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Christos Kontogiorgis, Anastasia Detsi & Dimitra Hadjipavlou-Litina. (2012) Coumarin-based drugs: a patent review (2008 – present). Expert Opinion on Therapeutic Patents 22:4, pages 437-454.
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Donald Poirier. (2010) 17β-Hydroxysteroid dehydrogenase inhibitors: a patent review. Expert Opinion on Therapeutic Patents 20:9, pages 1123-1145.
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Marie Bérubé & Donald Poirier. (2007) Chemical synthesis and in vitro biological evaluation of a phosphorylated bisubstrate inhibitor of type 3 17β-hydroxysteroid dehydrogenase. Journal of Enzyme Inhibition and Medicinal Chemistry 22:2, pages 201-211.
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Mohamed Sayed Gomaa, Sook Wah Yee, Ceri Elizabeth Milbourne, Maria Chiara Barbera, Claire Simons & Andrea Brancale. (2006) Homology Model of Human Retinoic Acid Metabolising Enzyme Cytochrome P450 26A1 (CYP26A1): Active Site Architecture and Ligand Binding. Journal of Enzyme Inhibition and Medicinal Chemistry 21:4, pages 361-369.
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Amarylla Horvath & Andreas Billich. (2005) Steroid sulfatase inhibitors. Expert Opinion on Therapeutic Patents 15:11, pages 1541-1553.
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Marc Angotti, Rolf W. Hartmann, Andrew J. Kirby, Claire Simons, Paul J. Nicholls, Robert D.E. Sewell & H. John Smith. (2005) Effect of 2-(4-aminophenylmethyl)-6-hydroxy-3,4-dihydronaphthalen-1(2H)-one on all-trans and 13-cis-retinoic acid levels in plasma quantified by high perfomance liquid chromatography coupled to tandem mass spectrometry. Journal of Enzyme Inhibition and Medicinal Chemistry 20:3, pages 219-226.
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Martin R. Tremblay, Roch P. Boivin, Van Luu-The & Donald Poirier. (2005) Inhibitors of type 1 17β-hydroxysteroid dehydrogenase with reduced estrogenic activity: Modifications of the positions 3 and 6 of estradiol. Journal of Enzyme Inhibition and Medicinal Chemistry 20:2, pages 153-163.
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Jean-Yves Winum, Andrea Scozzafava, Jean-Louis Montero & Claudiu T Supuran. (2004) Therapeutic applications of sulfamates. Expert Opinion on Therapeutic Patents 14:9, pages 1273-1308.
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Peter Mason, Valerie P. Greer, Andrew J. Kirby, Claire Simons, Paul J. Nicholls & H. John Smith. (2003) Some Aryl Substituted 2-(4-Nitrophenyl)-4-oxo-4-phenylbutanoates and 3-(4-Nitrophenyl)-1-phenyl-1,4-butanediols and Related Compounds as Inhibitors of Rat Liver Microsomal Retinoic Acid Metabolising Enzymes. Journal of Enzyme Inhibition and Medicinal Chemistry 18:6, pages 511-528.
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V.P. Greer, P. Mason, A.J. Kirby, H.J. Smith, P.J. Nicholls & C. Simons. (2003) Some 1,2-Diphenylethane Derivatives as Inhibitors of Retinoic Acid—Metabolising Enzymes. Journal of Enzyme Inhibition and Medicinal Chemistry 18:5, pages 431-443.
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Peter Nussbaumer & Andreas Billich. (2003) Steroid sulfatase inhibitors. Expert Opinion on Therapeutic Patents 13:5, pages 605-625.
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Tai K. Vinh, Paul J. Nicholls, Andrew J. Kirby & Claire Simons. (2001) Evaluation of 7-Hydroxy-Flavones as Inhibitors of Oestrone and Oestradiol Biosynthesis. Journal of Enzyme Inhibition 16:5, pages 417-424.
