & Jaehong Key. (2020) Therapeutic Efficacy of Curcumin Enhanced by Microscale Discoidal Polymeric Particles in a Murine Asthma Model. Pharmaceutics 12:8, pages 739.
Crossref
Yuri I. Glazachev, Anna A. Schlotgauer, Viktor A. Timoshnikov, Polina A. Kononova, Olga Yu. Selyutina, Ekaterina A. Shelepova, Maxim V. Zelikman, Mikhail V. Khvostov & Nikolay E. Polyakov. (2020) Effect of Glycyrrhizic Acid and Arabinogalactan on the Membrane Potential of Rat Thymocytes Studied by Potential-Sensitive Fluorescent Probe. The Journal of Membrane Biology 253:4, pages 343-356.
Crossref
Hui Wang, Yuanlong He, Yuzhen Hou, Yiwan Geng & Xianggen Wu. (2020) Novel self-nanomicellizing formulation based on Rebaudioside A: A potential nanoplatform for oral delivery of naringenin. Materials Science and Engineering: C 112, pages 110926.
Crossref
Yoon Tae Goo, Sun Young Park, Bo Ram Chae, Ho Yub Yoon, Chang Hyun Kim, Ji Yeh Choi, Seh Hyon Song & Young Wook Choi. (2020) Optimization of solid self-dispersing micelle for enhancing dissolution and oral bioavailability of valsartan using Box-Behnken design. International Journal of Pharmaceutics 585, pages 119483.
Crossref
Yiyan Song, Ling Cai, Zhongcheng Tian, Yuan Wu & Jin Chen. (2020) Phytochemical Curcumin-Coformulated, Silver-Decorated Melanin-like Polydopamine/Mesoporous Silica Composites with Improved Antibacterial and Chemotherapeutic Effects against Drug-Resistant Cancer Cells. ACS Omega 5:25, pages 15083-15094.
Crossref
O.Yu Selyutina, E.A. Shelepova, E.D. Paramonova, L.A. Kichigina, S.S. Khalikov & N.E. Polyakov. (2020) Glycyrrhizin-induced changes in phospholipid dynamics studied by 1H NMR and MD simulation. Archives of Biochemistry and Biophysics 686, pages 108368.
Crossref
Loanda Aparecida Cabral Rudnik, Paulo Vitor Farago, Jane Manfron Budel, Amanda Lyra, Fernanda Malaquias Barboza, Traudi Klein, Carla Cristine Kanunfre, Jessica Mendes Nadal, Matheus Coelho Bandéca, Vijayasankar Raman, Andressa Novatski, Alessandro Dourado Loguércio & Sandra Maria Warumby Zanin. (2020) Co-Loaded Curcumin and Methotrexate Nanocapsules Enhance Cytotoxicity against Non-Small-Cell Lung Cancer Cells. Molecules 25:8, pages 1913.
Crossref
Qihong Zhang, Wei Ren, Alexandr V. Dushkin & Weike Su. (2020) Preparation, characterization, in vitro and in vivo studies of olmesartan medoxomil in a ternary solid dispersion with N-methyl-D-glucamine and hydroxypropyl-β-cyclodextrin. Journal of Drug Delivery Science and Technology 56, pages 101546.
Crossref
Wen-hao Xu, Han-tao Wang, Ying Sun, Zhen-cheng Xue, Ming-li Liang & Wei-ke Su. (2020) Antihyperuricemic and nephroprotective effects of extracts from Orthosiphon stamineus in hyperuricemic mice . Journal of Pharmacy and Pharmacology 72:4, pages 551-560.
Crossref
Jingbo Yu, Ping Ying, Hao Wang, Keyu Xiang & Weike Su. (2020) Mechanochemical Asymmetric Cross‐Dehydrogenative Coupling Reaction: Liquid‐Assisted Grinding Enables Reaction Acceleration and Enantioselectivity Control. Advanced Synthesis & Catalysis 362:4, pages 893-902.
Crossref
Ziyue Xi, Wei Zhang, Yali Fei, Mingshu Cui, Luyao Xie, Lu Chen & Lu Xu. (2020) Evaluation of the Solid Dispersion System Engineered from Mesoporous Silica and Polymers for the Poorly Water Soluble Drug Indomethacin: In Vitro and In Vivo. Pharmaceutics 12:2, pages 144.
Crossref
Olga Yu. Selyutina, Salavat S. Khalikov & Nikolay E. Polyakov. (2019) Arabinogalactan and glycyrrhizin based nanopesticides as novel delivery systems for plant protection. Environmental Science and Pollution Research 27:6, pages 5864-5872.
