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Journal of Enzyme Inhibition and Medicinal Chemistry Volume 17, 2002 - Issue 6
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Research Article

New N -pyridinyl(methyl)-indole-2- and 3-(Alkyl)carboxamides and Derivatives Acting as Systemic and Topical Inflammation Inhibitors

Anne Breteche Laboratoires de Chimie Organique et de Chimie Thérapeutique, UPRES EA 1155, Faculté de Pharmacie, 1 rue Gaston Veil, Université de Nantes, 44035 Nantes Cedex 01- France
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Muriel Duflos Laboratoires de Chimie Organique et de Chimie Thérapeutique, UPRES EA 1155, Faculté de Pharmacie, 1 rue Gaston Veil, Université de Nantes, 44035 Nantes Cedex 01- France
,
Alexandra Dassonville Laboratoires de Chimie Organique et de Chimie Thérapeutique, UPRES EA 1155, Faculté de Pharmacie, 1 rue Gaston Veil, Université de Nantes, 44035 Nantes Cedex 01- France
,
Marie-Renee Nourrisson Laboratoires de Chimie Organique et de Chimie Thérapeutique, UPRES EA 1155, Faculté de Pharmacie, 1 rue Gaston Veil, Université de Nantes, 44035 Nantes Cedex 01- France
,
Jacques Brelet Laboratoires de Chimie Organique et de Chimie Thérapeutique, UPRES EA 1155, Faculté de Pharmacie, 1 rue Gaston Veil, Université de Nantes, 44035 Nantes Cedex 01- France
,
Guillaume Le Baut Laboratoires de Chimie Organique et de Chimie Thérapeutique, UPRES EA 1155, Faculté de Pharmacie, 1 rue Gaston Veil, Université de Nantes, 44035 Nantes Cedex 01- France
,
Nicole Grimaud Laboratoire de Pharmacologie et de Pharmacocinétique, UPRES EA 1155, Faculté de Pharmacie, 1 rue Gaston Veil, Université de Nantes, 44035 Nantes Cedex 01- France
&
Jean-Yves Petit Laboratoire de Pharmacologie et de Pharmacocinétique, UPRES EA 1155, Faculté de Pharmacie, 1 rue Gaston Veil, Université de Nantes, 44035 Nantes Cedex 01- France
 show all
Pages 415-424 | Published online: 30 Sep 2008

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Alexandra Dassonville, Morgane Lardic, Anne Breteche, Marie Renee Nourrisson, Guillaume Le Baut, Nicole Grimaud, Jean-Yves Petit & Muriel Duflos. (2008) N-Pyridinyl(methyl)-indole-1- or 3-propanamides and propenamides acting as topical and systemic inflammation inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 23:5, pages 728-738.
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Andre Kaessler, Marie-Renee Nourrisson, Muriel Duflos & Joachim Jose. (2008) Indole carboxamides inhibit bovine testes hyaluronidase at pH 7.0 and indole acetamides activate the enzyme at pH 3.5 by different mechanisms. Journal of Enzyme Inhibition and Medicinal Chemistry 23:5, pages 719-727.
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Anthony Gallard, Muriel Duflos, Marie-Renee Nourrisson, Guillaume Le Baut, Nicole Grimaud & Jean Yves Petit. (2003) New N-Pyridinyl(methyl)-N1-substituted-3-indolepropanamides Acting as Topical and Systemic Anti-inflammatory Agents. Journal of Enzyme Inhibition and Medicinal Chemistry 18:2, pages 201-208.
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Articles from other publishers (14)

