- Robert, J.M.H., Robert-Piessard, S., Courant J., Le Baut, G., Robert, B., Lang, F., Petit, J.Y., Grimaud, N. and Welin, L. (1995) "Non-carboxylic antiinflammatory compounds. III. N-(4,6-Dimethylpyridm-2-yl)arylcarboxamides and arylthiocarboxamides acting as brain edema inhibitors", European Journal of Medicinal Chemistry 30,915-924.
- Collin, X., Robert, J.M.H., Wielgosz, G., Le Baut, G., Bobin-Dubigeon, C., Grimaud, N. and Petit, J.Y. (2001) "New anti-inflammatory N-pyridinyl(alkyl)phthalimides acting as tumour necrosis factor-a production inhibitors", European Journal of Medicinal Chemistry 36, 639-649.
- Duflos, M., Nourrisson, M.R., Brelet, J., Courant, J., Le Baut, G., Grimaud, N. and Petit, J.Y. (2001) "N-pyridinyl-indol-3(alkyl)carboxamides and derivatives as potential systemic and topical inflammation inhibitors", European Journal of Medicinal Chemistry 36,545-553.
- Fagan, G.P., Chapleo, C.B., Lane, A.C., Myers, M., Roach, A.G., Smith, C.F.C., Stillings, M.R. and Welbourn, A.P. (1988) "Indoline analogues of idazoxan: potent a2-antagonists and a1-agonists", Journal of Medicinal Chemistry 31,944-948.
- Winter, C.A., Risley, E.A. and Nuss, G.W. (1962) "Carrageenin-induced oedema in hind paw of the rat as an assay for anti-inflammatory drugs", Proceedings of the Society for Experimental Biology and Medicine 111, 544-547.
- Carlson, R.P., O'Neill, D.D., Chang, J. and Lewis, A.J. (1985) "Modulation of mouse ear edema by cydooxygenase and lipoxygenase inhibitors and other pharmacologic agents", Agents Actions 17,197-204.
- Snyder, H.R., Thompson, C.B. and Hinman, R.L. (1952) "The synthesis of an indazole analog of DL-tryptophan", Journal of the American Chemical Society 74,2009-2012.
- Ferrari, M., Ripa, A., Ripa, G. and Sisti, M. (1989) "An improved synthesis of indazole-3-carboxylic acid", Journal of Heterocyclic Chemistry 26,531-532.
- Curtin, M.L., Davidsen, S.K., Heyman, H.R., Garland, R.B., Sheppard, G.S., Florjancic, A.S., Xu, L., Carrera, Jr., G.M., Steinman, D.H., Trautmann, J.A., Albert D.H., Magoc, T.J., Tapang, P., Rhein, D.A., Conway, R.G., Luo, G., Denissen, J.F., Marsh, K.C., Morgan, D.W. and Summers, J.B. (1998) "Discovery and evaluation of a series of 3-acylindole imidazopyridine platelet activating factor antagonists", Journal of Medicinal Chemistry 41, 74-95.
- Zenitz, B.L. (1996) "1-[(3-, 2-, and 1-indolyl)lower-alkyl-, lower-alkenyl-, and lower-alkylyl]piperidines". US Patent, 3, 238,215.
- Fouchard, F., Marchand, P., Le Baut, G., Emig, P. and Nickel, B. (2001) "Synthesis and pharmacological evaluation of (indol-3-yl)alkylamides as potent analgesic agents", Arzneimittel-Forschung/Drug Research 51,814-824.
- Yoshida, T., Matsuura, N., Yamamoto, K., Doi, M., Shimada, K., Morie, T. and Kato, S. (1996) "Practical synthesis of 1Hindazole-3-carboxylic acid and its derivatives", Heterocycles 43,2701-2712.
- Collin, X., Robert, J.M., Duflos, M., Wielgosz, G., Le Baut G., Bobin-Dubigeon, C., Grimaud, N., Lang, F. and Petit, J.Y. (2000) "Synthesis of N-pyridinyl(methyl)-1,2-dihydro-4-hydroxy-2-oxoquinoline-3-carboxamides and analogues andtheir anti-inflammatory activity in mice and rats", Journal ofPharmacy and Pharmacology 53,417-423.
- Voohrees, J.J. (1983) "Leukotrienes and other lipoxygenaseproducts in the pathogenesis and therapy of psoriasis andother dermatoses", Archives of Dermatology 119,541-547.
- Schwarz, T. and Lugert, E. (1992) "Pharmacology of cytokinesin the skin", Pharmacology of the Skin (CRC Press, BocaRaton, FL), pp. 283-313.
- Alfort, G.J., Stanley, P.L. and Todderud, G. (1992) "Infiltrationof leukocyte subsets into mouse skin inflammation withphorbol ester", Agents Actions 37,260-267.
Free access
New N -pyridinyl(methyl)-indole-2- and 3-(Alkyl)carboxamides and Derivatives Acting as Systemic and Topical Inflammation Inhibitors
Reprints and Corporate Permissions
Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?
To request a reprint or corporate permissions for this article, please click on the relevant link below:
Academic Permissions
Please note: Selecting permissions does not provide access to the full text of the article, please see our help page How do I view content?
Obtain permissions instantly via Rightslink by clicking on the button below:
If you are unable to obtain permissions via Rightslink, please complete and submit this Permissions form. For more information, please visit our Permissions help page.
Related research
People also read lists articles that other readers of this article have read.
Recommended articles lists articles that we recommend and is powered by our AI driven recommendation engine.
Cited by lists all citing articles based on Crossref citations.
Articles with the Crossref icon will open in a new tab.