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Small-molecule EGFR tyrosine kinase inhibitors for the treatment of cancer

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Jie Qian, Xueyan Zhang, Bo Zhang, Bo Yan, Lin Wang, Ping Gu, Weimin Wang, Huimin Wang & Baohui Han. (2020) Tyrosine Kinase Inhibitor-Related Hepatotoxicity in Patients with Advanced Lung Adenocarcinoma: A Real-World Retrospective Study. Cancer Management and Research 12, pages 3293-3299.
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Mu-Chun Li, Mohane Selvaraj Coumar, Shu-Yu Lin, Yih-Shyan Lin, Guan-Lin Huang, Chun-Hwa Chen, Tzu-Wen Lien, Yi-Wen Wu, Yen-Ting Chen, Ching-Ping Chen, Yu-Chen Huang, Kai-Chia Yeh, Chen-Ming Yang, Bikashita Kalita, Shiow-Lin Pan, Tsu-An Hsu, Teng-Kuang Yeh, Chiung-Tong Chen & Hsing-Pang Hsieh. (2023) Development of Furanopyrimidine-Based Orally Active Third-Generation EGFR Inhibitors for the Treatment of Non-Small Cell Lung Cancer. Journal of Medicinal Chemistry 66:4, pages 2566-2588.
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Rudradip Das, Gayatri Tambe & Amit Shard. (2023) Sulfonamides as tyrosine kinase modulators – A promising class of anticancer agents. Results in Chemistry 5, pages 100950.
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Xuejian Wang, Wenyan Jiang, Yanmei Du, Dongqi Zhu, Jian Zhang, Chunyan Fang, Fang Yan & Zhe-Sheng Chen. (2022) Targeting feedback activation of signaling transduction pathways to overcome drug resistance in cancer. Drug Resistance Updates 65, pages 100884.
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Christos Kiritsis, Antonio Shegani, Konstantina Makrypidi, Ioanna Roupa, Aristotelis Lazopoulos, Angeliki Panagiotopoulou, Sotiria Triantopoulou, Maria Paravatou-Petsotas, Hans-Jürgen Pietzsch, Maria Pelecanou, Minas Papadopoulos & Ioannis Pirmettis. (2022) Synthesis and preclinical evaluation of rhenium and technetium-99m “4 + 1” mixed-ligand complexes bearing quinazoline derivatives as potential EGFR imaging agents. Bioorganic & Medicinal Chemistry 73, pages 117012.
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Xue Liu, Xin Liu, Mikhail I. Kusaykin, Miansong Zhang, Xinfeng Bai, Tingting Cui, Yaping Shi, Changheng Liu & Airong Jia. (2022) Structural characterization of a P-selectin and EGFR dual-targeting fucoidan from Sargassum fusiforme. International Journal of Biological Macromolecules 199, pages 86-95.
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子繁 王. (2022) Study on First-Generation TKIs in the Treatment of Patients with Unresectable EGFR-Mutation-Positive Non-Small-Cell Lung Cancer. Advances in Clinical Medicine 12:02, pages 761-770.
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Yu-Li Lo, Hua-Ching Lin, Shu-Ting Hong, Chih-Hsien Chang, Chen-Shen Wang & Anya Maan-Yuh Lin. (2021) Lipid polymeric nanoparticles modified with tight junction-modulating peptides promote afatinib delivery across a blood–brain barrier model. Cancer Nanotechnology 12:1.
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Qizhang Li, Zhiying Wang, Qiang Zheng & Sen Liu. (2020) Potential clinical drugs as covalent inhibitors of the priming proteases of the spike protein of SARS-CoV-2. Computational and Structural Biotechnology Journal 18, pages 2200-2208.
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