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Jack Silver, Golzar Al-Jaff, Michael T. Wilson, Daniel den Engelsen, George R. Fern & Terry G. Ireland. (2022) Studies on the binding of nitrogenous bases to protoporphyrin IX iron(II) in aqueous solution at high pH values. JBIC Journal of Biological Inorganic Chemistry 27:3, pages 297-313.
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Nourhène Chouchène, Amani Toumi, Sarra Boudriga, Hayet Edziri, Mansour Sobeh, Mohamed A. O. Abdelfattah, Moheddine Askri, Michael Knorr, Carsten Strohmann, Lukas Brieger & Armand Soldera. (2022) Antimicrobial Activity and DFT Studies of a Novel Set of Spiropyrrolidines Tethered with Thiochroman-4-one/Chroman-4-one Scaffolds. Molecules 27:3, pages 582.
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Donald Poirier, Jenny Roy & René Maltais. (2021) A Targeted-Covalent Inhibitor of 17β-HSD1 Blocks Two Estrogen-Biosynthesis Pathways: In Vitro (Metabolism) and In Vivo (Xenograft) Studies in T-47D Breast Cancer Models. Cancers 13:8, pages 1841.
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Nguyen Hoang Anh, Nguyen Phuoc Long, Sun Jo Kim, Jung Eun Min, Sang Jun Yoon, Hyung Min Kim, Eugine Yang, Eun Sook Hwang, Jeong Hill Park, Soon-Sun Hong & Sung Won Kwon. (2019) Steroidomics for the Prevention, Assessment, and Management of Cancers: A Systematic Review and Functional Analysis. Metabolites 9:10, pages 199.
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Sui-Qun Yang, Xiao-Ming Li, Xin Li, Lu-Ping Chi & Bin-Gui Wang. (2018) Two New Diketomorpholine Derivatives and a New Highly Conjugated Ergostane-Type Steroid from the Marine Algal-Derived Endophytic Fungus Aspergillus alabamensis EN-547. Marine Drugs 16:4, pages 114.
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Étienne Ouellet, René Maltais, Charles Ouellet & Donald Poirier. (2013) Investigation of a tetrahydroisoquinoline scaffold as dual-action steroid sulfatase inhibitors generated by parallel solid-phase synthesis. MedChemComm 4:4, pages 681.
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Rebecca M. Maksymowicz, Philippe M. C. Roth, Amber L. Thompson & Stephen P. Fletcher. (2013) Hydrometallation-asymmetric conjugate addition: application to complex molecule synthesis. Chem. Commun. 49:39, pages 4211-4213.
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Evgenija A. Djurendić, Marina P. Savić, Olivera R. Klisurić, Marija N. Sakač, Gordana M. Bogdanović, Dimitar S. Jakimov & Katarina M. Penov Gaši. (2012) Synthesis, X-ray structural analysis, and cytotoxic activity of some new androstane d-homo lactone derivatives. Structural Chemistry 23:6, pages 1761-1767.
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René Maltais & Donald Poirier. (2011) Steroid sulfatase inhibitors: A review covering the promising 2000–2010 decade. Steroids 76:10-11, pages 929-948.
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Donald Poirier. (2011) Contribution to the development of inhibitors of 17β-hydroxysteroid dehydrogenase types 1 and 7: Key tools for studying and treating estrogen-dependent diseases. The Journal of Steroid Biochemistry and Molecular Biology 125:1-2, pages 83-94.
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Mohamed S. GomaaCaroline E. BridgensAhmed S. AboraiaGareth J. VealChristopher P. F. RedfernAndrea BrancaleJane L. ArmstrongClaire Simons. (2011) Small Molecule Inhibitors of Retinoic Acid 4-Hydroxylase (CYP26): Synthesis and Biological Evaluation of Imidazole Methyl 3-(4-(aryl-2-ylamino)phenyl)propanoates. Journal of Medicinal Chemistry 54:8, pages 2778-2791.
