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Patent Review

Quinazoline derivatives as anticancer drugs: a patent review (2011 – present)

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Kamal Tabti, Larbi Elmchichi, Abdelouahid Sbai, Hamid Maghat, Mohammed Bouachrine & Tahar Lakhlifi. (2022) Molecular modelling of antiproliferative inhibitors based on SMILES descriptors using Monte-Carlo method, docking, MD simulations and ADME/Tox studies. Molecular Simulation 48:17, pages 1575-1591.
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Shazia Parveen, Mohamad Hagar, Rua B. Alnoman, Hoda A. Ahmed, El Sayed H. El Ashry & Mohamed A. Zakaria. (2022) Synthesis, Docking and Density Functional Theory Approaches on 1,3-Bis-3-(4-Chlorophenyl)-2,3-Dihydroquinazolin-4(1H)-on-2-Thioxopropane toward the Discovery of Dual Kinase Inhibitor. Polycyclic Aromatic Compounds 42:6, pages 3736-3747.
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Parveen Kumar, Vijesh Tomar, Raj Kumar Joshi & Meena Nemiwal. (2022) Nanocatalyzed synthetic approach for quinazoline and quinazolinone derivatives: A review (2015–present). Synthetic Communications 52:6, pages 795-826.
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Ibrahim M. Z. Fares, Ahmed E. M. Mekky, Ahmed H. M. Elwahy & Ismail A. Abdelhamid. (2020) Microwave-assisted three component synthesis of novel bis-fused quinazolin-8(4H)-ones linked to aliphatic or aromatic spacer via amide linkages. Synthetic Communications 50:6, pages 893-903.
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Yaling Zhang, Li Chen, Xiabing Li, Li Gao, Yunxia Hao, Baolin Li & Yaping Yan. (2019) Novel 4-arylaminoquinazolines bearing N,N-diethyl(aminoethyl)amino moiety with antitumour activity as EGFRwt-TK inhibitor. Journal of Enzyme Inhibition and Medicinal Chemistry 34:1, pages 1668-1677.
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You-Guang Zheng, Xiao-Qing Wu, Jun Su, Ping Jiang, Liang Xu, Jian Gao, Bin Cai & Min Ji. (2017) Design and synthesis of a novel photoaffinity probe for labelling EGF receptor tyrosine kinases. Journal of Enzyme Inhibition and Medicinal Chemistry 32:1, pages 954-959.
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Wafa Mohamed Al Madhagi. 2024. Recent Advances on Quinazoline [Working Title]. Recent Advances on Quinazoline [Working Title].
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