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Drug Evaluations

A review of erlotinib – an oral, selective epidermal growth factor receptor tyrosine kinase inhibitor

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Pages 311-320 | Published online: 21 Jan 2010

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Jianying Dong, Arlene Sereno, Dikran Aivazian, Emma Langley, Brian R. Miller, William B Snyder, Eric Chan, Matt Cantele, Ronald Morena, Ingrid B.J.K. Joseph, Antonio Boccia, Cyrus Virata, James Gamez, Grace Yco, Michael Favis, Xiufeng Wu, Christilyn P. Graff, Qin Wang, Ellen Rohde, Rachel Rennard, Lisa Berquist, Flora Huang, Ying Zhang, Sharon X. Gao, Steffan N. Ho, Stephen J. Demarest, Mitchell E. Reff, Kandasamy Hariharan & Scott M. Glaser. (2011) A stable IgG-like bispecific antibody targeting the epidermal growth factor receptor and the type I insulin-like growth factor receptor demonstrates superior anti-tumor activity. mAbs 3:3, pages 273-288.
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Djoeke de Wit, Henk-Jan Guchelaar, Jan den Hartigh, Hans Gelderblom & Nielka P. van Erp. (2015) Individualized dosing of tyrosine kinase inhibitors: are we there yet?. Drug Discovery Today 20:1, pages 18-36.
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Yin-dong Song, Ke-fei Zhang, Dong Liu, Yan-qi Guo, Da-yong Wang, Ming-yu Cui, Gang Li, Yuan-xin Sun, Jian-hui Shen, Xin-gang Li, Long Zhang & Feng-jun Shi. (2014) Inhibition of EGFR-induced glucose metabolism sensitizes chondrosarcoma cells to cisplatin. Tumor Biology 35:7, pages 7017-7024.
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Joseph P. Garay & Joe W. Gray. (2012) Omics and therapy - A basis for precision medicine. Molecular Oncology 6:2, pages 128-139.
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Lisa Nolan Wright, Andrew Ryscavage, Glenn Merlino & Stuart H. Yuspa. (2012) Modeling the Transcriptional Consequences of Epidermal Growth Factor Receptor Ablation in Ras-Initiated Squamous Cancer. Clinical Cancer Research 18:1, pages 170-183.
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Ioannis N Melas, Alexander Mitsos, Dimitris E Messinis, Thomas S Weiss & Leonidas G Alexopoulos. (2011) Combined logical and data-driven models for linking signalling pathways to cellular response. BMC Systems Biology 5:1.
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Craig D. Woodworth, Laura P. Diefendorf, David F. Jette, Abdulmajid Mohammed, Michael A. Moses, Sylvia A. Searleman, Dan A. Stevens, Katelynn M. Wilton & Sumona Mondal. (2011) Inhibition of the epidermal growth factor receptor by erlotinib prevents immortalization of human cervical cells by Human Papillomavirus type 16. Virology 421:1, pages 19-27.
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Gregory E Holt, Eckhard R Podack & Luis E Raez. (2011) Immunotherapy as a strategy for the treatment of non-small-cell lung cancer. Therapy 8:1, pages 43-54.
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