Crossref
Vincenzo De Leo, Sante Di Gioia, Francesco Milano, Paola Fini, Roberto Comparelli, Erminia Mancini, Angela Agostiano, Massimo Conese & Lucia Catucci. (2020) Eudragit S100 Entrapped Liposome for Curcumin Delivery: Anti-Oxidative Effect in Caco-2 Cells. Coatings 10:2, pages 114.
Crossref
Daniel Hernandez-Patlan, Bruno Solis-Cruz, Karine P. Pontin, Juan D. Latorre, Xochitl Hernandez-Velasco, Ruben Merino-Guzman, Abraham Mendez-Albores, Billy M. Hargis, Raquel Lopez-Arellano & Guillermo Tellez-Isaias. (2019) Evaluation of Ascorbic Acid or Curcumin Formulated in a Solid Dispersion on Salmonella Enteritidis Infection and Intestinal Integrity in Broiler Chickens. Pathogens 8:4, pages 229.
Crossref
Jieying Cai, Shiwen Luo, Xueli Lv, Yingguang Deng, Hongyuan Huang, Boxin Zhao, Qing Zhang & Guofeng Li. (2019) Formulation of injectable glycyrrhizic acid-hydroxycamptothecin micelles as new generation of DNA topoisomerase I inhibitor for enhanced antitumor activity. International Journal of Pharmaceutics 571, pages 118693.
Crossref
Focsan, Polyakov & Kispert. (2019) Supramolecular Carotenoid Complexes of Enhanced Solubility and Stability—The Way of Bioavailability Improvement. Molecules 24:21, pages 3947.
Crossref
Vinod S. Ipar, Anisha Dsouza & Padma V. Devarajan. (2019) Enhancing Curcumin Oral Bioavailability Through Nanoformulations. European Journal of Drug Metabolism and Pharmacokinetics 44:4, pages 459-480.
Crossref
Alexandra V. Kim, Ekaterina A. Shelepova, Olga Yu Selyutina, Elizaveta S. Meteleva, Alexander V. Dushkin, Nikolai N. Medvedev, Nikolay E. Polyakov & Nikolay Z. Lyakhov. (2019) Glycyrrhizin-Assisted Transport of Praziquantel Anthelmintic Drug through the Lipid Membrane: An Experiment and MD Simulation. Molecular Pharmaceutics 16:7, pages 3188-3198.
Crossref
Huan Zhou, Wenjie Wang, Hang Hu, Xinye Ni, Su Ni, Ying Xu, Lei Yang & Defeng Xu. (2019) Co-precipitation of calcium carbonate and curcumin in an ethanol medium as a novel approach for curcumin dissolution enhancement. Journal of Drug Delivery Science and Technology 51, pages 397-402.
Crossref
Ying Gao, Guo Chen, Xiaojiao Luan, Meijuan Zou, Hongyu Piao & Gang Cheng. (2019) Improved Oral Absorption of Poorly Soluble Curcumin via the Concomitant Use of Borneol. AAPS PharmSciTech 20:4.
Crossref
Qihong Zhang, Lubov Suntsova, Yulia S. Chistyachenko, Veronika Evseenko, Mikhail V. Khvostov, Nikolay E. Polyakov, Alexandr V. Dushkin & Weike Su. (2019) Preparation, physicochemical and pharmacological study of curcumin solid dispersion with an arabinogalactan complexation agent. International Journal of Biological Macromolecules 128, pages 158-166.
Crossref
Elizaveta S. Meteleva, Yulia S. Chistyachenko, Lyubov P. Suntsova, Mikhail V. Khvostov, Nikolay E. Polyakov, Olga Yu Selyutina, Tatyana G. Tolstikova, Tatyana S. Frolova, Viatcheslav A. Mordvinov, Alexander V. Dushkin & Nikolay Z. Lyakhov. (2019) Disodium salt of glycyrrhizic acid – A novel supramolecular delivery system for anthelmintic drug praziquantel. Journal of Drug Delivery Science and Technology 50, pages 66-77.
Crossref
O.Yu. Selyutina & N.E. Polyakov. (2019) Glycyrrhizic acid as a multifunctional drug carrier – From physicochemical properties to biomedical applications: A modern insight on the ancient drug. International Journal of Pharmaceutics 559, pages 271-279.
Crossref
Ruiping Kong, Xingyi Zhu, Elizaveta S. Meteleva, Nikolay E. Polyakov, Mikhail V. Khvostov, Dmitry S. Baev, Tatjana G. Tolstikova, Alexander V. Dushkin & Weike Su. (2018) Atorvastatin calcium inclusion complexation with polysaccharide arabinogalactan and saponin disodium glycyrrhizate for increasing of solubility and bioavailability. Drug Delivery and Translational Research 8:5, pages 1200-1213.
Crossref