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Siham Farhane, Michelle-Audrey Fournier, René Maltais & Donald Poirier. (2011) Convergent stereoselective and efficient synthesis of furanic-steroid derivatives. Tetrahedron 67:13, pages 2434-2440.
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Marie Bérubé, Florian Delagoutte & Donald Poirier. (2010) Preparation of 16β-Estradiol Derivative Libraries as Bisubstrate Inhibitors of 17β-Hydroxysteroid Dehydrogenase Type 1 Using the Multidetachable Sulfamate Linker. Molecules 15:3, pages 1590-1631.
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Shinya Harusawa, Chihiro Kojima, Kensuke Fujii, Yuusaku Yamashita, Tomoya Tanaka, Lisa Araki, Toshinobu Yoshimura, Minoru Sakaguchi, Yoshihide Usami & Masanori Takaoka. (2010) Synthesis of Two Estradiol-Imidazole C-Ribonucleoside Hybrid Compounds Exhibiting Inhibitory Effects against Type 1 17β-Hydroxysteroid Dehydrogenase. HETEROCYCLES 81:12, pages 2817.
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René Maltais, Diane Fournier & Donald Poirier. (2009) Quantitative Structure-Activity Relationship (QSAR) Study with a Series of 17α-Derivatives of Estradiol: Model for the Development of Reversible Steroid Sulfatase Inhibitors. QSAR & Combinatorial Science 28:11-12, pages 1284-1299.
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Annamaria Lilienkampf, Sampo Karkola, Sari Alho-Richmond, Pasi Koskimies, Nina Johansson, Kaisa Huhtinen, Kimmo Vihko & Kristiina Wähälä. (2009)
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Michelle-Audrey Fournier & Donald Poirier. (2009) Estrogen formation in endometrial and cervix cancer cell lines: Involvement of aromatase, steroid sulfatase and 17β-hydroxysteroid dehydrogenases (types 1, 5, 7 and 12). Molecular and Cellular Endocrinology 301:1-2, pages 142-145.
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Mohamed Sayed Gomaa, Jane L. Armstrong, Beatrice Bobillon, Gareth J. Veal, Andrea Brancale, Christopher P.F. Redfern & Claire Simons. (2008) Novel azolyl-(phenylmethyl)]aryl/heteroarylamines: Potent CYP26 inhibitors and enhancers of all-trans retinoic acid activity in neuroblastoma cells. Bioorganic & Medicinal Chemistry 16:17, pages 8301-8313.
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Liviu C. Ciobanu & Donald Poirier. (2006) Synthesis of Libraries of 16β‐Aminopropyl Estradiol Derivatives for Targeting Two Key Steroidogenic Enzymes. ChemMedChem 1:11, pages 1249-1259.
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Stephane Pautus, Sook Wah Yee, Martyn Jayne, Michael P. Coogan & Claire Simons. (2006) Synthesis and CYP26A1 inhibitory activity of 1-[benzofuran-2-yl-(4-alkyl/aryl-phenyl)-methyl]-1H-triazoles. Bioorganic & Medicinal Chemistry 14:11, pages 3643-3653.
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Jean‐Yves Winum, Andrea Scozzafava, Jean‐Louis Montero & Claudiu T. Supuran. (2004) Sulfamates and their therapeutic potential. Medicinal Research Reviews 25:2, pages 186-228.
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Paul M. Wood, L.W. Lawrence Woo, Anna Humphreys, Surinder K. Chander, Atul Purohit, Michael J. Reed & Barry V.L. Potter. (2005) A letrozole-based dual aromatase–sulphatase inhibitor with in vivo activity. The Journal of Steroid Biochemistry and Molecular Biology 94:1-3, pages 123-130.
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Samir Yahiaoui, Christelle Pouget, Catherine Fagnere, Yves Champavier, Gérard Habrioux & Albert José Chulia. (2004) Synthesis and evaluation of 4-triazolylflavans as new aromatase inhibitors. Bioorganic & Medicinal Chemistry Letters 14:20, pages 5215-5218.
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