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Expert Opinion on Therapeutic Patents Volume 30, 2020 - Issue 7
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Review

Therapeutic modulators of the serotonin 5-HT4 receptor: a patent review (2014-present)

Caroline Lanthiera Normandie Univ, UNICAEN, CERMN (Centre d’Etudes et de Recherche sur le Médicament de Normandie), F-14032 Caen, FranceORCID Iconhttps://orcid.org/0000-0002-5814-3173View further author information
ORCID Icon,
Patrick Dallemagnea Normandie Univ, UNICAEN, CERMN (Centre d’Etudes et de Recherche sur le Médicament de Normandie), F-14032 Caen, FranceORCID Iconhttps://orcid.org/0000-0002-4845-615XView further author information
ORCID Icon,
Cédric Lecouteya Normandie Univ, UNICAEN, CERMN (Centre d’Etudes et de Recherche sur le Médicament de Normandie), F-14032 Caen, FranceORCID Iconhttps://orcid.org/0000-0003-4725-7738View further author information
ORCID Icon,
Sylvie Claeysenb IGF, Univ Montpellier, CNRS, INSERM, Montpellier, FranceORCID Iconhttps://orcid.org/0000-0002-0576-5518View further author information
ORCID Icon &
Christophe Rochaisa Normandie Univ, UNICAEN, CERMN (Centre d’Etudes et de Recherche sur le Médicament de Normandie), F-14032 Caen, FranceCorrespondence[email protected]
ORCID Iconhttps://orcid.org/0000-0001-7996-2082View further author information
ORCID Icon
Pages 495-508 | Received 20 Mar 2020, Accepted 07 May 2020, Published online: 18 Jun 2020

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Martina Bortolami, Daniele Rocco, Antonella Messore, Roberto Di Santo, Roberta Costi, Valentina Noemi Madia, Luigi Scipione & Fabiana Pandolfi. (2021) Acetylcholinesterase inhibitors for the treatment of Alzheimer’s disease – a patent review (2016–present). Expert Opinion on Therapeutic Patents 31:5, pages 399-420.
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Candice M. Roux, Marianne Leger & Thomas Freret. (2021) Memory Disorders Related to Hippocampal Function: The Interest of 5-HT4Rs Targeting. International Journal of Molecular Sciences 22:21, pages 12082.
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Patrick Dallemagne & Christophe Rochais. (2021) 5-HT4R modulators: a patent landscape. Pharmaceutical Patent Analyst.
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Alejandro Castro-Alvarez, Emigdio Chávez-Ángel & Ronald Nelson. (2021) Understanding the Molecular Basis of 5-HT4 Receptor Partial Agonists through 3D-QSAR Studies. International Journal of Molecular Sciences 22:7, pages 3602.
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Amin Charousaei, Mohammad Nasehi, Vahab Babapour, Salar Vaseghi & Mohammad-Reza Zarrindast. (2021) The effect of 5-HT4 serotonin receptors in the CA3 hippocampal region on D-AP5-induced anxiolytic-like effects: Isobolographic analyses. Behavioural Brain Research 397, pages 112933.
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