Weiwen Lin, Hanpeng Li, Zhiwen Wu, Jingyi Su, Zehong Zhang, Li Yang, Xianming Deng & Qingyan Xu. (2022) Paspalines C–D and Paxillines B–D: New Indole Diterpenoids from Penicillium brefeldianum WZW-F-69. Marine Drugs 20:11, pages 684.
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Kaja Keček Plešec, Dunja Urbančič, Martina Gobec, Aleksandra Pekošak, Tihomir Tomašič, Marko Anderluh, Irena Mlinarič-Raščan & Žiga Jakopin. (2016) Identification of indole scaffold-based dual inhibitors of NOD1 and NOD2. Bioorganic & Medicinal Chemistry 24:21, pages 5221-5234.
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C Couteau, E. Paparis, C. Chauvet & L. Coiffard. (2015) Tris-biphenyl triazine, a new ultraviolet filter studied in terms of photoprotective efficacy. International Journal of Pharmaceutics 487:1-2, pages 120-123.
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Parthasarathi Subramanian, Satrajit Indu & Krishna P. Kaliappan. (2014) A One-Pot Copper Catalyzed Biomimetic Route to N -Heterocyclic Amides from Methyl Ketones via Oxidative C–C Bond Cleavage . Organic Letters 16:23, pages 6212-6215.
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C. Couteau, C. Chauvet, E. Paparis & L.J.M. Coiffard. (2014) Study of the persistence of the anti-inflammatory effect observed after application of preparations containing organic ultraviolet filters. International Journal of Pharmaceutics 476:1-2, pages 160-163.
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Romain Gastineau, François Turcotte, Jean-Bernard Pouvreau, Michèle Morançais, Joël Fleurence, Eko Windarto, Fiddy Prasetiya, Sulastri Arsad, Pascal Jaouen, Mathieu Babin, Laurence Coiffard, Céline Couteau, Jean-François Bardeau, Boris Jacquette, Vincent Leignel, Yann Hardivillier, Isabelle Marcotte, Nathalie Bourgougnon, Réjean Tremblay, Jean-Sébastien Deschênes, Hope Badawy, Pamela Pasetto, Nikolai Davidovich, Gert Hansen, Jens Dittmer & Jean-Luc Mouget. (2014) Marennine, Promising Blue Pigments from a Widespread Haslea Diatom Species Complex. Marine Drugs 12:6, pages 3161-3189.
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C. Couteau, O. Couteau, C. Chauvet, E. Paparis & L.J.M. Coiffard. (2013) The effect of ultraviolet radiation on the anti-inflammatory effect of filters. International Journal of Pharmaceutics 452:1-2, pages 124-127.
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Céline Couteau, Catherine Chauvet, Eva Paparis & Laurence Coiffard. (2012) UV Filters, Ingredients with a Recognized Anti-Inflammatory Effect. PLoS ONE 7:12, pages e46187.
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Céline Couteau, Catherine Chauvet, Eva Paparis & Laurence J. M. Coiffard. (2012) Influence of certain ingredients on the SPF determined in vivo. Archives of Dermatological Research 304:10, pages 817-821.
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Keika Hattori, Kazuya Yamaguchi, Junichiro Yamaguchi & Kenichiro Itami. (2012) Pd- and Cu-catalyzed C–H arylation of indazoles. Tetrahedron 68:37, pages 7605-7612.
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Delphine Carbonnelle, Morgane Lardic, Alexandra Dassonville, Elise Verron, Jean-Yves Petit, Muriel Duflos & François Lang. (2007) Synthetic N-pyridinyl(methyl)-indol-3-ylpropanamides as new potential immunosuppressive agents. European Journal of Medicinal Chemistry 42:5, pages 686-693.
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S. B. Kale & B. K. Karale. (2009) Synthesis and characterization of some important indazolyl derivatives. Journal of Heterocyclic Chemistry 44:2, pages 289-301.
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Deyi Zhang, Dan Kohlman, Joseph Krushinski, Sidney Liang, Bai-Ping Ying, John E. Reilly, Sean R. Dinn, David B. Wainscott, Suzanne Nutter, Wendy Gough, David L.G. Nelson, John M. Schaus & Yao-Chang Xu. (2004) Design, synthesis and evaluation of bicyclic benzamides as novel 5-HT1F receptor agonists. Bioorganic & Medicinal Chemistry Letters 14:24, pages 6011-6016.
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Alexandra Dassonville, Anne Bretéché, Johan Evano, Muriel Duflos, Guillaume le Baut, Nicole Grimaud & Jean-Yves Petit. (2004) New N-pyridinyl(methyl)-indolalkanamides acting as topical inflammation inhibitors. Bioorganic & Medicinal Chemistry Letters 14:21, pages 5441-5444.
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