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Archives of Physiology and Biochemistry
The Journal of Metabolic Diseases
Volume 124, 2018 - Issue 1
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Original Article

Synthesis of chalcone-imide derivatives and investigation of their anticancer and antimicrobial activities, carbonic anhydrase and acetylcholinesterase enzymes inhibition profiles

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Pages 61-68 | Received 18 Jul 2017, Accepted 25 Jul 2017, Published online: 09 Aug 2017

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Murat Boztas, Parham Taslimi, Mirali Akbar Yavari, Ilhami Gulcin, Ertan Sahin & Abdullah Menzek. (2019) Synthesis and biological evaluation of bromophenol derivatives with cyclopropyl moiety: Ring opening of cyclopropane with monoester. Bioorganic Chemistry 89, pages 103017.
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Parham Taslimi, Fatih Mehmet Kandemir, Yeliz Demir, Mustafa İleritürk, Yusuf Temel, Cuneyt Caglayan & İlhami Gulçin. (2019) The antidiabetic and anticholinergic effects of chrysin on cyclophosphamide‐induced multiple organ toxicity in rats: Pharmacological evaluation of some metabolic enzyme activities. Journal of Biochemical and Molecular Toxicology 33:6.
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Beyhan Yiğit, Ruya Kaya, Parham Taslimi, Yılmaz Işık, Muhammet Karaman, Murat Yiğit, İsmail Özdemir & İlhami Gulçin. (2019) Imidazolinium chloride salts bearing wingtip groups: Synthesis, molecular docking and metabolic enzymes inhibition. Journal of Molecular Structure 1179, pages 709-718.
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Adnan Cetin, Fikret Türkan, Parham Taslimi & İlhami Gulçin. (2018) Synthesis and characterization of novel substituted thiophene derivatives and discovery of their carbonic anhydrase and acetylcholinesterase inhibition effects. Journal of Biochemical and Molecular Toxicology 33:3.
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Aydın Aktaş, Duygu Barut Celepci, Ruya Kaya, Parham Taslimi, Yetkin Gök, Muhittin Aygün & İlhami Gülçin. (2019) Novel morpholine liganded Pd-based N-heterocyclic carbene complexes: Synthesis, characterization, crystal structure, antidiabetic and anticholinergic properties. Polyhedron 159, pages 345-354.
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Abel Maharramov, Ruya Kaya, Parham Taslimi, Malahat Kurbanova, Arzu Sadigova, Vagif Farzaliyev, Afsun Sujayev & İlhami Gulçin. (2019) Synthesis, crystal structure, and biological evaluation of optically active 2‐amino‐4‐aryl‐7,7‐dimethyl‐5‐oxo‐5,6,7,8‐tetrahydro‐4 H ‐chromen‐3‐carbonitriles: Antiepileptic, antidiabetic, and anticholinergics potentials . Archiv der Pharmazie 352:2.
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Emre Güzel, Ümit M. Koçyiğit, Barış S. Arslan, Mehmet Ataş, Parham Taslimi, Faik Gökalp, Mehmet Nebioğlu, İlkay Şişman & İlhami Gulçin. (2019) Aminopyrazole‐substituted metallophthalocyanines: Preparation, aggregation behavior, and investigation of metabolic enzymes inhibition properties. Archiv der Pharmazie 352:2.
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Mustafa Zengin, Hayriye Genc, Parham Taslimi, Ali Kestane, Ertugrul Guclu, Aziz Ogutlu, Oguz Karabay & İlhami Gulçin. (2018) Novel thymol bearing oxypropanolamine derivatives as potent some metabolic enzyme inhibitors – Their antidiabetic, anticholinergic and antibacterial potentials. Bioorganic Chemistry 81, pages 119-126.
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Gunel Maharramova, Parham Taslimi, Afsun Sujayev, Vagif Farzaliyev, Lokman Durmaz & İlhami Gulçin. (2018) Synthesis, characterization, antioxidant, antidiabetic, anticholinergic, and antiepileptic properties of novel N‐substituted tetrahydropyrimidines based on phenylthiourea. Journal of Biochemical and Molecular Toxicology 32:12.
