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Journal of Enzyme Inhibition and Medicinal Chemistry Volume 36, 2021 - Issue 1
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Brief Report

Selective inhibition of carbonic anhydrase IX and XII by coumarin and psoralen derivatives

Rita Meleddua Department of Life and Environmental Sciences, University of Cagliari, Monserrato, ItalyORCID Iconhttps://orcid.org/0000-0003-1629-7454
ORCID Icon,
Serenella Deplanoa Department of Life and Environmental Sciences, University of Cagliari, Monserrato, Italy
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Elias Maccionia Department of Life and Environmental Sciences, University of Cagliari, Monserrato, ItalyCorrespondence[email protected]
ORCID Iconhttps://orcid.org/0000-0003-2175-2802
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Francesco Ortusob Dipartimento di Scienze della Salute, Università Magna Graecia di Catanzaro, Catanzaro, ItalyORCID Iconhttps://orcid.org/0000-0001-6235-8161
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Filippo Cottigliaa Department of Life and Environmental Sciences, University of Cagliari, Monserrato, Italy
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Daniela Seccia Department of Life and Environmental Sciences, University of Cagliari, Monserrato, Italy
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Alessia Onalia Department of Life and Environmental Sciences, University of Cagliari, Monserrato, Italy
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Erica Sannaa Department of Life and Environmental Sciences, University of Cagliari, Monserrato, Italy
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Andrea Angelic Dipartimento NEUROFARBA, Sezione di Scienze Farmaceutiche, Università degli Studi di Firenze, Sesto Fiorentino, ItalyORCID Iconhttps://orcid.org/0000-0002-1470-7192
ORCID Icon,
Rossella Angiusd Laboratorio NMR e Tecnologie Bioanalitiche, Sardegna Ricerche, Pula, Italy
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Stefano Alcarob Dipartimento di Scienze della Salute, Università Magna Graecia di Catanzaro, Catanzaro, ItalyORCID Iconhttps://orcid.org/0000-0002-0437-358X
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Claudiu T. Supuranc Dipartimento NEUROFARBA, Sezione di Scienze Farmaceutiche, Università degli Studi di Firenze, Sesto Fiorentino, ItalyCorrespondence[email protected]
ORCID Iconhttps://orcid.org/0000-0003-4262-0323
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Simona Distintoa Department of Life and Environmental Sciences, University of Cagliari, Monserrato, ItalyORCID Iconhttps://orcid.org/0000-0003-1620-6225
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Pages 685-692 | Received 08 Jan 2021, Accepted 01 Feb 2021, Published online: 18 Feb 2021

Citations (13)

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Lisa Sequeira, Simona Distinto, Rita Meleddu, Marco Gaspari, Andrea Angeli, Filippo Cottiglia, Daniela Secci, Alessia Onali, Erica Sanna, Fernanda Borges, Eugenio Uriarte, Stefano Alcaro, Claudiu T. Supuran & Elias Maccioni. (2023) 2H-chromene and 7H-furo-chromene derivatives selectively inhibit tumour associated human carbonic anhydrase IX and XII isoforms. Journal of Enzyme Inhibition and Medicinal Chemistry 38:1.
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Satyajit Khatua & Srabani Taraphder. (2023) In the footsteps of an inhibitor unbinding from the active site of human carbonic anhydrase II. Journal of Biomolecular Structure and Dynamics 41:8, pages 3187-3204.
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Mateusz Kciuk, Adrianna Gielecińska, Somdutt Mujwar, Mariusz Mojzych, Beata Marciniak, Rafał Drozda & Renata Kontek. (2022) Targeting carbonic anhydrase IX and XII isoforms with small molecule inhibitors and monoclonal antibodies. Journal of Enzyme Inhibition and Medicinal Chemistry 37:1, pages 1278-1298.
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Simone Giovannuzzi, Viviana De Luca, Alessio Nocentini, Clemente Capasso & Claudiu T. Supuran. (2022) Coumarins inhibit η-class carbonic anhydrase from Plasmodium falciparum. Journal of Enzyme Inhibition and Medicinal Chemistry 37:1, pages 680-685.
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Yinbo Pan, Teng Liu, Xiaojing Wang & Jie Sun. (2022) Research progress of coumarins and their derivatives in the treatment of diabetes. Journal of Enzyme Inhibition and Medicinal Chemistry 37:1, pages 616-628.
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Simone Giovannuzzi, Chad S. Hewitt, Alessio Nocentini, Clemente Capasso, Daniel P. Flaherty & Claudiu T. Supuran. (2022) Coumarins effectively inhibit bacterial α-carbonic anhydrases. Journal of Enzyme Inhibition and Medicinal Chemistry 37:1, pages 333-338.
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Alma Fuentes-Aguilar, Penélope Merino-Montiel, Sara Montiel-Smith, Socorro Meza-Reyes, José Luis Vega-Báez, Adrián Puerta, Miguel X. Fernandes, José M. Padrón, Andrea Petreni, Alessio Nocentini, Claudiu T. Supuran, Óscar López & José G. Fernández-Bolaños. (2022) 2-Aminobenzoxazole-appended coumarins as potent and selective inhibitors of tumour-associated carbonic anhydrases. Journal of Enzyme Inhibition and Medicinal Chemistry 37:1, pages 168-177.
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Articles from other publishers (6)

