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Devendra S. Puntambekar, Rajani Giridhar & Mange Ram Yadav. (2007) Inhibition of farnesyltransferase: A rational approach to treat cancer?. Journal of Enzyme Inhibition and Medicinal Chemistry 22:2, pages 127-140.
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Peter Norman. (2003) Merck & Co., Inc.: analysis of patenting 1998 – 2002. Expert Opinion on Therapeutic Patents 13:7, pages 1037-1044.
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Ian M Bell. (2000) Inhibitors of protein prenylation 2000. Expert Opinion on Therapeutic Patents 10:12, pages 1813-1831.
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Articles from other publishers (17)
Laurence Goossens, Sophie Deweer, Jean Pommery, Jean-Pierre Hénichart & Jean-François Goossens. (2005) Spectroscopic study of fluorescent peptides for prenyl transferase assays. Journal of Pharmaceutical and Biomedical Analysis 37:3, pages 417-422.
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Ian M. Bell. (2004) Inhibitors of Farnesyltransferase: A Rational Approach to Cancer Chemotherapy?. Journal of Medicinal Chemistry 47:8, pages 1869-1878.
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Katja Kettler, Jacek Sakowski, Katrin Silber, Isabel Sattler, Gerhard Klebe & Martin Schlitzer. (2003) Non-thiol farnesyltransferase inhibitors: n -(4-acylamino-3-benzoylphenyl)-3-[5-(4-nitrophenyl)-2-furyl]acrylic acid amides. Bioorganic & Medicinal Chemistry 11:7, pages 1521-1530.
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Andreas Mitsch, Markus Böhm, Pia Wißner, Isabel Sattler & Martin Schlitzer. (2002) Non-Thiol farnesyltransferase inhibitors: utilization of an aryl binding site by 5-arylacryloylaminobenzophenones. Bioorganic & Medicinal Chemistry 10:8, pages 2657-2662.
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Ian M. Bell, Steven N. Gallicchio, Marc Abrams, Lorena S. Beese, Douglas C. Beshore, Hema Bhimnathwala, Michael J. Bogusky, Carolyn A. Buser, J. Christopher Culberson, Joseph Davide, Michelle Ellis-Hutchings, Christine Fernandes, Jackson B. Gibbs, Samuel L. Graham, Kelly A. Hamilton, George D. Hartman, David C. Heimbrook, Carl F. Homnick, Hans E. Huber, Joel R. Huff, Kelem Kassahun, Kenneth S. Koblan, Nancy E. Kohl, Robert B. Lobell, Joseph J. Lynch,, Ronald Robinson, A. David Rodrigues, Jeffrey S. Taylor, Eileen S. Walsh, Theresa M. Williams & C. Blair Zartman. (2002) 3-Aminopyrrolidinone Farnesyltransferase Inhibitors: Design of Macrocyclic Compounds with Improved Pharmacokinetics and Excellent Cell Potency. Journal of Medicinal Chemistry 45:12, pages 2388-2409.
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Martin Schlitzer, Markus Böhm & Isabel Sattler. (2002) Non-thiol farnesyltransferase inhibitors: structure–activity relationships of benzophenone-based bisubstrate analogue farnesyltransferase inhibitors. Bioorganic & Medicinal Chemistry 10:3, pages 615-620.
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Jacek Sakowski, Isabel Sattler & Martin Schlitzer. (2002) Non-thiol Farnesyltransferase Inhibitors: N-(4-Acylamino-3-benzoylphenyl)-4-nitrocinnamic Acid Amides. Bioorganic & Medicinal Chemistry 10:2, pages 233-239.
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Raymond Houssin, Jean Pommery, Marie-Catherine Salaün, Sophie Deweer, Jean-François Goossens, Philippe Chavatte & Jean-Pierre Hénichart. (2001) Design, Synthesis, and Pharmacological Evaluation of New Farnesyl Protein Transferase Inhibitors. Journal of Medicinal Chemistry 45:2, pages 533-536.
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Douglas C Beshore, Ian M Bell, Christopher J Dinsmore, Carl F Homnick, J.Christopher Culberson, Ronald G Robinson, Christine Fernandes, Eileen S Walsh, Marc T Abrams, Hema G Bhimnathwala, Joseph P Davide, Michelle S Ellis-Hutchings, Hans A Huber, Kenneth S Koblan, Carolyn A Buser, Nancy E Kohl, Robert B Lobell, I-Wu Chen, Debra A McLoughlin, Timothy V Olah, Samuel L Graham, George D Hartman & Theresa M Williams. (2001) Evaluation of amino acid-based linkers in potent macrocyclic inhibitors of farnesyl-protein transferase. Bioorganic & Medicinal Chemistry Letters 11:14, pages 1817-1821.
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Christopher J Dinsmore, Jeffrey M Bergman, Donna D Wei, C.Blair Zartman, Joseph P Davide, Ian B Greenberg, Dongming Liu, Timothy J O'Neill, Jackson B Gibbs, Kenneth S Koblan, Nancy E Kohl, Robert B Lobell, I-Wu Chen, Debra A McLoughlin, Timothy V Olah, Samuel L Graham, George D Hartman & Theresa M Williams. (2001) Oxo-piperazine Derivatives of N-Arylpiperazinones as Inhibitors of Farnesyltransferase. Bioorganic & Medicinal Chemistry Letters 11:4, pages 537-540.
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Martin Schlitzer, Ann Winter-Vann & Patrick J Casey. (2001) Non-peptidic, non-prenylic inhibitors of the prenyl protein-specific protease Rce1. Bioorganic & Medicinal Chemistry Letters 11:3, pages 425-427.
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Andreas Mitsch, Pia Wißner, Isabel Sattler & Martin Schlitzer. (2001) Non-Thiol Farnesyltransferase Inhibitors: Structure-Activity Relationships of Aralkylsubsituted Benzophenones. Archiv der Pharmazie 334:2, pages 40-44.
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H
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Seung-Ho Lee, Hyun-Mi Kang, Ho-Chul Song, Heesoon Lee, Un Chul Lee, Kwang-Hee Son, Sung-Hoon Kim & Byoung-Mog Kwon. (2000) Sesquiterpene Lactones, Inhibitors of Farnesyl Protein Transferase, Isolated from the Flower of Artemisia sylvatica. Tetrahedron 56:27, pages 4711-4715.
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Jackson B. Gibbs. (2000) Mechanism-Based Target Identification and Drug Discovery in Cancer Research. Science 287:5460, pages 1969-1973.
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Charles Z Ding, John T Hunt, Carol Ricca & Veeraswamy Manne. (2000) 3-Imidazolylmethylaminophenylsulfonyltetrahydroquinolines, a novel series of farnesyltransferase inhibitors. Bioorganic & Medicinal Chemistry Letters 10:3, pages 273-275.
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