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Research Article

Quantitative structure-activity relationships (QSARs) in inhibitors of various cytochromes P450: The importance of compound lipophilicity

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Pages 1-6 | Received 24 Feb 2006, Accepted 17 Jul 2006, Published online: 20 Oct 2008

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Robert J. Young, Darren V.S. Green, Christopher N. Luscombe & Alan P. Hill. (2011) Getting physical in drug discovery II: the impact of chromatographic hydrophobicity measurements and aromaticity. Drug Discovery Today 16:17-18, pages 822-830.
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Marie M. Ahlström & Ismael Zamora. (2008) Characterization of Type II Ligands in CYP2C9 and CYP3A4. Journal of Medicinal Chemistry 51:6, pages 1755-1763.
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