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Original

ASSESSING PREGNANCY RISKS OF AZOLE ANTIFUNGALS USING A HIGH THROUGHPUT AROMATASE INHIBITION ASSAY

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Pages 129-140 | Published online: 07 Jul 2009

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Mukesh C. Gohel & Stavan A. Nagori. (2009) Fabrication and design of transdermal fluconazole spray. Pharmaceutical Development and Technology 14:2, pages 208-215.
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Eva R. Trösken, Karoline Scholz, Roman W. Lutz, Wolfgang Völkel, Jürg A. Zarn & Werner K. Lutz. (2004) Comparative Assessment of the Inhibition of Recombinant Human CYP19 (Aromatase) by Azoles Used in Agriculture and as Drugs for Humans. Endocrine Research 30:3, pages 387-394.
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Laura Kragie. (2002) AROMATASE IN PRIMATE PREGNANCY: A REVIEW. Endocrine Research 28:3, pages 121-128.
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Monica Kam Draskau & Terje Svingen. (2022) Azole Fungicides and Their Endocrine Disrupting Properties: Perspectives on Sex Hormone-Dependent Reproductive Development. Frontiers in Toxicology 4.
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E P Garvey, A D Sharp, P A Warn, C M Yates & R J Schotzinger. (2018) The novel fungal CYP51 inhibitor VT-1598 is efficacious alone and in combination with liposomal amphotericin B in a murine model of cryptococcal meningitis. Journal of Antimicrobial Chemotherapy 73:10, pages 2815-2822.
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Carly A. Elston & Dirk M. Elston. (2013) Treatment of common skin infections and infestations during pregnancy. Dermatologic Therapy 26:4, pages 312-320.
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Christa E. Flück & Amit V. Pandey. 2013. Genetic Steroid Disorders. Genetic Steroid Disorders 125 143 .
Christa E. Flück, Primus E. Mullis & Amit V. Pandey. (2010) Reduction in hepatic drug metabolizing CYP3A4 activities caused by P450 oxidoreductase mutations identified in patients with disordered steroid metabolism. Biochemical and Biophysical Research Communications 401:1, pages 149-153.
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Catherine Nicolo, Christa E. Flück, Primus E. Mullis & Amit V. Pandey. (2010) Restoration of mutant cytochrome P450 reductase activity by external flavin. Molecular and Cellular Endocrinology 321:2, pages 245-252.
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Nehama Linder, Mandola Amarilla, Adriana Hernandez, Tsippy Tamiri, Lea Sirota, Gil Klinger, Itzhak Levy & Paul Merlob. (2009) Association of high‐dose bifonazole administration during early pregnancy and severe limb reduction defects in the newborn. Birth Defects Research Part A: Clinical and Molecular Teratology 88:3, pages 201-204.
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N.W. Jacobsen, B. Halling-Sørensen & F.K. Birkved. (2008) Inhibition of human aromatase complex (CYP19) by antiepileptic drugs. Toxicology in Vitro 22:1, pages 146-153.
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Nga Ta & Thomas Walle. (2007) Aromatase inhibition by bioavailable methylated flavones. The Journal of Steroid Biochemistry and Molecular Biology 107:1-2, pages 127-129.
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Eva R. Trösken, Kathrin Fischer, Wolfgang Völkel & Werner K. Lutz. (2006) Inhibition of human CYP19 by azoles used as antifungal agents and aromatase inhibitors, using a new LC–MS/MS method for the analysis of estradiol product formation. Toxicology 219:1-3, pages 33-40.
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