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Expert Opinion on Therapeutic Patents Volume 27, 2017 - Issue 2
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Review

Inhibitors of phospholipase A2 and their therapeutic potential: an update on patents (2012-2016)

Maroula G. KokotouDepartment of Chemistry, National and Kapodistrian University of Athens, Athens, GreeceView further author information
,
Dimitris LimniosDepartment of Chemistry, National and Kapodistrian University of Athens, Athens, GreeceView further author information
,
Aikaterini NikolaouDepartment of Chemistry, National and Kapodistrian University of Athens, Athens, GreeceView further author information
,
Anastasia PsarraDepartment of Chemistry, National and Kapodistrian University of Athens, Athens, GreeceView further author information
&
George KokotosDepartment of Chemistry, National and Kapodistrian University of Athens, Athens, GreeceCorrespondence[email protected]
View further author information
Pages 217-225 | Received 26 Jul 2016, Accepted 05 Oct 2016, Published online: 22 Oct 2016

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Charikleia S. Batsika, Anna-Dimitra D. Gerogiannopoulou, Christiana Mantzourani, Sofia Vasilakaki & George Kokotos. (2021) The design and discovery of phospholipase A2 inhibitors for the treatment of inflammatory diseases. Expert Opinion on Drug Discovery 16:11, pages 1287-1305.
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Sofia Vasilakaki, Johannes Kraml, Michael Schauperl, Klaus R. Liedl & George Kokotos. (2021) Hydration thermodynamics of cytosolic phospholipase A2 GIVA predict its membrane-associated parts and its highly hydrated binding site. Journal of Biomolecular Structure and Dynamics 39:3, pages 953-959.
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J. Abhithaj, K. G. Arun, C. S. Sharanya, M. Haridas & E. Jayadevi Variyar. (2019) Isozymes inhibited by active site blocking: versatility of calcium indifferent hesperidin binding to phospholipase A2 and its significance. Journal of Receptors and Signal Transduction 39:1, pages 60-66.
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Jiangyong Gu, Li Li, Dongmei Wang, Wei Zhu, Ling Han, Ruizhi Zhao, Xiaojie Xu & Chuanjian Lu. (2018) Deciphering metabonomics biomarkers-targets interactions for psoriasis vulgaris by network pharmacology. Annals of Medicine 50:4, pages 323-332.
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Anastasia Psarra, Aikaterini Nikolaou, Maroula G Kokotou, Dimitris Limnios & George Kokotos. (2017) Microsomal prostaglandin E2 synthase-1 inhibitors: a patent review. Expert Opinion on Therapeutic Patents 27:9, pages 1047-1059.
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