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Journal of Enzyme Inhibition and Medicinal Chemistry Volume 36, 2021 - Issue 1
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Research Paper

Development of 3-methyl/3-(morpholinomethyl)benzofuran derivatives as novel antitumor agents towards non-small cell lung cancer cells

Mohammad M. Al-Saneaa Department of Pharmaceutical Chemistry, College of Pharmacy, Jouf University, Sakaka, Saudi ArabiaCorrespondence[email protected]
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Ghada H. Al-Ansaryb Department of Pharmaceutical Chemistry, Pharmacy Program, Batterejee Medical College, Jeddah, Saudi Arabia;c Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Ain Shams University, Cairo, EgyptCorrespondence[email protected]
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Zainab M. Elsayedd Scientific Research and Innovation Support Unit, Faculty of Pharmacy, Kafrelsheikh University, Kafrelsheikh, EgyptView further author information
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Raed M. Maklade Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Kafrelsheikh University, Kafrelsheikh, Egypt;f Institute of Drug Discovery and Development, Kafrelsheikh University, Kafrelsheikh, EgyptView further author information
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Eslam B. Elkaeedg Department of Pharmaceutical Sciences, College of Pharmacy, AlMaarefa University, Ad Diriyah, Riyadh, Saudi Arabia;h Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy (Boys), Al-Azhar University, Nasr City, Cairo, EgyptView further author information
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Mohamed A. Abdelgawada Department of Pharmaceutical Chemistry, College of Pharmacy, Jouf University, Sakaka, Saudi Arabia;i Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Beni-Suef University, Beni-Suef, EgyptView further author information
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Syed Nasir Abbas Bukharia Department of Pharmaceutical Chemistry, College of Pharmacy, Jouf University, Sakaka, Saudi ArabiaView further author information
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Marwa M. Abdel-Azizj The Regional Center for Mycology & Biotechnology, Al-Azhar University, Cairo, EgyptView further author information
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Howayda Sulimank Department of Medical Biochemistry, Faculty of Medicine, Alexandria University, Alexandria, EgyptView further author information
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Wagdy M. Eldehnae Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Kafrelsheikh University, Kafrelsheikh, EgyptCorrespondence[email protected]
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Pages 987-999 | Received 28 Feb 2021, Accepted 06 Apr 2021, Published online: 13 May 2021

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Jayashree V. Patil, Shweta Umar, Rina Soni, Shubhangi S. Soman & Suresh Balakrishnan. (2023) Design, synthesis and anticancer activity of amide derivatives of substituted 3-methyl-benzofuran-2-carboxylic acid. Synthetic Communications 53:3, pages 217-233.
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Heba S. A. Elzahabi, Eman S. Nossier, Rania A. Alasfoury, May El-Manawaty, Sara M. Sayed, Eslam B. Elkaeed, Ahmed M. Metwaly, Mohamed Hagras & Ibrahim H. Eissa. (2022) Design, synthesis, and anti-cancer evaluation of new pyrido[2,3-d]pyrimidin-4(3H)-one derivatives as potential EGFRWT and EGFRT790M inhibitors and apoptosis inducers. Journal of Enzyme Inhibition and Medicinal Chemistry 37:1, pages 1053-1076.
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Longjia Yan, Qin Wang, Li Liu & Yi Le. (2022) Design, synthesis and biological evaluation of a series of dianilinopyrimidines as EGFR inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry 37:1, pages 832-843.
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Mohamed Hagras, Marwa A. Saleh, Rogy R. Ezz Eldin, Abdelrahman A. Abuelkhir, Emad Gamil Khidr, Ahmed A. El-Husseiny, Hesham A. El-Mahdy, Eslam B. Elkaeed & Ibrahim H. Eissa. (2022) 1,3,4-Oxadiazole-naphthalene hybrids as potential VEGFR-2 inhibitors: design, synthesis, antiproliferative activity, apoptotic effect, and in silico studies. Journal of Enzyme Inhibition and Medicinal Chemistry 37:1, pages 386-402.
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Mohammed M. Alanazi, Alaa Elwan, Nawaf A. Alsaif, Ahmad J. Obaidullah, Hamad M. Alkahtani, Abdulrahman A. Al-Mehizia, Sultan M. Alsubaie, Mohammed S. Taghour & Ibrahim H. Eissa. (2021) Discovery of new 3-methylquinoxalines as potential anti-cancer agents and apoptosis inducers targeting VEGFR-2: design, synthesis, and in silico studies. Journal of Enzyme Inhibition and Medicinal Chemistry 36:1, pages 1732-1750.
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