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Review

Solid lipid microparticles: formulation, preparation, characterisation, drug release and applications

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Pages 75-87 | Published online: 22 Apr 2005

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Giada Botti, Anna Bianchi, Alessandro Dalpiaz, Paola Tedeschi, Valentina Albanese, Milena Sorrenti, Laura Catenacci, Maria Cristina Bonferoni, Sarah Beggiato & Barbara Pavan. (2023) Dimeric ferulic acid conjugate as a prodrug for brain targeting after nasal administration of loaded solid lipid microparticles. Expert Opinion on Drug Delivery 0:0, pages 1-23.
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Hongyi Ouyang, Soon Jun Ang, Zong Yang Lee, Tze Ning Hiew, Paul Wan Sia Heng & Lai Wah Chan. (2022) Effect of drug load and lipid–wax blends on drug release and stability from spray-congealed microparticles. Pharmaceutical Development and Technology 27:10, pages 1069-1082.
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Maie S. Tawfik, Khaled A. Abdel-Ghaffar, Ahmed Y. Gamal, Fatma H. El-Demerdash & Heba A. Gad. (2019) Lycopene solid lipid microparticles with enhanced effect on gingival crevicular fluid protein carbonyl as a biomarker of oxidative stress in patients with chronic periodontitis. Journal of Liposome Research 29:4, pages 375-382.
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Padmini Ravikumar, Mahesh Katariya, Sushil Patil, Pratima Tatke & Raviraj Pillai. (2019) Skin delivery of resveratrol encapsulated lipidic formulation for melanoma chemoprevention. Journal of Microencapsulation 36:6, pages 535-551.
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Jingying Liu, Philip C. Christophersen, Mingshi Yang, Hanne M. Nielsen & Huiling Mu. (2017) The impact of particle preparation methods and polymorphic stability of lipid excipients on protein distribution in microparticles. Drug Development and Industrial Pharmacy 43:12, pages 2032-2042.
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Isabella Martignoni, Valentina Trotta, Wing-Hin Lee, Ching-Yee Loo, Michele Pozzoli, Paul M. Young, Santo Scalia & Daniela Traini. (2016) Resveratrol solid lipid microparticles as dry powder formulation for nasal delivery, characterization and in vitro deposition study. Journal of Microencapsulation 33:8, pages 735-742.
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Chinazom Agbo, Chukwuebuka Umeyor, Franklin Kenechukwu, John Ogbonna, Salome Chime, Charles Lovelyn, Obumneme Agubata, Kenneth Ofokansi & Anthony Attama. (2016) Formulation design, in vitro characterizations and anti-malarial investigations of artemether and lumefantrine-entrapped solid lipid microparticles. Drug Development and Industrial Pharmacy 42:10, pages 1708-1721.
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Franklin C. Kenechukwu, Mumuni A. Momoh, Petra O. Nnamani & Anthony A. Attama. (2015) Solid lipid micro-dispersions (SLMs) based on PEGylated solidified reverse micellar solutions (SRMS): a novel carrier system for gentamicin. Drug Delivery 22:6, pages 710-722.
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Ikechukwu V. Onyishi, Salome A. Chime & Echezona O. Ogudiegwu. (2015) Formulation of novel sustained release rifampicin-loaded solid lipid microparticles based on structured lipid matrices from Moringa oleifera. Pharmaceutical Development and Technology 20:5, pages 546-554.
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E. E. Chinaeke, S. A. Chime, V. I. Onyishi, A. A. Attama & V. C. Okore. (2015) Formulation development and evaluation of the anti-malaria properties of sustained release artesunate-loaded solid lipid microparticles based on phytolipids. Drug Delivery 22:5, pages 652-665.
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Santo Scalia, Paul M Young & Daniela Traini. (2015) Solid lipid microparticles as an approach to drug delivery. Expert Opinion on Drug Delivery 12:4, pages 583-599.
