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Journal of Enzyme Inhibition and Medicinal Chemistry Volume 34, 2019 - Issue 1
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Original Articles

Synthesis and characterisation of a new benzamide-containing nitrobenzoxadiazole as a GSTP1-1 inhibitor endowed with high stability to metabolic hydrolysis

Veronica Di PaoloDepartment of Pharmaceutical and Pharmacological Sciences, University of Padova, Padova, Italy; View further author information
,
Chiara FulciDepartment of Experimental Medicine, “Tor Vergata” University of Rome, Rome, Italy; View further author information
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Dante RotiliDepartment of Drug Chemistry and Technologies, “Sapienza” University of Rome, Rome, Italy; ORCID Iconhttp://orcid.org/0000-0002-8428-8763View further author information
ORCID Icon,
Francesca SciarrettaDepartment of Experimental Medicine, “Tor Vergata” University of Rome, Rome, Italy; View further author information
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Alessia LucidiDepartment of Drug Chemistry and Technologies, “Sapienza” University of Rome, Rome, Italy; View further author information
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Blasco Morozzo della RoccaDepartment of Biology, “Tor Vergata” University of Rome, Rome, Italy; View further author information
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Anastasia De LucaDepartment of Biology, “Tor Vergata” University of Rome, Rome, Italy; View further author information
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Antonio RosatoDepartment of Surgery, Oncology and Gastroenterology, University of Padova, Padova, Italy; ;Istituto Oncologico Veneto IRCCS, Padova, Italy; Correspondence[email protected]
ORCID Iconhttp://orcid.org/0000-0002-5263-8386View further author information
ORCID Icon,
Luigi QuintieriDepartment of Pharmaceutical and Pharmacological Sciences, University of Padova, Padova, Italy; Correspondence[email protected]
ORCID Iconhttp://orcid.org/0000-0001-7403-0921View further author information
ORCID Icon &
Anna Maria CaccuriDepartment of Experimental Medicine, “Tor Vergata” University of Rome, Rome, Italy; ;The NAST Centre for Nanoscience and Nanotechnology and Innovative Instrumentation, “Tor Vergata” University of Rome, Rome, ItalyCorrespondence[email protected]
ORCID Iconhttp://orcid.org/0000-0002-3756-4163View further author information
ORCID Icon show all
Pages 1131-1139 | Received 27 Mar 2019, Accepted 05 May 2019, Published online: 06 Jun 2019

Citations (7)

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Patrick E. Hanna & M. W. Anders. (2019) The mercapturic acid pathway. Critical Reviews in Toxicology 49:10, pages 819-929.
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Articles from other publishers (6)

Kebin Xu, Ziyi Chen, Jialong Hou, Chenlin Dong, Chengge Shi, Linglin Gao, Zhixian Huang, Ge Shen, Te Wang & Yan Zhou. (2022) Praeruptorin B inhibits osteoclastogenesis by targeting GSTP1 and impacting on the S-glutathionylation of IKKβ. Biomedicine & Pharmacotherapy 154, pages 113529.
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Giulia Siciliano, Veronica Di Paolo, Dante Rotili, Rossella Migale, Francesca Pedini, Marialuisa Casella, Serena Camerini, Daniele Dalzoppo, Rob Henderson, Tonnie Huijs, Koen J. Dechering, Antonello Mai, Anna Maria Caccuri, Marco Lalle, Luigi Quintieri & Pietro Alano. (2022) The Nitrobenzoxadiazole Derivative NBDHEX Behaves as Plasmodium falciparum Gametocyte Selective Inhibitor with Malaria Parasite Transmission Blocking Activity. Pharmaceuticals 15:2, pages 168.
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Ross S. Mancini, Christopher J. Barden, Donald F. Weaver & Mark A. Reed. (2021) Furazans in Medicinal Chemistry. Journal of Medicinal Chemistry 64:4, pages 1786-1815.
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Lei Wang & Todd L. Lowary. (2020) Synthesis of Rhamnolipid Derivatives Containing Ester Isosteres. Organic Letters 22:24, pages 9633-9637.
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Veronica Di Paolo, Chiara Fulci, Dante Rotili, Anastasia De Luca, Stefano Tomassi, Massimo Serra, Manuel Scimeca, Cristina Geroni, Luigi Quintieri & Anna Maria Caccuri. (2020) Characterization of water-soluble esters of nitrobenzoxadiazole-based GSTP1-1 inhibitors for cancer treatment. Biochemical Pharmacology 178, pages 114060.
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Imane Almi, Salah Belaidi, Enfale Zerroug, Mebarka Alloui, Ridha Ben Said, Roberto Linguerri & Majdi Hochlaf. (2020) QSAR investigations and structure-based virtual screening on a series of nitrobenzoxadiazole derivatives targeting human glutathione-S-transferases. Journal of Molecular Structure 1211, pages 128015.
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