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Journal of Enzyme Inhibition and Medicinal Chemistry Volume 34, 2019 - Issue 1
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Research Paper

Synthesis and biological evaluation of novel 8-substituted quinoline-2-carboxamides as carbonic anhydrase inhibitors

Pavitra S. ThackerDepartment of Medicinal Chemistry, National Institute of Pharmaceutical Education and Research (NIPER), Hyderabad, India; View further author information
,
Pirpasha ShaikhDepartment of Medicinal Chemistry, National Institute of Pharmaceutical Education and Research (NIPER), Hyderabad, India; View further author information
,
Andrea AngeliNeurofarba Department, Section of Pharmaceutical Chemistry, University of Florence, Florence, ItalyORCID Iconhttp://orcid.org/0000-0002-1470-7192View further author information
ORCID Icon,
Mohammed ArifuddinDepartment of Medicinal Chemistry, National Institute of Pharmaceutical Education and Research (NIPER), Hyderabad, India; Correspondence[email protected]
View further author information
&
Claudiu T. SupuranNeurofarba Department, Section of Pharmaceutical Chemistry, University of Florence, Florence, ItalyCorrespondence[email protected]
ORCID Iconhttp://orcid.org/0000-0003-4262-0323View further author information
ORCID Icon
Pages 1172-1177 | Received 02 May 2019, Accepted 28 May 2019, Published online: 20 Jun 2019

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Yogesh Walunj, Abhijit Shinde, Krishna Borde, Yogita Abhale, Vivek Bobade & Pravin C. Mhaske. (2022) Synthesis, Anticancer and Antimicrobial Screening of New Naphthalenyl-Thiazole and Quinolinyl-Thiazole. Polycyclic Aromatic Compounds 42:10, pages 6891-6907.
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Sinan Bilginer, Halise Inci Gul, Feyza Sena Erdal, Hiroshi Sakagami, Serkan Levent, Ilhami Gulcin & Claudiu T. Supuran. (2019) Synthesis, cytotoxicities, and carbonic anhydrase inhibition potential of 6-(3-aryl-2-propenoyl)-2(3H)-benzoxazolones. Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 1722-1729.
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Małgorzata Jeleń, Beata Morak-Młodawska & Rafał Korlacki. (2023) Anticancer activities of tetra-, penta-, and hexacyclic phenothiazines modified with quinoline moiety.. Journal of Molecular Structure 1287, pages 135700.
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Moataz Shaldam, Alessio Nocentini, Zainab M. Elsayed, Tamer M. Ibrahim, Rofaida Salem, Ramadan A. El-Domany, Clemente Capasso, Claudiu T. Supuran & Wagdy M. Eldehna. (2021) Development of Novel Quinoline-Based Sulfonamides as Selective Cancer-Associated Carbonic Anhydrase Isoform IX Inhibitors. International Journal of Molecular Sciences 22:20, pages 11119.
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N. Stellenboom, R. Hunter, M. Caira, A. Oztekin & K. Zilbeyaz. (2021) Unsymmetrical Cysteine Disulfides as Carbonic Anhydrase Inhibitors. Russian Journal of Bioorganic Chemistry 47:5, pages 1020-1027.
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Sinan Bilginer, Halise I. Gul, Baris Anil, Yeliz Demir & Ilhami Gulcin. (2020) Synthesis and in silico studies of triazene‐substituted sulfamerazine derivatives as acetylcholinesterase and carbonic anhydrases inhibitors. Archiv der Pharmazie 354:1, pages 2000243.
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Pavitra S. Thacker, Nerella Sridhar Goud, Omkar S. Argulwar, Jyothsna Soman, Andrea Angeli, Mallika Alvala, Mohammed Arifuddin & Claudiu T. Supuran. (2020) Synthesis and biological evaluation of some coumarin hybrids as selective carbonic anhydrase IX and XII inhibitors. Bioorganic Chemistry 104, pages 104272.
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Sinan Bilginer, Halise I. Gul, Feyza S. Erdal, Hiroshi Sakagami & Ilhami Gulcin. (2020) New halogenated chalcones with cytotoxic and carbonic anhydrase inhibitory properties: 6‐(3‐Halogenated phenyl‐2‐propen‐1‐oyl)‐2(3 H )‐benzoxazolones . Archiv der Pharmazie 353:6, pages 1900384.
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Pavitra S. Thacker, Andrea Angeli, Omkar S. Argulwar, Prerna L. Tiwari, Mohammed Arifuddin & Claudiu T. Supuran. (2020) Design, synthesis and biological evaluation of coumarin linked 1,2,4-oxadiazoles as selective carbonic anhydrase IX and XII inhibitors. Bioorganic Chemistry 98, pages 103739.
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Sinan BİLGİNER. (2020) Benzoksazolon Türevi Şalkon Bileşiklerinin Sentezi ve Biyoaktivitelerinin AraştırılmasıSynthesis and Bioactivities of Benzoxazolone Derivative Chalcone Compounds. Erzincan Üniversitesi Fen Bilimleri Enstitüsü Dergisi 13:1, pages 334-347.
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