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Journal of Enzyme Inhibition and Medicinal Chemistry Volume 34, 2019 - Issue 1
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Research Paper

Exploring new structural features of the 4-[(3-methyl-4-aryl-2,3-dihydro-1,3-thiazol-2-ylidene)amino]benzenesulphonamide scaffold for the inhibition of human carbonic anhydrases

Simona DistintoDepartment of Life and Environmental Sciences, University of Cagliari, Cagliari, Italy; ORCID Iconhttps://orcid.org/0000-0003-1620-6225
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Rita MeledduDepartment of Life and Environmental Sciences, University of Cagliari, Cagliari, Italy; Correspondence[email protected]
ORCID Iconhttps://orcid.org/0000-0003-1629-7454
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Francesco OrtusoDipartimento di Scienze della Salute, Università Magna Graecia di Catanzaro, Catanzaro, Italy; ORCID Iconhttps://orcid.org/0000-0001-6235-8161
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Filippo CottigliaDepartment of Life and Environmental Sciences, University of Cagliari, Cagliari, Italy;
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Serenella DeplanoDepartment of Life and Environmental Sciences, University of Cagliari, Cagliari, Italy;
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Lisa SequeiraDepartment of Life and Environmental Sciences, University of Cagliari, Cagliari, Italy; ORCID Iconhttps://orcid.org/0000-0002-5801-9455
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Claudia MelisDepartment of Life and Environmental Sciences, University of Cagliari, Cagliari, Italy;
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Benedetta FoisDepartment of Life and Environmental Sciences, University of Cagliari, Cagliari, Italy;
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Andrea AngeliDipartimento NEUROFARBA, Sezione di Scienze Farmaceutiche, Università degli Studi di Firenze, Sesto Fiorentino, Italy; ORCID Iconhttp://orcid.org/0000-0002-1470-7192
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Clemente CapassoIstituto di Bioscienze e Biorisorse, CNR, Napoli, Italy; ORCID Iconhttp://orcid.org/0000-0003-3314-2411
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Rossella AngiusLaboratorio NMR e Tecnologie Bioanalitiche, Pula, Italy
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Stefano AlcaroDipartimento di Scienze della Salute, Università Magna Graecia di Catanzaro, Catanzaro, Italy; ORCID Iconhttps://orcid.org/0000-0002-0437-358X
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Claudiu T. SupuranDipartimento NEUROFARBA, Sezione di Scienze Farmaceutiche, Università degli Studi di Firenze, Sesto Fiorentino, Italy; Correspondence[email protected]
ORCID Iconhttp://orcid.org/0000-0003-4262-0323
ORCID Icon &
Elias MaccioniDepartment of Life and Environmental Sciences, University of Cagliari, Cagliari, Italy; ORCID Iconhttps://orcid.org/0000-0003-2175-2802
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Pages 1526-1533 | Received 18 Jun 2019, Accepted 06 Aug 2019, Published online: 20 Aug 2019

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Lisa Sequeira, Simona Distinto, Rita Meleddu, Marco Gaspari, Andrea Angeli, Filippo Cottiglia, Daniela Secci, Alessia Onali, Erica Sanna, Fernanda Borges, Eugenio Uriarte, Stefano Alcaro, Claudiu T. Supuran & Elias Maccioni. (2023) 2H-chromene and 7H-furo-chromene derivatives selectively inhibit tumour associated human carbonic anhydrase IX and XII isoforms. Journal of Enzyme Inhibition and Medicinal Chemistry 38:1.
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Claudiu T. Supuran. (2020) Coumarin carbonic anhydrase inhibitors from natural sources. Journal of Enzyme Inhibition and Medicinal Chemistry 35:1, pages 1462-1470.
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Articles from other publishers (6)

Nurcan Berber, Arif Sercan Şahutoğlu, Başak Gökçe, Kübra Çıkrıkçı & Nahit Gençer. (2023) Synthesis, characterization, carbonic anhydrase inhibitor activity, and docking studies of phenylthiazol-2(3h)-ylidene-isoquinoline-5-amine Derivatives. Journal of Molecular Structure 1291, pages 136061.
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Pavitra S. Thacker, Vaishnavi Newaskar, Andrea Angeli, Dilep Kumar Sigalapalli, Nerella Sridhar Goud, Hepsibha Chirra, Afzal B. Shaik, Mohammed Arifuddin & Claudiu T. Supuran. (2022) Synthesis and biological evaluation of coumarin‐thiazole hybrids as selective carbonic anhydrase IX and XII inhibitors. Archiv der Pharmazie 355:12.
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Sergei Simakov, Victor Kartsev, Anthi Petrou, Ioannis Nicolaou, Athina Geronikaki, Marija Ivanov, Marina Kostic, Jasmina Glamočlija, Marina Soković, Despoina Talea & Ioannis S. Vizirianakis. (2021) 4-(Indol-3-yl)thiazole-2-amines and 4-ιndol-3-yl)thiazole Acylamines as Νovel Antimicrobial Agents: Synthesis, In Silico and In Vitro Evaluation. Pharmaceuticals 14:11, pages 1096.
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András Gy. Németh, Bence Marlok, Attila Domján, Qinghe Gao, Xinya Han, György M. Keserű & Péter Ábrányi‐Balogh. (2021) Convenient Multicomponent One‐Pot Synthesis of 2‐Iminothiazolines and 2‐Aminothiazoles Using Elemental Sulfur Under Aqueous Conditions. European Journal of Organic Chemistry 2021:25, pages 3587-3597.
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Anthi Petrou, Maria Fesatidou & Athina Geronikaki. (2021) Thiazole Ring—A Biologically Active Scaffold. Molecules 26:11, pages 3166.
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Rita Meleddu, Simona Distinto, Filippo Cottiglia, Rossella Angius, Pierluigi Caboni, Andrea Angeli, Claudia Melis, Serenella Deplano, Stefano Alcaro, Francesco Ortuso, Claudiu T. Supuran & Elias Maccioni. (2020) New Dihydrothiazole Benzensulfonamides: Looking for Selectivity toward Carbonic Anhydrase Isoforms I, II, IX, and XII. ACS Medicinal Chemistry Letters 11:5, pages 852-856.
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