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Drug Evaluations

Fasiglifam as a new potential treatment option for patients with type 2 diabetes

, MD
Pages 2591-2600 | Published online: 06 Nov 2013

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Billy J. Molloy, Adam King, Lee A. Gethings, Robert S. Plumb, Russell J. Mortishire-Smith & Ian D. Wilson. (2023) Investigation of the pharmacokinetics and metabolic fate of Fasiglifam (TAK-875) in male and female rats following oral and intravenous administration. Xenobiotica 53:2, pages 93-105.
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Akifumi Kogame, Ronald Lee, Liping Pan, Miyako Sudo, Masami Nonaka, Yuu Moriya, Tomoaki Higuchi & Yoshihiko Tagawa. (2019) Disposition and metabolism of the G protein-coupled receptor 40 agonist TAK-875 (fasiglifam) in rats, dogs, and humans. Xenobiotica 49:4, pages 433-445.
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André J. Scheen. (2016) Investigational insulin secretagogues for type 2 diabetes. Expert Opinion on Investigational Drugs 25:4, pages 405-422.
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