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Journal of Enzyme Inhibition and Medicinal Chemistry Volume 35, 2020 - Issue 1
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Research Paper

The structural basis for the selectivity of sulfonamido dicarbaboranes toward cancer-associated carbonic anhydrase IX

Michael Kuglera Deparment of Structural Biology, Institute of Organic Chemistry and Biochemistry of the Czech Academy of Sciences, Prague, Czech Republic;b Deparment of Structural Biology, Institute of Molecular Genetics of the Czech Academy of Sciences, Prague, Czech RepublicORCID Iconhttps://orcid.org/0000-0002-0752-9682View further author information
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Josef Holubc Department of Syntheses, Institute of Inorganic Chemistry of the Czech Academy of Sciences, Řež, Czech RepublicView further author information
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Jiří Bryndaa Deparment of Structural Biology, Institute of Organic Chemistry and Biochemistry of the Czech Academy of Sciences, Prague, Czech Republic;b Deparment of Structural Biology, Institute of Molecular Genetics of the Czech Academy of Sciences, Prague, Czech RepublicORCID Iconhttps://orcid.org/0000-0003-3675-6769View further author information
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Klára Pospíšilováa Deparment of Structural Biology, Institute of Organic Chemistry and Biochemistry of the Czech Academy of Sciences, Prague, Czech RepublicView further author information
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Suzan El Anwarc Department of Syntheses, Institute of Inorganic Chemistry of the Czech Academy of Sciences, Řež, Czech RepublicView further author information
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Dmytro Bavolc Department of Syntheses, Institute of Inorganic Chemistry of the Czech Academy of Sciences, Řež, Czech RepublicView further author information
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Miroslav Havránekd Chemistry Department, Apigenex, s.r.o., Prague, Czech RepublicView further author information
,
Vlastimil Králb Deparment of Structural Biology, Institute of Molecular Genetics of the Czech Academy of Sciences, Prague, Czech RepublicView further author information
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Milan Fábryb Deparment of Structural Biology, Institute of Molecular Genetics of the Czech Academy of Sciences, Prague, Czech RepublicView further author information
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Bohumír Grünerc Department of Syntheses, Institute of Inorganic Chemistry of the Czech Academy of Sciences, Řež, Czech RepublicCorrespondence[email protected]
ORCID Iconhttps://orcid.org/0000-0002-2595-9125View further author information
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Pavlína Řezáčováa Deparment of Structural Biology, Institute of Organic Chemistry and Biochemistry of the Czech Academy of Sciences, Prague, Czech Republic;b Deparment of Structural Biology, Institute of Molecular Genetics of the Czech Academy of Sciences, Prague, Czech RepublicCorrespondence[email protected]
ORCID Iconhttps://orcid.org/0000-0001-9626-346XView further author information
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Pages 1800-1810 | Received 22 May 2020, Accepted 21 Aug 2020, Published online: 23 Sep 2020

Citations (8)

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Mateusz Kciuk, Adrianna Gielecińska, Somdutt Mujwar, Mariusz Mojzych, Beata Marciniak, Rafał Drozda & Renata Kontek. (2022) Targeting carbonic anhydrase IX and XII isoforms with small molecule inhibitors and monoclonal antibodies. Journal of Enzyme Inhibition and Medicinal Chemistry 37:1, pages 1278-1298.
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Wenting Chen, Jinxi Liu, Caiyun Zheng, Que Bai, Qian Gao, Yanni Zhang, Kai Dong & Tingli Lu. (2022) Research Progress on Improving the Efficiency of CDT by Exacerbating Tumor Acidification. International Journal of Nanomedicine 17, pages 2611-2628.
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Articles from other publishers (6)

Simone Giovannuzzi, Anna Nikitjuka, Bruna Rafaela Pereira Resende, Michael Smietana, Alessio Nocentini, Claudiu T. Supuran & Jean-Yves Winum. (2024) Boron-containing carbonic anhydrases inhibitors. Bioorganic Chemistry 143, pages 106976.
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Sebastian Braun, Svetlana Paskas, Markus Laube, Sven George, Bettina Hofmann, Peter Lönnecke, Dieter Steinhilber, Jens Pietzsch, Sanja S. Mijatović, Danijela Maksimović‐Ivanić & Evamarie Hey‐Hawkins. (2023) In Vitro Cytostatic Effect on Tumor Cells by Carborane‐Based Dual Cyclooxygenase‐2 and 5‐Lipoxygenase Inhibitors. Advanced Therapeutics 6:4.
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Michael Kugler, Martin Hadzima, Rastislav Dzijak, Robert Rampmaier, Pavel Srb, Lukáš Vrzal, Zdeněk Voburka, Pavel Majer, Pavlína Řezáčová & Milan Vrabel. (2023) Identification of specific carbonic anhydrase inhibitors via in situ click chemistry, phage-display and synthetic peptide libraries: comparison of the methods and structural study . RSC Medicinal Chemistry 14:1, pages 144-153.
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Jindřich Fanfrlík, Jiří Brynda, Michael Kugler, Martin Lepšík, Klára Pospíšilová, Josef Holub, Drahomír Hnyk, Jan Nekvinda, Bohumír Grüner & Pavlína Řezáčová. (2023) B–H⋯π and C–H⋯π interactions in protein–ligand complexes: carbonic anhydrase II inhibition by carborane sulfonamides. Physical Chemistry Chemical Physics 25:3, pages 1728-1733.
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An-Ping Xiang, Xiao-Nong Chen, Peng-Fei Xu, Si-Hai Shao & Yue-Fan Shen. (2022) Expression and prognostic value of carbonic anhydrase IX (CA-IX) in bladder urothelial carcinoma. BMC Urology 22:1.
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Michael Kugler, Jan Nekvinda, Josef Holub, Suzan El Anwar, Viswanath Das, Václav Šícha, Klára Pospíšilová, Milan Fábry, Vlastimil Král, Jiří Brynda, Václav Kašička, Marián Hajdúch, Pavlína Řezáčová & Bohumír Grüner. (2021) Inhibitors of CA IX Enzyme Based on Polyhedral Boron Compounds. ChemBioChem 22:18, pages 2741-2761.
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