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Eric E. Chinaeke, Salome A. Chime, John D. N. Ogbonna, Anthony A. Attama, C. C. Müller-Goymann & Vincent C. Okore. (2014) Evaluation of dika wax-soybean oil-based artesunate-loaded lipospheres: in vitro–in vivo correlation studies. Journal of Microencapsulation 31:8, pages 796-804.
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Valentina Trotta, Filipa Goios, Helena Monteiro, Isabel F. Almeida & Santo Scalia. (2014) Influence of lipid microparticle encapsulation on in vitro efficacy, photostability and water resistance of the sunscreen agents, octyl methoxycinnamate and butyl methoxydibenzoylmethane. Drug Development and Industrial Pharmacy 40:9, pages 1233-1239.
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Salome Amarachi Chime, Ikechukwu V. Onyishi, Paschal U. Ugwoke & Anthony A. Attama. (2014) Evaluation of the Properties of Gongronema latifolium in Phospholipon 90H Based Solid Lipid Microparticles (SLMs): An Antidiabetic Study. Journal of Dietary Supplements 11:1, pages 7-18.
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Kenneth Chibuzor Ofokansi, Franklin Chimaobi Kenechukwu & A.B. Isah. (2013) Poloxamer-Stabilized Topical Miconazole Nitrate-Loaded Microemulsion: Formulation Design and Characterization. Journal of Dispersion Science and Technology 34:11, pages 1563-1574.
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Moayad Alhariri, Ali Azghani & Abdelwahab Omri. (2013) Liposomal antibiotics for the treatment of infectious diseases. Expert Opinion on Drug Delivery 10:11, pages 1515-1532.
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Salome Amarachi Chime, Anthony Amaechi Attama, Philip F. Builders & Godswill C. Onunkwo. (2013) Sustained-release diclofenac potassium-loaded solid lipid microparticle based on solidified reverse micellar solution: in vitro and in vivo evaluation. Journal of Microencapsulation 30:4, pages 335-345.
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Santo Scalia, Daniela Traini, Paul M. Young, Marcello Di Sabatino, Nadia Passerini & Beatrice Albertini. (2013) Comparison of spray congealing and melt emulsification methods for the incorporation of the water-soluble salbutamol sulphate in lipid microparticles. Pharmaceutical Development and Technology 18:1, pages 266-273.
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Emmanuel Chukwuebuka Umeyor, Franklin Chimaobi Kenechukwu, John Dike Ogbonna, Salome Amarachi Chime & Anthony Attama. (2012) Preparation of novel solid lipid microparticles loaded with gentamicin and its evaluation in vitro and in vivo. Journal of Microencapsulation 29:3, pages 296-307.
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Santo Scalia, Rania Salama, Paul Young & Daniela Traini. (2012) Preparation and in vitro evaluation of salbutamol-loaded lipid microparticles for sustained release pulmonary therapy. Journal of Microencapsulation 29:3, pages 225-233.
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Luigi Battaglia & Marina Gallarate. (2012) Lipid nanoparticles: state of the art, new preparation methods and challenges in drug delivery. Expert Opinion on Drug Delivery 9:5, pages 497-508.
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Yahya Rahimpour & Hamed Hamishehkar. (2012) Liposomes in cosmeceutics. Expert Opinion on Drug Delivery 9:4, pages 443-455.
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Y. A. Gomaa, I. A. Darwish, N. A. Boraei & L. K. El-Khordagui. (2010) Formulation of wax oxybenzone microparticles using a factorial approach. Journal of Microencapsulation 27:7, pages 628-639.
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Santo Scalia & Matteo Mezzena. (2009) Co-loading of a Photostabilizer with the Sunscreen Agent, Butyl Methoxydibenzoylmethane in Solid Lipid Microparticles. Drug Development and Industrial Pharmacy 35:2, pages 192-198.
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Amal H. El-Kamel, Iman M. Al-Fagih & Ibrahim A. Alsarra. (2007) Testosterone solid lipid microparticles for transdermal drug delivery. Formulation and physicochemical characterization. Journal of Microencapsulation 24:5, pages 457-475.
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