Angélica Salinas-Torres, Elizabeth Jiménez, Diana Becerra, José J. Martínez, Hugo Rojas, Juan-Carlos Castillo & Mario A. Macías. (2023) Synthesis, anticancer evaluation, thermal and X-ray crystallographic analysis of 2-oxo-2H-chromen-7-yl 4-chlorobenzoate using a conductively heated sealed-vessel reactor. Journal of Molecular Structure 1274, pages 134414.
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Nadia Arif, Zahid Shafiq, Khalid Mahmood, Muhammad Rafiq, Sadia Naz, Sohail Anjum Shahzad, Umar Farooq, Ali H. Bahkali, Abdallah M. Elgorban, Muhammad Yaqub & Ahmed El-Gokha. (2022) Synthesis, Biological Evaluation, and In Silico Studies of Novel Coumarin-Based 4 H ,5 H -pyrano[3,2- c ]chromenes as Potent β-Glucuronidase and Carbonic Anhydrase Inhibitors . ACS Omega 7:32, pages 28605-28617.
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Pavitra S. Thacker, Arifuddin Mohammed, Claudiu T. Supuran, Prerna L. Tiwari, Nerella S. Goud, Danaboina Srikanth & Andrea Angeli. (2022) Synthesis and Biological Evaluation of Coumarin Carboxamides as Selective and Potent Inhibitors of Carbonic Anhydrases IX and XII. Anti-Cancer Agents in Medicinal Chemistry 22:14, pages 2647-2654.
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Giulia Arrighi, Adrián Puerta, Andrea Petrini, Francisco J. Hicke, Alessio Nocentini, Miguel X. Fernandes, José M. Padrón, Claudiu T. Supuran, José G. Fernández-Bolaños & Óscar López. (2022) Squaramide-Tethered Sulfonamides and Coumarins: Synthesis, Inhibition of Tumor-Associated CAs IX and XII and Docking Simulations. International Journal of Molecular Sciences 23:14, pages 7685.
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Dmitry Dar'in, Grigory Kantin, Stanislav Kalinin, Tatiana Sharonova, Alexander Bunev, Gennady I. Ostapenko, Alessio Nocentini, Vladimir Sharoyko, Claudiu T. Supuran & Mikhail Krasavin. (2021) Investigation of 3-sulfamoyl coumarins against cancer-related IX and XII isoforms of human carbonic anhydrase as well as cancer cells leads to the discovery of 2-oxo-2H-benzo[h]chromene-3-sulfonamide – A new caspase-activating proapoptotic agent. European Journal of Medicinal Chemistry 222, pages 113589.
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Diana Becerra, Jaime Portilla & Juan-Carlos Castillo. (2021) 2-Oxo-2H-chromen-7-yl 4-chlorobenzoate. Molbank 2021:3, pages M1279.
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