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Shahla Daryadel, Ufuk Atmaca, Parham Taslimi, İlhami Gülçin & Murat Çelik. (2018) Novel sulfamate derivatives of menthol: Synthesis, characterization, and cholinesterases and carbonic anhydrase enzymes inhibition properties. Archiv der Pharmazie 351:11, pages 1800209.
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Fikret Turkan, Adnan Cetin, Parham Taslimi & İlhami Gulçin. (2018) Some pyrazoles derivatives: Potent carbonic anhydrase, α‐glycosidase, and cholinesterase enzymes inhibitors. Archiv der Pharmazie 351:10.
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Gulnar Gondolova, Parham Taslimi, Ajdar Medjidov, Vagif Farzaliyev, Afsun Sujayev, Mansura Huseynova, Onur Şahin, Bahattin Yalçın, Fikret Turkan & İlhami Gulçin. (2018) Synthesis, crystal structure and biological evaluation of spectroscopic characterization of Ni(II) and Co(II) complexes with N -salicyloil- N ′-maleoil-hydrazine as anticholinergic and antidiabetic agents . Journal of Biochemical and Molecular Toxicology 32:9, pages e22197.
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Parham Taslimi, Sabiya Osmanova, Cuneyt Caglayan, Fikret Turkan, Sabira Sardarova, Vagif Farzaliyev, Afsun Sujayev, Nastaran Sadeghian & İlhami Gulçin. (2018) Novel amides of 1,1-bis-(carboxymethylthio)-1-arylethanes: Synthesis, characterization, acetylcholinesterase, butyrylcholinesterase, and carbonic anhydrase inhibitory properties. Journal of Biochemical and Molecular Toxicology 32:9, pages e22191.
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Makbule Ekiz, Ahmet Tutar, Salih Ökten, Burcu Bütün, Ümit M. Koçyiğit, Parham Taslimi & Gülaçtı Topçu. (2018) Synthesis, characterization, and SAR of arylated indenoquinoline-based cholinesterase and carbonic anhydrase inhibitors. Archiv der Pharmazie 351:9, pages 1800167.
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Kadir Aksu, Hülya Akıncıoğlu, Akın Akıncıoğlu, Süleyman Göksu, Ferhan Tümer & İlhami Gülçin. (2018) Synthesis of novel sulfamides incorporating phenethylamines and determination of their inhibition profiles against some metabolic enzymes. Archiv der Pharmazie 351:9, pages 1800150.
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Ferhat Türker, Duygu Barut Celepci, Aydın Aktaş, Parham Taslimi, Yetkin Gök, Muhittin Aygün & İlhami Gülçin. (2018) meta -Cyanobenzyl substituted benzimidazolium salts: Synthesis, characterization, crystal structure and carbonic anhydrase, α-glycosidase, butyrylcholinesterase, and acetylcholinesterase inhibitory properties . Archiv der Pharmazie 351:7, pages 1800029.
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Parham Taslimi & İlhami Gulçin. (2018) Antioxidant and anticholinergic properties of olivetol. Journal of Food Biochemistry 42:3, pages e12516.
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Ísmail Çelik, Zeliha Atioğlu, Gamze Ordu, Hayrettin Gezegen & Mehmet Akkurt. (2018) N -(4-Acetylphenyl)- N ′-(4-fluorophenyl)urea . IUCrData 3:4.
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Parham Taslimi, Cuneyt Caglayan, Vagif Farzaliyev, Oruj Nabiyev, Afsun Sujayev, Fikret Turkan, Ruya Kaya & İlhami Gulçin. (2018) Synthesis and discovery of potent carbonic anhydrase, acetylcholinesterase, butyrylcholinesterase, and α-glycosidase enzymes inhibitors: The novel N , N ′-bis-cyanomethylamine and alkoxymethylamine derivatives . Journal of Biochemical and Molecular Toxicology 32:4, pages e22042.
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