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Polymorphisms of the drug transporters ABCB1, ABCG2, ABCC2 and ABCC3 and their impact on drug bioavailability and clinical relevance

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Tsvetelin Lukanov, Milena Ivanova, Petya Yankova, Bushra Al Hadra, Anastasiya Mihaylova, Marianka Genova, Dobrin Svinarov & Elisaveta Naumova. (2022) Impact of CYP3A7, CYP2D6 and ABCC2/ABCC3 polymorphisms on tacrolimus steady state concentrations in Bulgarian kidney transplant recipients. Biotechnology & Biotechnological Equipment 36:1, pages 362-369.
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Tamara Božina, Lana Ganoci, Ena Karačić, Livija Šimičević, Majda Vrkić-Kirhmajer, Iva Klarica-Domjanović, Tena Križ, Zrinka Sertić & Nada Božina. (2022) ABCG2 and SLCO1B1 gene polymorphisms in the Croatian population. Annals of Human Biology 49:7-8, pages 323-331.
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Henrike Bruckmueller & Ingolf Cascorbi. (2021) ABCB1, ABCG2, ABCC1, ABCC2, and ABCC3 drug transporter polymorphisms and their impact on drug bioavailability: what is our current understanding?. Expert Opinion on Drug Metabolism & Toxicology 17:4, pages 369-396.
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Ingolf Cascorbi & Anneke Nina Werk. (2017) Advances and challenges in hereditary cancer pharmacogenetics. Expert Opinion on Drug Metabolism & Toxicology 13:1, pages 73-82.
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David E. Amacher. (2016) The regulation of human hepatic drug transporter expression by activation of xenobiotic-sensing nuclear receptors. Expert Opinion on Drug Metabolism & Toxicology 12:12, pages 1463-1477.
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Elena Arrigoni, Sara Galimberti, Mario Petrini, Romano Danesi & Antonello Di Paolo. (2016) ATP-binding cassette transmembrane transporters and their epigenetic control in cancer: an overview. Expert Opinion on Drug Metabolism & Toxicology 12:12, pages 1419-1432.
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Anne Mahringer & Gert Fricker. (2016) ABC transporters at the blood–brain barrier. Expert Opinion on Drug Metabolism & Toxicology 12:5, pages 499-508.
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Seok Hwee Koo, Ying Li Lo, Jie Yin Yee & Edmund Jon Deoon Lee. (2015) Genetic and/or non-genetic causes for inter-individual and inter-cellular variability in transporter protein expression: implications for understanding drug efficacy and toxicity. Expert Opinion on Drug Metabolism & Toxicology 11:12, pages 1821-1837.
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Iben Kümler, Jan Stenvang, José Moreira, Nils Brünner & Dorte Lisbet Nielsen. (2015) Drug transporters in breast cancer: response to anthracyclines and taxanes. Expert Review of Anticancer Therapy 15:9, pages 1075-1092.
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