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Eric T Whalley, Carlos D Figueroa, Lajos Gera & Kanti D Bhoola. (2012) Discovery and therapeutic potential of kinin receptor antagonists. Expert Opinion on Drug Discovery 7:12, pages 1129-1148.
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Éva Bozó, János Éles & György M Keserű. (2012) Bradykinin B1 receptor antagonists: a patent update 2009 – 2012. Expert Opinion on Therapeutic Patents 22:12, pages 1443-1452.
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Christopher I Fincham, Alessandro Bressan, Marielle Paris, Cristina Rossi & Daniela Fattori. (2009) Bradykinin receptor antagonists – a review of the patent literature 2005 – 2008. Expert Opinion on Therapeutic Patents 19:7, pages 919-941.
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Articles from other publishers (12)
Juan J. Perez. (2021) Exploiting Knowledge on Structure–Activity Relationships for Designing Peptidomimetics of Endogenous Peptides. Biomedicines 9:6, pages 651.
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Gerasimos Rassias, Sofia Leonardi, Dionisia Rigopoulou, Eleanna Vachlioti, Konstantinos Afratis, Zoi Piperigkou, Christos Koutsakis, Nikos K. Karamanos, Haralambos Gavras & Dionissios Papaioannou. (2021) Potent antiproliferative activity of bradykinin B2 receptor selective agonist FR-190997 and analogue structures thereof: A paradox resolved?. European Journal of Medicinal Chemistry 210, pages 112948.
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B. Rasaeifar, C.S. Lupala, P. Gomez-Gutierrez & Juan J. Perez. (2019) Molecular features characterizing non-peptide selectivity to the human B1 and B2 bradykinin receptors. Bioorganic & Medicinal Chemistry Letters 29:1, pages 11-14.
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Cecylia S. Lupala, Patricia Gomez-Gutierrez & Juan J. Perez. (2015) New insights into the stereochemical requirements of the bradykinin B2 receptor antagonists binding. Journal of Computer-Aided Molecular Design 30:1, pages 85-101.
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S Meini, F Bellucci, C Catalani, P Cucchi, A Giolitti, S Giuliani, L Quartara, L Rotondaro, S Zappitelli & CA Maggi. (2011) Comparison of the molecular interactions of two antagonists, MEN16132 or icatibant, at the human kinin B2 receptor. British Journal of Pharmacology 162:5, pages 1202-1212.
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Yoo Lim Kam, Hee-Kyung Rhee, Hwa-Jung Kim, Seung Keun Back, Heung Sik Na & Hea-Young Park Choo. (2010) Synthesis and bradykinin inhibitory activity of novel non-peptide compounds, and evaluation of in vivo analgesic activity. Bioorganic & Medicinal Chemistry 18:6, pages 2327-2336.
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Christoph Gibson, Karsten Schnatbaum, Jochen R. Pfeifer, Elsa Locardi, Matthias Paschke, Ulf Reimer, Uwe Richter, Dirk Scharn, Alexander Faussner & Thomas Tradler. (2009)
Novel Small Molecule Bradykinin B
2
Receptor Antagonists
. Journal of Medicinal Chemistry 52:14, pages 4370-4379.
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Scott D. Kuduk, Ronald K. Chang, Robert M. DiPardo, Christina N. Di Marco, Kathy L. Murphy, Richard W. Ransom, Duane R. Reiss, Cuyue Tang, Thomayant Prueksaritanont, Douglas J. Pettibone & Mark G. Bock. (2008) Bradykinin B1 receptor antagonists: An α-hydroxy amide with an improved metabolism profile. Bioorganic & Medicinal Chemistry Letters 18:18, pages 5107-5110.
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Dong-Mei Feng, Robert M. DiPardo, Jenny M. Wai, Ronald K. Chang, Christina N. Di Marco, Kathy L. Murphy, Richard W. Ransom, Duane R. Reiss, Cuyue Tang, Thomayant Prueksaritanont, Douglas J. Pettibone, Mark G. Bock & Scott D. Kuduk. (2008) A new class of bradykinin B1 receptor antagonists with high oral bioavailability and minimal PXR activity. Bioorganic & Medicinal Chemistry Letters 18:2, pages 682-687.
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Scott D. Kuduk, Robert M. DiPardo, Ronald K. Chang, Christina N. Di Marco, Kathy L. Murphy, Richard W. Ransom, Duane R. Reiss, Cuyue Tang, Thomayant Prueksaritanont, Douglas J. Pettibone & Mark G. Bock. (2007) Bradykinin B1 antagonists: Biphenyl SAR studies in the cyclopropanecarboxamide series. Bioorganic & Medicinal Chemistry Letters 17:13, pages 3608-3612.
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Daniela Fattori, Cristina Rossi, Christopher I. Fincham, Marco Berettoni, Federico Calvani, Fernando Catrambone, Patrizia Felicetti, Martina Gensini, Rosa Terracciano, Maria Altamura, Alessandro Bressan, Sandro Giuliani, Carlo A. Maggi, Stefania Meini, Claudio Valenti & Laura Quartara. (2006)
Design and Synthesis of Novel Sulfonamide-Containing Bradykinin hB
2
Receptor Antagonists. 1. Synthesis and SAR of α,α-Dimethylglycine Sulfonamides
. Journal of Medicinal Chemistry 49:12, pages 3602-3613.
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Guillaume Morissette, Johanne Bouthillier & François Marceau. (2006) Dual antagonists of the bradykinin B1 and B2 receptors based on a postulated common pharmacophore from existing non-peptide antagonists. Biological Chemistry 387:2.
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