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Drug Evaluations

Entinostat for treatment of solid tumors and hematologic malignancies

, MD & , MD
Pages 1455-1467 | Published online: 02 Sep 2011

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Ma Su, Xingyu Gong & Feng Liu. (2021) An update on the emerging approaches for histone deacetylase (HDAC) inhibitor drug discovery and future perspectives. Expert Opinion on Drug Discovery 16:7, pages 745-761.
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Kristin C. Hicks, Massimo Fantini, Renee N. Donahue, Angie Schwab, Karin M. Knudson, Sarah R. Tritsch, Caroline Jochems, Paul E. Clavijo, Clint T. Allen, James W. Hodge, Kwong Y. Tsang, Jeffrey Schlom & Sofia R. Gameiro. (2018) Epigenetic priming of both tumor and NK cells augments antibody-dependent cellular cytotoxicity elicited by the anti-PD-L1 antibody avelumab against multiple carcinoma cell types. OncoImmunology 7:11.
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Hai-Tao Qin, Huan-Qiu Li & Feng Liu. (2017) Selective histone deacetylase small molecule inhibitors: recent progress and perspectives. Expert Opinion on Therapeutic Patents 27:5, pages 621-636.
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Rossana Ruiz, Luis E Raez & Christian Rolfo. (2015) Entinostat (SNDX-275) for the treatment of non-small cell lung cancer. Expert Opinion on Investigational Drugs 24:8, pages 1101-1109.
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Geneviève P Delcuve, Dilshad H Khan & James R Davie. (2013) Targeting class I histone deacetylases in cancer therapy. Expert Opinion on Therapeutic Targets 17:1, pages 29-41.
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Léa Madegard, Melissa Girard, Benjamin Riss Yaw, Karine Porte, Davide Audisio, Sébastien Papot & Frédéric Taran. (2023) Bioorthogonal Drug Release from Nanometric Micelles in Living Cells. Chemistry – A European Journal 29:43.
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