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Review

Pharmacogenetics of tyrosine kinase inhibitors in gastrointestinal stromal tumor and chronic myeloid leukemia

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Pages 733-742 | Received 05 Mar 2016, Accepted 27 Apr 2016, Published online: 17 May 2016

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Xuehui Jiang, Qun Fu, Yan Jing, Ying Kong, Hong Liu, Hongwei Peng, Kaisaner Rexiti & Xiaohua Wei. (2023) Personalized Dose of Adjuvant Imatinib in Patients with Gastrointestinal Stromal Tumors: Results from a Population Pharmacokinetic Analysis. Drug Design, Development and Therapy 17, pages 809-820.
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Maddalena Centanni, Abel Thijs, Ingrid Desar, Mats O. Karlsson & Lena E. Friberg. (2022) Optimization of blood pressure measurement practices for pharmacodynamic analyses of tyrosine‐kinase inhibitors. Clinical and Translational Science 16:1, pages 73-84.
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Yan Li, Baohui Yang & Xingwang Zhang. (2019) Oral delivery of imatinib through galactosylated polymeric nanoparticles to explore the contribution of a saccharide ligand to absorption. International Journal of Pharmaceutics 568, pages 118508.
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Gloria Ravegnini, Giulia Sammarini, César Serrano, Margherita Nannini, Maria A. Pantaleo, Patrizia Hrelia & Sabrina Angelini. (2019) Clinical relevance of circulating molecules in cancer: focus on gastrointestinal stromal tumors. Therapeutic Advances in Medical Oncology 11, pages 175883591983190.
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Margherita Nannini & Guido Biasco. 2019. Oncogenomics. Oncogenomics 329 337 .
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H-B Qiu, W Zhuang, T Wu, S Xin, C-Z Lin, H-L Ruan, X Zhu, M Huang, J-L Li, X-Y Hou, Z-W Zhou & X-D Wang. (2017) Imatinib-induced ophthalmological side-effects in GIST patients are associated with the variations of EGFR, SLC22A1, SLC22A5 and ABCB1. The Pharmacogenomics Journal 18:3, pages 460-466.
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Michiel C. Verboom, Jacqueline S.L. Kloth, Jesse J. Swen, Tahar van der Straaten, Judith V.M.G. Bovée, Stefan Sleijfer, Anna K.L. Reyners, Ron H.J. Mathijssen, Henk-Jan Guchelaar, Neeltje Steeghs & Hans Gelderblom. (2017) Genetic polymorphisms in angiogenesis-related genes are associated with worse progression-free survival of patients with advanced gastrointestinal stromal tumours treated with imatinib. European Journal of Cancer 86, pages 226-232.
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Zhi-Ping Jiang, Xie-Lan Zhao, Naoto Takahashi, Sabrina Angelini, Biswajit Dubashi, Li Sun & Ping Xu. (2017) Trough concentration and ABCG2 polymorphism are better to predict imatinib response in chronic myeloid leukemia: a meta-analysis . Pharmacogenomics 18:1, pages 35-56.
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